Distinct function of the cytoplasmic tail in human D1-like receptor ligand binding and coupling

FEBS Letters

Volumn 470, Issue 2, 2000, Pages 183-188

  Jackson, Adele ^a   Iwasiow, Rafal M ^a   Tiberi, Mario ^a  

^a OTTAWA HOSPITAL RESEARCH INSTITUTE   (Canada)

Author keywords

Binding affinity; Constitutive activity; D1 like receptor; Dopamine; G protein activation; G protein coupled receptor

Indexed keywords

8 CHLORO 2,3,4,5 TETRAHYDRO 3 METHYL 5 PHENYL 1H 3 BENZAZEPIN 7 OL HYDROGEN MALEATE; ADENYLATE CYCLASE; BUTACLAMOL; CHIMERIC PROTEIN; CYCLIC AMP; DOPAMINE; DOPAMINE 1 RECEPTOR; EXTRACHROMOSOMAL DNA; FLUPENTIXOL; G PROTEIN COUPLED RECEPTOR;

ARTICLE; BINDING AFFINITY; CYTOPLASM; DRUG POTENCY; HUMAN; HUMAN CELL; KIDNEY CELL; LIGAND BINDING; NONHUMAN; PRIORITY JOURNAL; PROTEIN EXPRESSION; RECEPTOR BINDING; TAIL;

ADENYLATE CYCLASE; ANTIPSYCHOTIC AGENTS; BINDING SITES; CELL LINE; CELL MEMBRANE; CYCLIC AMP; DOPAMINE; DOPAMINE ANTAGONISTS; DOSE-RESPONSE RELATIONSHIP, DRUG; ENZYME ACTIVATION; GENE EXPRESSION; HUMANS; LIGANDS; RECEPTORS, DOPAMINE D1; RECEPTORS, DOPAMINE D5; RECOMBINANT FUSION PROTEINS; STRUCTURE-ACTIVITY RELATIONSHIP; THERMODYNAMICS; TRANSFECTION;

EID: 0034708805     PISSN: 00145793     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-5793(00)01315-6     Document Type: Article

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