메뉴 건너뛰기




Volumn 28, Issue 4, 1998, Pages 322-338

Studies of the biogenic amine transporters. VII. Characterization of a novel cocaine binding site identified with [125I]RTI-55 in membranes prepared from human, monkey and guinea pig caudate

Author keywords

Benztropine; Bupropion; Cocaine; Dopamine; GBR12909; GBR12935; Mazindol; Nomifensine; Transmitter uptake inhibitors neuronal

Indexed keywords

3BETA (4 IODOPHENYL) 2BETA TROPANECARBOXYLIC ACID METHYL ESTER; DOPAMINE TRANSPORTER; IODINE 125; SEROTONIN TRANSPORTER;

EID: 6844236997     PISSN: 08874476     EISSN: None     Source Type: Journal    
DOI: 10.1002/(SICI)1098-2396(199804)28:4<322::AID-SYN8>3.0.CO;2-B     Document Type: Article
Times cited : (28)

References (92)
  • 1
    • 0026614687 scopus 로고
    • 3H]Cocaine labels a binding site associated with the serotonin transporter in guinea pig brain: Allosteric modulation by paroxetine
    • 3H]Cocaine labels a binding site associated with the serotonin transporter in guinea pig brain: Allosteric modulation by paroxetine. Neurochem. Res., 17:1275-1283.
    • (1992) Neurochem. Res. , vol.17 , pp. 1275-1283
    • Akunne, H.C.1    De Costa, B.R.2    Jacobson, A.E.3    Rice, K.C.4    Rothman, R.B.5
  • 3
    • 0025923591 scopus 로고
    • 3H]1-[1-(2-thienyl)cyclohexyl]piperidine labels two high affinity binding sites in human cortex: Further evidence for phencyclidine binding sites associated with the biogenic amine reuptake complex
    • 3H]1-[1-(2-thienyl)cyclohexyl]piperidine labels two high affinity binding sites in human cortex: Further evidence for phencyclidine binding sites associated with the biogenic amine reuptake complex. Synapse, 8:289-300.
    • (1991) Synapse , vol.8 , pp. 289-300
    • Akunne, H.C.1    Reid, A.A.2    Thurkauf, A.3    Jacobson, A.E.4    De Costa, B.R.5    Rice, K.C.6    Heyes, M.P.7    Rothman, R.B.8
  • 4
    • 0025269813 scopus 로고
    • Drug abuse, psychiatric disorders, and AIDS. Dual and triple diagnosis
    • Batki, S.L. (1990) Drug abuse, psychiatric disorders, and AIDS. Dual and triple diagnosis. West. J. Med., 152:547-552.
    • (1990) West. J. Med. , vol.152 , pp. 547-552
    • Batki, S.L.1
  • 5
    • 0027497491 scopus 로고
    • Clinical pharmacology and toxicology of cocaine
    • erratum 72(6):343
    • Benowitz, N.L. (1993) Clinical pharmacology and toxicology of cocaine. Pharmacol. Toxicol., 72:3-12; (erratum 72(6):343).
    • (1993) Pharmacol. Toxicol. , vol.72 , pp. 3-12
    • Benowitz, N.L.1
  • 6
    • 0024585705 scopus 로고
    • Treatment of cocaine abuse with mazindol
    • Berger, P., Gawin, F., and Kosten, T.R. (1989) Treatment of cocaine abuse with mazindol (letter). Lancet, 1:283.
    • (1989) Lancet , vol.1 , pp. 283
    • Berger, P.1    Gawin, F.2    Kosten, T.R.3
  • 7
    • 0024460030 scopus 로고
    • Effects of cocaine and related drugs in nonhuman primates. III. Self-administration by squirrel monkeys
    • Bergman, J., Madras, B.K., Johnson, S.E., and Spealman, R.D. (1989) Effects of cocaine and related drugs in nonhuman primates. III. Self-administration by squirrel monkeys. J. Pharmacol. Exp. Ther., 251:150-155.
    • (1989) J. Pharmacol. Exp. Ther. , vol.251 , pp. 150-155
    • Bergman, J.1    Madras, B.K.2    Johnson, S.E.3    Spealman, R.D.4
  • 8
    • 0024268972 scopus 로고
    • Effect of methimazole-induced hypothyroidism on multiple opioid receptors in rat brain regions
    • Bhargava, H.N., Ramarao, P., and Gulati, A. (1988) Effect of methimazole-induced hypothyroidism on multiple opioid receptors in rat brain regions. Pharmacology, 37:356-364.
    • (1988) Pharmacology , vol.37 , pp. 356-364
    • Bhargava, H.N.1    Ramarao, P.2    Gulati, A.3
  • 10
    • 0026507640 scopus 로고
    • Expression of a single dopamine transporter cDNA can confer two cocaine binding sites
    • Boja, J.W., Markham, L., Patel, A., Uhl, G., and Kuhar, M.J. (1992a) Expression of a single dopamine transporter cDNA can confer two cocaine binding sites. Neuroscience/NeuroReport, 3: 247-248.
    • (1992) Neuroscience/NeuroReport , vol.3 , pp. 247-248
    • Boja, J.W.1    Markham, L.2    Patel, A.3    Uhl, G.4    Kuhar, M.J.5
  • 12
    • 0028901757 scopus 로고
    • Selective labeling of the dopamine transporter by the high affinity ligand 3 beta-(4-[125I]iodophenyl)tropane-2 beta-carboxylic acid isopropyl ester
    • Boja, J.W., Cadet, J.L., Kopajtic, T.A., Lever, J., Seltzman, H.H., Wyrick, C.D., Lewin, A.H., Abraham, P., and Carroll, F.I. (1995) Selective labeling of the dopamine transporter by the high affinity ligand 3 beta-(4-[125I]iodophenyl)tropane-2 beta-carboxylic acid isopropyl ester. Mol. Pharmacol., 47:779-786.
    • (1995) Mol. Pharmacol. , vol.47 , pp. 779-786
    • Boja, J.W.1    Cadet, J.L.2    Kopajtic, T.A.3    Lever, J.4    Seltzman, H.H.5    Wyrick, C.D.6    Lewin, A.H.7    Abraham, P.8    Carroll, F.I.9
  • 14
    • 0026009418 scopus 로고
    • Synthesis, ligand binding, QSAR, and CoMFA study of 3β-(p-substituted phenyl)tropane-2β-carboxylic acid methyl esters
    • Carroll, F.I., Gao, Y.G., Rahman, M.A., Abraham, P., Parham, K., Lewin, A.H., Boja, J.W., and Kuhar, M.J. (1991) Synthesis, ligand binding, QSAR, and CoMFA study of 3β-(p-substituted phenyl)tropane-2β-carboxylic acid methyl esters. J. Med. Chem., 34:2719-2727.
    • (1991) J. Med. Chem. , vol.34 , pp. 2719-2727
    • Carroll, F.I.1    Gao, Y.G.2    Rahman, M.A.3    Abraham, P.4    Parham, K.5    Lewin, A.H.6    Boja, J.W.7    Kuhar, M.J.8
  • 15
    • 0026647629 scopus 로고
    • Isopropyl and phenyl esters of 3β-(4-substituted phenyl)tropan-2β-carboxylic acids. Potent and selective compounds for the dopamine transporter
    • Carroll, F.I., Abraham, P., Lewin, A.H., Parham, K.A., Boja, J.W., and Kuhar, M.J. (1992) Isopropyl and phenyl esters of 3β-(4-substituted phenyl)tropan-2β-carboxylic acids. Potent and selective compounds for the dopamine transporter. J. Med. Chem., 35:2497-2500.
    • (1992) J. Med. Chem. , vol.35 , pp. 2497-2500
    • Carroll, F.I.1    Abraham, P.2    Lewin, A.H.3    Parham, K.A.4    Boja, J.W.5    Kuhar, M.J.6
  • 16
    • 0022311917 scopus 로고
    • Pharmacological approaches to cocaine addiction
    • Dackis, C.A., and Gold, M.S. (1985) Pharmacological approaches to cocaine addiction. J. Subst. Abuse Treat., 2:139-145.
    • (1985) J. Subst. Abuse Treat. , vol.2 , pp. 139-145
    • Dackis, C.A.1    Gold, M.S.2
  • 17
  • 19
    • 0027253985 scopus 로고
    • Cocaine abuse in North America: A milestone in history
    • Das, G. (1993a) Cocaine abuse in North America: A milestone in history. J. Clin. Pharmacol., 33:296-310.
    • (1993) J. Clin. Pharmacol. , vol.33 , pp. 296-310
    • Das, G.1
  • 20
  • 22
    • 0343933624 scopus 로고
    • Drugs abused by humans preferentially increase synaptic dopamine concentrations in the mesolimbic system of freely moving rats
    • Di Chiara, G., and Imperato, A. (1988) Drugs abused by humans preferentially increase synaptic dopamine concentrations in the mesolimbic system of freely moving rats. Proc. Natl. Acad. Sci. USA, 85:5274-5278.
    • (1988) Proc. Natl. Acad. Sci. USA , vol.85 , pp. 5274-5278
    • Di Chiara, G.1    Imperato, A.2
  • 23
    • 0025562551 scopus 로고
    • Mazindol treatment of cocaine abuse. A double-blind investigation
    • Diakogiannis, I.A., Steinberg, M., and Kosten, T.R. (1991) Mazindol treatment of cocaine abuse. A double-blind investigation. NIDA Res. Monogr., 105:514.
    • (1991) NIDA Res. Monogr. , vol.105 , pp. 514
    • Diakogiannis, I.A.1    Steinberg, M.2    Kosten, T.R.3
  • 25
    • 0022591327 scopus 로고
    • Abstinence symptomatology and psychiatric diagnosis in cocaine abusers
    • Gawin, F.H., and Kleber, H.D. (1986) Abstinence symptomatology and psychiatric diagnosis in cocaine abusers. Arch. Gen. Psychiatry, 43:107-113.
    • (1986) Arch. Gen. Psychiatry , vol.43 , pp. 107-113
    • Gawin, F.H.1    Kleber, H.D.2
  • 26
    • 84907120346 scopus 로고
    • Cocaine abuse treated with phenelzine
    • Golwyn, D.H. (1988) Cocaine abuse treated with phenelzine. Int. J. Addict., 23:897-905.
    • (1988) Int. J. Addict. , vol.23 , pp. 897-905
    • Golwyn, D.H.1
  • 28
    • 0023864222 scopus 로고
    • A versatile method for simultaneous analysis of families of curves
    • Guardabasso, V., Munson, P.J., and Rodbard, D. (1988) A versatile method for simultaneous analysis of families of curves. FASEB J., 2:209-215.
    • (1988) FASEB J. , vol.2 , pp. 209-215
    • Guardabasso, V.1    Munson, P.J.2    Rodbard, D.3
  • 29
    • 0027759664 scopus 로고
    • Further studies of the structure-activity relationships of 1-[1-(2-benzo[b]thienyl)cyclohexyl]piperidine. Synthesis and evaluation of 1-(2-benzo[b]thienyl)-N,N-dialkylcyclohexylamines at dopamine uptake and phencyclidine binding sites
    • He, X., Raymon, L.P., Mattson, M.V., Eldefrawi, M.E., and de Costa, B.R. (1993a) Further studies of the structure-activity relationships of 1-[1-(2-benzo[b]thienyl)cyclohexyl]piperidine. Synthesis and evaluation of 1-(2-benzo[b]thienyl)-N,N-dialkylcyclohexylamines at dopamine uptake and phencyclidine binding sites. J. Med. Chem., 36:4075-4081.
    • (1993) J. Med. Chem. , vol.36 , pp. 4075-4081
    • He, X.1    Raymon, L.P.2    Mattson, M.V.3    Eldefrawi, M.E.4    De Costa, B.R.5
  • 30
    • 0027196727 scopus 로고
    • Synthesis and biological evaluation of 1-[1-(2-benzo[b]thienyl)cyclohexyl]piperidine homologues at dopamineuptake and phencyclidine- and sigma-binding sites
    • He, X.S., Raymon, L.P., Mattson, M.V., Eldefrawi, M.E., and de Costa, B.R. (1993b) Synthesis and biological evaluation of 1-[1-(2-benzo[b]thienyl)cyclohexyl]piperidine homologues at dopamineuptake and phencyclidine- and sigma-binding sites. J. Med. Chem., 36:1188-1193.
    • (1993) J. Med. Chem. , vol.36 , pp. 1188-1193
    • He, X.S.1    Raymon, L.P.2    Mattson, M.V.3    Eldefrawi, M.E.4    De Costa, B.R.5
  • 31
    • 0020416931 scopus 로고
    • Citalopram - Pharmacological profile of a specific serotonin uptake inhibitor with antidepressant activity
    • Hyttel, J. (1982) Citalopram - pharmacological profile of a specific serotonin uptake inhibitor with antidepressant activity. Prog. Neuropsychopharmacol. Biol. Psychiat., 6:277-295.
    • (1982) Prog. Neuropsychopharmacol. Biol. Psychiat. , vol.6 , pp. 277-295
    • Hyttel, J.1
  • 32
    • 0021843333 scopus 로고
    • Neurochemical profile of LU 19-005. A potent inhibitor of uptake of dopamine, noradrenaline and serotonin
    • Hyttel, J., and Larsen, J.J. (1985) Neurochemical profile of LU 19-005. A potent inhibitor of uptake of dopamine, noradrenaline and serotonin. J. Neurochem., 44:1615-1620.
    • (1985) J. Neurochem. , vol.44 , pp. 1615-1620
    • Hyttel, J.1    Larsen, J.J.2
  • 33
    • 0026470770 scopus 로고
    • Neuroreceptor imaging with SPECT
    • Innis, R.B. (1992) Neuroreceptor imaging with SPECT. J. Clin. Psychiat., 53(11):29-34.
    • (1992) J. Clin. Psychiat. , vol.53 , Issue.11 , pp. 29-34
    • Innis, R.B.1
  • 34
    • 0021287012 scopus 로고
    • 3H]mazindol binding associated with neuronal dopamine and norepinephrine uptake sites
    • 3H]mazindol binding associated with neuronal dopamine and norepinephrine uptake sites. Mol. Pharmacol., 26:35-44.
    • (1984) Mol. Pharmacol. , vol.26 , pp. 35-44
    • Javitch, J.A.1    Blaustein, R.O.2    Snyder, S.H.3
  • 36
    • 0024268361 scopus 로고
    • Differential diagnosis of psychiatric comorbidity in substance abusers
    • Kosten, T.R., and Kleber, H.D. (1988) Differential diagnosis of psychiatric comorbidity in substance abusers. J. Subst. Abuse Treat., 5:201-206.
    • (1988) J. Subst. Abuse Treat. , vol.5 , pp. 201-206
    • Kosten, T.R.1    Kleber, H.D.2
  • 37
    • 0023973764 scopus 로고
    • Bromocriptine treatment of cocaine abuse in patients maintained on methadone
    • Kosten, T.R., Schumann, B., and Wright, D. (1988) Bromocriptine treatment of cocaine abuse in patients maintained on methadone [letter]. Am. J. Psych., 145:381-382.
    • (1988) Am. J. Psych. , vol.145 , pp. 381-382
    • Kosten, T.R.1    Schumann, B.2    Wright, D.3
  • 38
    • 0026564117 scopus 로고
    • Pharmacotherapy for cocaine-abusing methadone-maintained patients using amantadine or desipramine
    • Kosten, T.R., Morgan, C.M., Falcione, J., and Schottenfeld, R.S. (1992) Pharmacotherapy for cocaine-abusing methadone-maintained patients using amantadine or desipramine. Arch. Gen. Psychiatry, 49:894-898.
    • (1992) Arch. Gen. Psychiatry , vol.49 , pp. 894-898
    • Kosten, T.R.1    Morgan, C.M.2    Falcione, J.3    Schottenfeld, R.S.4
  • 39
    • 0025855256 scopus 로고
    • The dopamine hypothesis of the reinforcing properties of cocaine
    • Kuhar, M.J., Ritz, M.C., and Boja, J.W. (1991) The dopamine hypothesis of the reinforcing properties of cocaine. Trends. Neurosci., 14:299-302.
    • (1991) Trends. Neurosci. , vol.14 , pp. 299-302
    • Kuhar, M.J.1    Ritz, M.C.2    Boja, J.W.3
  • 40
    • 84907125024 scopus 로고
    • Depression as an antecedent of frequency of intravenous drug use in an urban, nontreatment sample
    • Latkin, C.A., and Mandell, W. (1993) Depression as an antecedent of frequency of intravenous drug use in an urban, nontreatment sample. Int. J. Addict., 28:1601-1612.
    • (1993) Int. J. Addict. , vol.28 , pp. 1601-1612
    • Latkin, C.A.1    Mandell, W.2
  • 42
    • 0027472644 scopus 로고
    • A rat brain cDNA encoding a neurotransmitter trnasporter with an unusual structure
    • Liu, Q.-R., Mandiyan, S., Lopez-Corcuera, B., Nelson, H., and Nelson, N. (1993) A rat brain cDNA encoding a neurotransmitter trnasporter with an unusual structure. FEBS Lett., 315:114-118.
    • (1993) FEBS Lett. , vol.315 , pp. 114-118
    • Liu, Q.-R.1    Mandiyan, S.2    Lopez-Corcuera, B.3    Nelson, H.4    Nelson, N.5
  • 46
    • 0025549806 scopus 로고
    • An open pilot study of bupropion and psychotherapy for the treatment of cocaine abuse in methadone-maintained patients
    • Margolin, A., Kosten, T., Petrakis, I., and Avants, S.K. (1991) An open pilot study of bupropion and psychotherapy for the treatment of cocaine abuse in methadone-maintained patients. NIDA Res. Monogr., 105:367-368.
    • (1991) NIDA Res. Monogr. , vol.105 , pp. 367-368
    • Margolin, A.1    Kosten, T.2    Petrakis, I.3    Avants, S.K.4
  • 47
    • 0026582712 scopus 로고
    • Prevalence of cocaine use among residents of New York City who committed suicide during a one-year period
    • Marzuk, P.M., Tardiff, K., Leon, A.C., Stajic, M., Morgan, E.B., and Mann, J.J. (1992) Prevalence of cocaine use among residents of New York City who committed suicide during a one-year period. Am. J. Psychiatry, 149:371-375.
    • (1992) Am. J. Psychiatry , vol.149 , pp. 371-375
    • Marzuk, P.M.1    Tardiff, K.2    Leon, A.C.3    Stajic, M.4    Morgan, E.B.5    Mann, J.J.6
  • 49
  • 50
    • 0023029035 scopus 로고
    • A quantitative method of analyzing the interaction of slightly selective radioligands with multiple receptor subtypes
    • McGonigle, P., Neve, K.A., and Molinoff, P.B. (1986)A quantitative method of analyzing the interaction of slightly selective radioligands with multiple receptor subtypes. Mol. Pharmacol., 30:329-337.
    • (1986) Mol. Pharmacol. , vol.30 , pp. 329-337
    • McGonigle, P.1    Neve, K.A.2    Molinoff, P.B.3
  • 51
    • 21844489841 scopus 로고
    • Prevalence and treatment models for addiction in psychiatric populations
    • Miller, N.S. (1994) Prevalence and treatment models for addiction in psychiatric populations. Psychiatr. Ann., 24:399-406.
    • (1994) Psychiatr. Ann. , vol.24 , pp. 399-406
    • Miller, N.S.1
  • 52
    • 0006730463 scopus 로고
    • Safety and efficacy of bupropion in combination with bromocriptine for treatment of cocaine dependence
    • Montoya, I.D., Preston, K.L., Cone, E.J., Rothman, R.B., and Gorelick, D.A. (1995) Safety and efficacy of bupropion in combination with bromocriptine for treatment of cocaine dependence. NIDA Res. Monogr. 153:304.
    • (1995) NIDA Res. Monogr. , vol.153 , pp. 304
    • Montoya, I.D.1    Preston, K.L.2    Cone, E.J.3    Rothman, R.B.4    Gorelick, D.A.5
  • 53
    • 0026493343 scopus 로고
    • Cocaine's history, especially the American experience
    • Musto, D.F. (1992) Cocaine's history, especially the American experience. Ciba Foundation Symposium, 166:7-14.
    • (1992) Ciba Foundation Symposium , vol.166 , pp. 7-14
    • Musto, D.F.1
  • 54
    • 0023740509 scopus 로고
    • Extracellular cocaine and dopamine concentrations are linearly related in rat striatum
    • Nicolaysen, L.C., Pan, H.T., and Justice, J.B. Jr. (1988) Extracellular cocaine and dopamine concentrations are linearly related in rat striatum. Brain Res., 456:317-323.
    • (1988) Brain Res. , vol.456 , pp. 317-323
    • Nicolaysen, L.C.1    Pan, H.T.2    Justice Jr., J.B.3
  • 55
    • 6844221232 scopus 로고
    • Effect of dopamine receptor antagonists on cocaine-induced subjective effects: A naturalistic case study
    • Ohuoha, D.C., Maxwell, J.W., Cadet, J.L., and Rothman, R.B. (1994) Effect of dopamine receptor antagonists on cocaine-induced subjective effects: A naturalistic case study. NIDA Res. Monogr., 141:442.
    • (1994) NIDA Res. Monogr. , vol.141 , pp. 442
    • Ohuoha, D.C.1    Maxwell, J.W.2    Cadet, J.L.3    Rothman, R.B.4
  • 56
    • 0023086656 scopus 로고
    • Neuropharmacology of cocaine: Role of monoaminergic systems
    • Pitts, D.K., and Marwah, J. (1987) Neuropharmacology of cocaine: Role of monoaminergic systems. Monogr. Neural Sci., 13:34-54.
    • (1987) Monogr. Neural Sci. , vol.13 , pp. 34-54
    • Pitts, D.K.1    Marwah, J.2
  • 57
    • 0016641108 scopus 로고
    • Cocaine psychoses: A continuum model
    • Post, R.M. (1975) Cocaine psychoses: A continuum model. Am. J. Psych., 132:225-231.
    • (1975) Am. J. Psych. , vol.132 , pp. 225-231
    • Post, R.M.1
  • 59
    • 0022438717 scopus 로고
    • Psychological issues in the treatment of cocaine abuse
    • Resnick, R.B., and Resnick, E. (1986) Psychological issues in the treatment of cocaine abuse. NIDA Res. Monogr., 67:290-294.
    • (1986) NIDA Res. Monogr. , vol.67 , pp. 290-294
    • Resnick, R.B.1    Resnick, E.2
  • 60
    • 0023265754 scopus 로고
    • Cocaine receptors on dopamine transporters are related to self-administration of cocaine
    • Ritz, M.C., Lamb, R.J., Goldberg, S.R., and Kuhar, M.J. (1987) Cocaine receptors on dopamine transporters are related to self-administration of cocaine. Science, 237:1219-1223.
    • (1987) Science , vol.237 , pp. 1219-1223
    • Ritz, M.C.1    Lamb, R.J.2    Goldberg, S.R.3    Kuhar, M.J.4
  • 61
    • 0026468751 scopus 로고
    • Molecular mechanisms associated with cocaine effects. Possible relationships with effects of ethanol
    • Ritz, M.C., Kuhar, M.J., and George, F.R. (1992) Molecular mechanisms associated with cocaine effects. Possible relationships with effects of ethanol. Recent Dev. Alcohol., 10:273-302.
    • (1992) Recent Dev. Alcohol. , vol.10 , pp. 273-302
    • Ritz, M.C.1    Kuhar, M.J.2    George, F.R.3
  • 62
    • 0017250843 scopus 로고
    • Statistical characterization of the random errors in the radioimmunoassay dose-response variable
    • Rodbard, D., Lenox, R.H., Wray, H.L., and Ramseth, D. (1976) Statistical characterization of the random errors in the radioimmunoassay dose-response variable. Clin. Chem., 22:350-358.
    • (1976) Clin. Chem. , vol.22 , pp. 350-358
    • Rodbard, D.1    Lenox, R.H.2    Wray, H.L.3    Ramseth, D.4
  • 63
    • 0014157852 scopus 로고
    • Inhibition of the uptake of tritiated catecholamines by anti-depressants and related compounds
    • Ross, S.B., and Renyi, A.L. (1967) Inhibition of the uptake of tritiated catecholamines by anti-depressants and related compounds. Eur. J. Pharmacol., 2:181-186.
    • (1967) Eur. J. Pharmacol. , vol.2 , pp. 181-186
    • Ross, S.B.1    Renyi, A.L.2
  • 64
    • 0021061881 scopus 로고
    • Analysis of binding surfaces: A methodology appropriate for the investigation of complex receptor mechanisms and multiple neurotransmitter receptors
    • Rothman, R.B. (1983) Analysis of binding surfaces: A methodology appropriate for the investigation of complex receptor mechanisms and multiple neurotransmitter receptors. Neuropeptides, 4: 41-44.
    • (1983) Neuropeptides , vol.4 , pp. 41-44
    • Rothman, R.B.1
  • 65
    • 0022297965 scopus 로고
    • Binding surface analysis: An intuitive yet quantitative method for the design and analysis of ligand binding studies
    • Rothman, R.B. (1986) Binding surface analysis: An intuitive yet quantitative method for the design and analysis of ligand binding studies. Alcohol Drug Res., 6:309-325.
    • (1986) Alcohol Drug Res. , vol.6 , pp. 309-325
    • Rothman, R.B.1
  • 66
    • 0029348098 scopus 로고
    • A review of the effects of dopaminergic agents on humans, animals and drug seeking behavior, and its implications for medication development: Focus on GBR12909
    • Rothman, R.B., and Glowa, J.R. (1995) A review of the effects of dopaminergic agents on humans, animals and drug seeking behavior, and its implications for medication development: Focus on GBR12909. Mol. Neurobiol., 11:1-19.
    • (1995) Mol. Neurobiol. , vol.11 , pp. 1-19
    • Rothman, R.B.1    Glowa, J.R.2
  • 68
    • 0025924672 scopus 로고
    • 3H]1,3-Di(2-tolyl)guanidine of two high affinity binding sites in guinea pig brain: Evidence for allosteric regulation by calcium channel antagonists and pseudoallosteric modulation by ¶ ligands
    • 3H]1,3-Di(2-tolyl)guanidine of two high affinity binding sites in guinea pig brain: Evidence for allosteric regulation by calcium channel antagonists and pseudoallosteric modulation by ¶ ligands. Mol. Pharmacol., 39:222-232.
    • (1991) Mol. Pharmacol. , vol.39 , pp. 222-232
    • Rothman, R.B.1    Reid, A.A.2    Mahboubi, A.3    Kim, C.-H.4    De Costa, B.R.5    Jacobson, A.E.6    Rice, K.C.7
  • 69
    • 0027174387 scopus 로고
    • Identification of a GBR12935 homolog, LR1111, which is over 4000-fold selective for the dopamine transporter, relative to serotonin and norepinephrine transporters
    • Rothman, R.B., Lewis, B., Dersch, C.M., Xu, H., Radesca, L., de Costa, B.R., Rice, K.C., Kilburn, R.B., Akunne, H.C., and Pert, A. (1993) Identification of a GBR12935 homolog, LR1111, which is over 4000-fold selective for the dopamine transporter, relative to serotonin and norepinephrine transporters. Synapse, 14:34-39.
    • (1993) Synapse , vol.14 , pp. 34-39
    • Rothman, R.B.1    Lewis, B.2    Dersch, C.M.3    Xu, H.4    Radesca, L.5    De Costa, B.R.6    Rice, K.C.7    Kilburn, R.B.8    Akunne, H.C.9    Pert, A.10
  • 71
    • 0028434555 scopus 로고
    • Combined use of fenfluramine and phentermine in the treatment of cocaine addiction: A pilot case series
    • Rothman, R.B., Gendron, T.M., and Hitzig, P. (1994b) Combined use of fenfluramine and phentermine in the treatment of cocaine addiction: A pilot case series. J. Subst. Abuse Treat., 11:273-275.
    • (1994) J. Subst. Abuse Treat. , vol.11 , pp. 273-275
    • Rothman, R.B.1    Gendron, T.M.2    Hitzig, P.3
  • 74
    • 0025186557 scopus 로고
    • DESIGN: Computerized optimization of experimental design for estimating Kd and Bmax in ligand binding experiments. II. Simultaneous analysis of homologous and heterologous competition curves and analysis blocking and of "multiligand" dose-response surfaces
    • Rovati, G.E., Rodbard, D., and Munson, P.J. (1990) DESIGN: Computerized optimization of experimental design for estimating Kd and Bmax in ligand binding experiments. II. Simultaneous analysis of homologous and heterologous competition curves and analysis blocking and of "multiligand" dose-response surfaces. Anal. Biochem., 184:172-183.
    • (1990) Anal. Biochem. , vol.184 , pp. 172-183
    • Rovati, G.E.1    Rodbard, D.2    Munson, P.J.3
  • 76
    • 0023115464 scopus 로고
    • Metaphit irreversibly inhibits [3H]threo-(+/-)-methylphenidate binding to rat striatal tissue
    • Schweri, M.M., Jacobson, A.E., Lessor, R.A., and Rice, K.C. (1987) Metaphit irreversibly inhibits [3H]threo-(+/-)-methylphenidate binding to rat striatal tissue. J. Neurochem., 48:102-105.
    • (1987) J. Neurochem. , vol.48 , pp. 102-105
    • Schweri, M.M.1    Jacobson, A.E.2    Lessor, R.A.3    Rice, K.C.4
  • 77
    • 0026766934 scopus 로고
    • Fourphit: A selective probe for the methylphenidate binding site on the dopamine transporter
    • Schweri, M.M., Thurkauf, A., Mattson, M.V., and Rice, K.C. (1992) Fourphit: A selective probe for the methylphenidate binding site on the dopamine transporter. J. Pharmacol. Exp. Ther., 261:936-942.
    • (1992) J. Pharmacol. Exp. Ther. , vol.261 , pp. 936-942
    • Schweri, M.M.1    Thurkauf, A.2    Mattson, M.V.3    Rice, K.C.4
  • 78
    • 0023799734 scopus 로고
    • Metaphit prevents locomotor activation induced by various psychostimulants and interferes with the dopaminergic system in mice
    • Sershen, H., Berger, P., Jacobson, A.E., Rice, K.C., and Reith, M.E. (1988) Metaphit prevents locomotor activation induced by various psychostimulants and interferes with the dopaminergic system in mice. Neuropharmacology, 27:23-30.
    • (1988) Neuropharmacology , vol.27 , pp. 23-30
    • Sershen, H.1    Berger, P.2    Jacobson, A.E.3    Rice, K.C.4    Reith, M.E.5
  • 81
    • 0024456087 scopus 로고
    • Effects of cocaine and related drugs in nonhuman primates. II. Stimulant effects on schedule-controlled behavior
    • Spealman, R.D., Madras, B.K., and Bergman, J. (1989) Effects of cocaine and related drugs in nonhuman primates. II. Stimulant effects on schedule-controlled behavior. J. Pharmacol. Exp. Ther., 251:142-149.
    • (1989) J. Pharmacol. Exp. Ther. , vol.251 , pp. 142-149
    • Spealman, R.D.1    Madras, B.K.2    Bergman, J.3
  • 83
    • 84907131417 scopus 로고
    • Drug injecting and HIV infection: New directions for social science research
    • Stimson, G. (1992) Drug injecting and HIV infection: New directions for social science research. Int. J. Addict., 27:147-163.
    • (1992) Int. J. Addict. , vol.27 , pp. 147-163
    • Stimson, G.1
  • 84
    • 0026610297 scopus 로고
    • 3H]Nisoxetine: A radioligand for quantitation of norepinephrine uptake sites by autoradiography or by homogenate binding
    • 3H]Nisoxetine: A radioligand for quantitation of norepinephrine uptake sites by autoradiography or by homogenate binding. J. Pharmacol. Exp. Ther., 260:427-436.
    • (1992) J. Pharmacol. Exp. Ther. , vol.260 , pp. 427-436
    • Tejani-Butt, S.M.1
  • 85
    • 0026697266 scopus 로고
    • Amantadine in the treatment of cocaine withdrawal
    • Thompson, D.F. (1992) Amantadine in the treatment of cocaine withdrawal. Ann. Pharmacother., 26:933-934.
    • (1992) Ann. Pharmacother. , vol.26 , pp. 933-934
    • Thompson, D.F.1
  • 86
    • 0027048887 scopus 로고
    • Neurotransmitter transporter family cDNAs in a rat midbrain library: 'Orphan transporters' suggest sizable structural variations
    • Uhl, G.R., Kitayama, S., Gregor, P., Nanthakumar, E., Persico, A., and Shimada, S. (1992) Neurotransmitter transporter family cDNAs in a rat midbrain library: 'Orphan transporters' suggest sizable structural variations. Brain Res. Mol. Brain Res., 16:353-359.
    • (1992) Brain Res. Mol. Brain Res. , vol.16 , pp. 353-359
    • Uhl, G.R.1    Kitayama, S.2    Gregor, P.3    Nanthakumar, E.4    Persico, A.5    Shimada, S.6
  • 87
    • 0019219948 scopus 로고
    • Aryl 1,4-dialk(en)ylpiperazines as selective and very potent inhibitors of dopamine uptake
    • Van der Zee, P., Koger, H.S., Gootjes, J., and Hespe, W. (1980) Aryl 1,4-dialk(en)ylpiperazines as selective and very potent inhibitors of dopamine uptake. Eur. J. Med. Chem., 15:363-370.
    • (1980) Eur. J. Med. Chem. , vol.15 , pp. 363-370
    • Van Der Zee, P.1    Koger, H.S.2    Gootjes, J.3    Hespe, W.4
  • 88
    • 0026761657 scopus 로고
    • A human dopamine transporter cDNA predicts reduced glycosylation, displays a novel repetitive element and provides racially-dimorphic Taq1 RFLPs
    • Vandenbergh, D.J., Persico, A.M., and Uhl, G.R. (1992) A human dopamine transporter cDNA predicts reduced glycosylation, displays a novel repetitive element and provides racially-dimorphic Taq1 RFLPs. Mol. Brain Res., 15:161-166.
    • (1992) Mol. Brain Res. , vol.15 , pp. 161-166
    • Vandenbergh, D.J.1    Persico, A.M.2    Uhl, G.R.3
  • 91
    • 0002660912 scopus 로고
    • Brain dopamine and reward
    • Cooper, S.J. (ed.) London/NY: Academic Press
    • Wise, R.A. Brain dopamine and reward. In: Theory in Psychopharmacology. Cooper, S.J. (ed.) London/NY: Academic Press, 1981, pp. 103-122.
    • (1981) Theory in Psychopharmacology , pp. 103-122
    • Wise, R.A.1
  • 92
    • 0025615080 scopus 로고
    • A pilot trial of levodopa/ carbidopa in early cocaine abstinence
    • Wolfsohn, R., and Angrist, B. (1990) A pilot trial of levodopa/ carbidopa in early cocaine abstinence (letter). J. Clin. Psychopharmacol., 10:440-442.
    • (1990) J. Clin. Psychopharmacol. , vol.10 , pp. 440-442
    • Wolfsohn, R.1    Angrist, B.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.