Effects of various muscarinic ligands on M2AChR-Gi1α fusion protein expressed in Sf9 insect cells

Acta Pharmacologica Sinica

Volumn 23, Issue 3, 2002, Pages 230-236

  Wang, Hao ^a   Guo, Zheng Dong ^a   Li, Zhi ^a   Liu, Hong Rui ^a  

^a CHINA MEDICAL UNIVERSITY   (China)

Author keywords

Adenosine triphosphate; Guanosine diphosphate; Guanosine triphosphate; Inhibitory Gi G protein; Muscarinic agonists; Muscarinic antagonists; Muscarinic receptors; Radio ligand assay; Recombinant fusion proteins

Indexed keywords

[4 [(3 CHLOROPHENYL)CARBAMOYLOXY] 2 BUTYNYL]TRIMETHYLAMMONIUM; ACETYLCHOLINE; ADENOSINE TRIPHOSPHATE; ATROPINE; CARBACHOL; G PROTEIN COUPLED RECEPTOR; GUANOSINE 5' O (3 THIOTRIPHOSPHATE); GUANOSINE DIPHOSPHATE; GUANOSINE TRIPHOSPHATE; HYBRID PROTEIN; INHIBITORY GUANINE NUCLEOTIDE BINDING PROTEIN; MAGNESIUM CHLORIDE; MAGNESIUM ION; MUSCARINIC AGENT; MUSCARINIC M2 RECEPTOR; MUSCARINIC RECEPTOR BLOCKING AGENT; PILOCARPINE; QUINUCLIDINYL BENZILATE; CHRM1 PROTEIN, HUMAN; HETEROTRIMERIC GUANINE NUCLEOTIDE BINDING PROTEIN; LIGAND; MUSCARINIC RECEPTOR;

ANIMAL CELL; ARTICLE; BACULOVIRUS; CONTROLLED STUDY; DRUG RECEPTOR BINDING; INSECT CELL; LIGAND BINDING; NONHUMAN; POLYMERASE CHAIN REACTION; RECEPTOR AFFINITY; ANIMAL; BIOSYNTHESIS; CATTLE; CELL CULTURE; CYTOLOGY; GENETICS; HUMAN; INSECT; METABOLISM; RADIOASSAY;

ANIMALS; BACULOVIRIDAE; CATTLE; CELLS, CULTURED; GTP-BINDING PROTEIN ALPHA SUBUNITS, GI-GO; HETEROTRIMERIC GTP-BINDING PROTEINS; HUMANS; INSECTS; LIGANDS; MAGNESIUM CHLORIDE; RADIOLIGAND ASSAY; RECEPTOR, MUSCARINIC M2; RECEPTORS, MUSCARINIC; RECOMBINANT FUSION PROTEINS;

EID: 0036185620     PISSN: 16714083     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (13)

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