SCOPUS 정보 검색 플랫폼

Proceedings of the National Academy of Sciences of the United States of America

Volumn 98, Issue 9, 2001, Pages 5312-5316

The binding conformation of Taxol in β-tubulin: A model based on electron crystallographic density

(5) Snyder, James P a Nettles, James H a Cornett, Ben a Downing, Kenneth H b Nogales, Eva b,c

a EMORY UNIVERSITY (United States)

b LAWRENCE BERKELEY NATIONAL LABORATORY (United States)

c UNIVERSITY OF CALIFORNIA (United States)

Author keywords

[No Author keywords available]

Indexed keywords

BETA TUBULIN; PACLITAXEL;

ARTICLE; BINDING AFFINITY; CRYSTALLOGRAPHY; DRUG BINDING SITE; DRUG CONFORMATION; DRUG PROTEIN BINDING; DRUG STRUCTURE; HUMAN; HUMAN CELL; MUTATION; PHOTOAFFINITY LABELING; PRIORITY JOURNAL; STRUCTURE ACTIVITY RELATION;

BINDING SITES; CRYSTALLOGRAPHY; DRUG RESISTANCE, NEOPLASM; MICROSCOPY, ELECTRON; MODELS, MOLECULAR; MOLECULAR CONFORMATION; PACLITAXEL; PHOTOAFFINITY LABELS; STRUCTURE-ACTIVITY RELATIONSHIP; TAXOIDS; TUBULIN;

EID: 0035942226 PISSN: 00278424 EISSN: None Source Type: Journal
DOI: 10.1073/pnas.051309398 Document Type: Article

Times cited : (372)

References (49)

1
- 0001881989
- eds. Georg, G. I., Chen, T. T., Ojima, I. & Vyas, D. M. (Am. Chem. Soc., Washington, DC), ACS Symposium Series 583
- (1995) Taxane Anticancer Agents , pp. 31
- Holmes, F.A.¹ Kudelka, A.P.² Kavanagh, J.J.³ Huber, M.H.⁴ Ajani, J.A.⁵ Valero, V.⁶

2
- 0001843250
- eds. Georg, G. I., Chen, T. T., Ojima, I. & Vyas, D. M. (Am. Chem. Soc., Washington, DC), ACS Symposium Series 583
- (1995) Taxane Anticancer Agents , pp. 138-153
- Jordon, M.A.¹ Wilson, L.²

3
- 33748226949
- (1994) Angew. Chem. Int. Ed. Engl. , vol.33 , pp. 15-44
- Nicolaou, K.C.¹ Dai, W.M.² Guy, R.K.³

4
- 0019859353
- (1981) J. Cell Biol. , vol.91 , pp. 479-587
- Parness, J.¹ Horwitz, S.B.²

5
- 0027467778
- (1993) Biochemistry , vol.32 , pp. 2747-2755
- Diaz, J.F.¹ Andreu, J.M.²

6
- 0026747827
- (1992) J. Natl. Cancer Inst. , vol.84 , pp. 785-788
- Rao, S.¹ Horwitz, S.B.² Ringel, I.³

7
- 0028169689
- (1994) J. Biol. Chem. , vol.269 , pp. 3132-3134
- Rao, S.¹ Krauss, N.E.² Heerding, J.M.³ Swindell, C.S.⁴ Ringel, I.⁵ Orr, G.A.⁶ Horwitz, S.B.⁷

8
- 0028123221
- (1994) J. Med. Chem. , vol.37 , pp. 2976-2980
- Dasagupta, D.¹ Park, H.² Harriman, G.C.B.³ Georg, G.I.⁴ Himes, R.⁵

9
- 0028178514
- (1994) Biochemistry , vol.33 , pp. 6676-6683
- Combeau, C.¹ Commerçon, A.² Mioskowski, C.³ Rousseau, B.⁴ Aubert, F.⁵ Goeldner, M.⁶

10
- 0028861177
- (1995) J. Biol. Chem. , vol.270 , pp. 20235-20238
- Rao, S.¹ Orr, G.A.² Chaudhary, A.G.³ Kingston, D.G.I.⁴ Horwitz, S.B.⁵

11
- 0030611015
- (1997) Biochemistry , vol.36 , pp. 3820-3825
- Loeb, C.¹ Combeau, C.² Shret-Sabatier, L.³ Breton-Gilet, A.⁴ Faucher, D.⁵ Rousseau, B.⁶ Commerçon, A.⁷ Goeldner, M.⁸

12
- 0032495513
- Nature (London)
- (1998) , vol.391 , pp. 199-202
- Nogales, E.¹ Wolf, S.G.² Downing, K.H.³

13
- 0000813445
- (1990) Acta Crystallogr. C , vol.46 , pp. 781-784
- Guéritte-Voegelein, F.¹ Guenard, D.² Mangatal, L.³ Potier, P.⁴ Guilhem, J.⁵ Cesario, M.⁶

14
- 0033534629
- (1999) Cell , vol.96 , pp. 79-88
- Nogales, E.¹ Whittaker, M.² Milligan, R.A.³ Downing, K.H.⁴

15
- 0028920209
- (1995) Pharm. Res. , vol.12 , pp. 337-341
- Gao, Q.¹ Wei, J.-M.² Chen, S.-H.³

16
- 0029901458
- (1996) Tetrahedron Lett. , vol.37 , pp. 3425-3428
- Gao, Q.¹ Chen, S.-H.²

17
- 0027213794
- (1993) Tetrahedron , vol.49 , pp. 6533-6544
- Dubois, J.¹ Guénard, D.² Guéritte-Voegelein, F.³ Guedira, N.⁴ Potier, P.⁵ Gillet, B.⁶ Beloeil, J.-C.⁷

18
- 0027305373
- (1993) Tetrahedron , vol.49 , pp. 6545-6560
- Williams, H.J.¹ Scott, A.I.² Dieden, R.A.³ Swindell, C.S.⁴ Chirlian, L.E.⁵ Francl, M.M.⁶ Heerding, J.M.⁷ Krauss, N.E.⁸

19
- 0028383232
- (1994) Supercomput. Appl. High Perform. Comput. , vol.6 , pp. 24-34
- Cachau, R.E.¹ Gussio, R.² Beutler, J.A.³ Chmurny, G.N.⁴ Hilton, B.D.⁵ Muschik, G.M.⁶ Erickson, J.W.⁷

20
- 0027730478
- (1993) J. Am. Chem. Soc. , vol.113 , pp. 11650-11651
- Vander Velde, D.G.¹ Georg, G.I.² Grunewald, G.L.³ Gunn, C.W.⁴ Mitscher, L.A.⁵

21
- 0028519119
- (1994) Chem. Biol. , vol.1 , pp. 107-112
- Paloma, L.G.¹ Guy, R.K.² Wrasidlo, W.³ Nicolaou, K.C.⁴

22
- 0030750497
- (1997) J. Am. Chem. Soc. , vol.119 , pp. 5519-5527
- Ojima, I.¹ Kuduk, S.D.² Chakravarty, S.³ Ourevitch, M.⁴ Bégue, J.-P.⁵

23
- 0040283025
- (1998) Biorg. Med. Chem. , vol.6 , pp. 1857-1863
- Jiménez-Barbero, J.¹ Souto, A.A.² Abal, M.³ Barasoain, I.⁴ Evangelio, J.A.⁵ Acuña, A.U.⁶ Andreu, J.M.⁷ Amat-Guerri, F.⁸

24
- 83755208229
- (2000) J. Am. Chem. Soc. , vol.172 , pp. 724-725
- Snyder, J.P.¹ Nevins, N.² Cicero, D.O.³ Jansen, J.J.⁴

25
- 6244283606
- (1997) J. Comp. Chem. , vol.18 , pp. 1175-1189
- Ewing, T.J.A.¹ Kuntz, E.D.²

26
- 0030599010
- (1996) J. Mol. Biol. , vol.261 , pp. 470-489
- Rarey, M.¹ Kramer, B.² Lengauer, T.³ Klebe, G.⁴

27
- 0029156949
- (1995) Proc. Natl. Acad. Sci. USA , vol.92 , pp. 6920-6924
- Mastropaolo, D.¹ Camerman, A.² Luo, Y.³ Brayer, G.D.⁴ Camerman, N.⁵

28
- 0033551046
- (1999) Proc. Nad. Acad. Sci. USA , vol.96 , pp. 4256-4261
- Ojima, I.¹ Chakravarty, S.² Inoue, T.³ Lin, L.⁴ He, L.⁵ Horwitz, S.B.⁶ Kuduk, S.D.⁷ Danishefsky, S.J.⁸

29
- 0033621479
- (1999) J. Biol. Chem. , vol.274 , pp. 37990-37994
- Rao, S.¹ He, L.² Chakravarty, S.³ Ojima, I.⁴ Orr, G.A.⁵ Horwitz, S.B.⁶

30
- 0034681179
- (2000) Biochemistry , vol.39 , pp. 281-291
- Li, Y.¹ Poliks, B.² Cegelski, L.³ Poliks, M.⁴ Gryczynski, Z.⁵ Piszczek, G.⁶ Jagtap, P.G.⁷ Studelska, D.R.⁸ Kingston, D.G.I.⁹ Schaefer, J.¹⁰ Bane, S.¹¹

31
- 0032937808
- (1999) J. Med. Chem. , vol.42 , pp. 291-299
- Milanesio, M.¹ Ugliengo, P.² Viterho, D.³ Appendino, G.⁴

32
- 0002659224
- (1995) Perspect. Drug Discovery Des. , vol.3 , pp. 85-105
- Klebe, G.¹

33
- 0034636084
- (2000) Biochemistry , vol.39 , pp. 3972-3978
- He, L.¹ Jagtap, P.G.² Kingston, D.G.I.³ Shen, H.-J.⁴ Orr, G.A.⁵ Horwitz, S.B.⁶

34
- 0033581642
- (1999) Biorg. Med. Chem. Lett. , vol.9 , pp. 3047-3052
- Boge, T.C.¹ Wu, Z.-J.² Himes, R.H.³ Vander Velde, D.G.⁴ Georg, G.I.⁵

35
- 0034712232
- (2000) J. Org. Chem. , vol.65 , pp. 1059-1068
- Wang, M.¹ Cornett, B.² Nettles, J.³ Liotta, D.C.⁴ Snyder, J.P.⁵

36
- 0004122931
- (Sanders College Pub., New York), 2nd Ed.
- (1999) Biochemistry , pp. 534-535
- Garret, R.H.¹ Grisham, C.M.²

37
- 0000655508
- eds. Georg, G. I., Chen, T. T., Ojima, I. & Vyas, D. M. (Am. Chem. Soc., Washington, DC), ACS Symposium Series 583
- (1995) Taxane Anticancer Agents , pp. 203-216
- Kingston, D.G.I.¹

38
- 0025804190
- (1991) J. Med. Chem. , vol.34 , pp. 992-998
- Guéritte-Voegelein, F.¹ Guénard, D.² Lavell, F.³ LeGoff, M.-T.⁴ Mangatal, L.⁵ Potier, P.⁶

39
- 0025827992
- (1991) J. Med. Chem. , vol.34 , pp. 1176-1184
- Swindell, C.S.¹ Krauss, N.E.² Horwitz, S.B.³ Ringel, I.⁴

40
- 0029968838
- (1996) J. Med. Chem. , vol.39 , pp. 1555-1559
- Williams, H.J.¹ Moyna, G.² Scott, A.I.³ Swindell, C.S.⁴ Chirlian, L.E.⁵ Heerding, J.M.⁶ Williams, D.K.⁷

41
- 0027935479
- (1994) J. Med. Chem. , vol.37 , pp. 2602-2608
- Ojima, I.¹ Duclos, O.² Zucco, M.³ Bissery, M.-C.⁴ Combeau, C.⁵ Vrignaud, P.⁶ Riou, J.F.⁷ Lavelle, F.⁸

42
- 0028097492
- (1994) J. Med. Chem. , vol.37 , pp. 3337-3343
- Boge, T.C.¹ Himes, R.H.² Vander Velde, D.G.³ Georg, G.I.⁴

43
- 0028791932
- (1995) Bioorg. Med. Chem. Lett. , vol.5 , pp. 2741-2746
- Chen, S.-H.¹ Wei, J.-M.² Long, B.H.³ Fairchild, C.A.⁴ Carboni, J.⁵ Mamber, W.W.⁶ Rose, W.C.⁷ Johnston, K.⁸ Casazza, A.M.⁹ Kadow, J.F.¹⁰

44
- 0028235069
- (1994) J. Am. Chem. Soc. , vol.116 , pp. 4097-4098
- Chaudhary, A.G.¹ Gharpure, M.M.² Rimoldi, J.M.³ Chordia, M.D.⁴ Gunatilaka, A.A.L.⁵ Kingston, D.G.I.⁶ Grover, S.⁷ Lin, C.⁸ Hamel, E.⁹

45
- 0030812058
- (1997) Bioorg. Med. Chem. Lett. , vol.7 , pp. 1941-1944
- Wender, P.A.¹ Lee, D.² Lal, T.K.³

46
- 0031562458
- (1997) Tetrahedron , vol.53 , pp. 3441-3456
- Liang, X.¹ Kingston, D.G.I.² Long, B.H.³ Fairchild, C.A.⁴ Johnston, K.A.⁵

47
- 0030758777
- (1997) J. Biol. Chem. , vol.272 , pp. 17118-17125
- Giannakakou, P.¹ Sackett, D.L.² Kang, Y.-K.³ Shan, Z.⁴ Buters, J.T.M.⁵ Fojo, T.⁶ Poruchynsky, M.S.⁷

48
- 12944277104
- First Published February 25, 2000; 10.1073/pnas.040546297
- (2000) Proc. Natl. Acad. Sci. USA , vol.97 , pp. 2904-2909
- Giannakakou, P.¹ Gussio, R.² Nogales, E.³ Downing, K.H.⁴ Zaharevitz, D.⁵ Bollbuck, B.⁶ Poy, G.⁷ Sackett, D.⁸ Nicolaou, K.C.⁹ Fojo, T.¹⁰

49
- 0034728938
- (2000) Tetrahedron Lett. , vol.41 , pp. 3331-3334
- Dubois, J.¹ Thoret, S.² Guéritte, F.³ Guénard, D.⁴

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.