The human 5-HT7 serotonin receptor splice variants: Constitutive activity and inverse agonist effects

British Journal of Pharmacology

Volumn 135, Issue 6, 2002, Pages 1563-1571

  Krobert, Kurt A ^a,b   Levy, Finn Olav ^a,b  

^a UNIVERSITY OF OSLO   (Norway)

^b UNIVERSITY OF OSLO   (Norway)

Author keywords

Adenylyl cyclase; Constitutive activity; Inverse agonism; Splice variants

Indexed keywords

ADENYLATE CYCLASE; SEROTONIN 7 RECEPTOR; SEROTONIN AGONIST; SEROTONIN ANTAGONIST; SEROTONIN RECEPTOR; CLOZAPINE; FORSKOLIN; KETANSERIN; MESULERGINE; METERGOLINE; METHYSERGIDE; METITEPINE; RECEPTOR SUBTYPE; RITANSERIN; SPIPERONE;

ALTERNATIVE RNA SPLICING; ARTICLE; BIOSYNTHESIS; CELL LINE; DOSE RESPONSE; DRUG ANTAGONISM; DRUG EFFECT; GENETIC TRANSFECTION; GENETIC VARIABILITY; GENETICS; HUMAN; METABOLISM; PHYSIOLOGY; CELL CULTURE; CELL MEMBRANE; CONCENTRATION RESPONSE; CONTROLLED STUDY; CORRELATION ANALYSIS; CULTURE MEDIUM; DRUG EFFICACY; DRUG POTENCY; ENZYME ACTIVATION; ENZYME ACTIVITY; ENZYME INHIBITION; HUMAN CELL; PRIORITY JOURNAL; PROTEIN EXPRESSION; PROTEIN FUNCTION; RECEPTOR BLOCKING; RECEPTOR DENSITY;

ADENYLATE CYCLASE; ALTERNATIVE SPLICING; CELL LINE; DOSE-RESPONSE RELATIONSHIP, DRUG; HUMANS; RECEPTORS, SEROTONIN; SEROTONIN AGONISTS; SEROTONIN ANTAGONISTS; TRANSFECTION; VARIATION (GENETICS);

EID: 0036009759     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0704588     Document Type: Article

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