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Current Medicinal Chemistry

Volumn 8, Issue 8, 2001, Pages 893-907

Macrocycles mimic the extended peptide conformation recognized by aspartic, serine, cysteine and metallo proteases

(2) Tyndall, J D A a Fairlie, D P a

a UNIVERSITY OF QUEENSLAND (Australia)

Author keywords

[No Author keywords available]

Indexed keywords

AMINO ACID; AMINOPEPTIDASE; AMPRENAVIR; ASPARTIC PROTEINASE; ASPARTIC PROTEINASE INHIBITOR; CYCLOSPORIN; CYCLOTHEONAMIDE; CYSTEINE PROTEINASE; DIPEPTIDYL CARBOXYPEPTIDASE INHIBITOR; ENKEPHALINASE INHIBITOR; GELATINASE A; GELATINASE B; IMMUNOSUPPRESSIVE AGENT; INDINAVIR; INTERSTITIAL COLLAGENASE; MACROCYCLIC COMPOUND; MATRIX METALLOPROTEINASE 8 INHIBITOR; MATRIX METALLOPROTEINASE 9 INHIBITOR; MATRIX METALLOPROTEINASE INHIBITOR; METALLOPROTEINASE; METALLOPROTEINASE INHIBITOR; PLASMEPSIN II INHIBITOR; PROTEINASE INHIBITOR; RENIN INHIBITOR; SERINE PROTEINASE; SERINE PROTEINASE INHIBITOR; STROMELYSIN; TUMOR NECROSIS FACTOR ALPHA; TUMOR NECROSIS FACTOR ALPHA CONVERTING ENZYME; UNCLASSIFIED DRUG; UNINDEXED DRUG;

AMINO ACID SEQUENCE; ARTHRITIS; ARTICLE; CANCER; CONGESTIVE HEART FAILURE; DRUG ABSORPTION; DRUG BIOAVAILABILITY; DRUG DEGRADATION; DRUG DESIGN; DRUG POTENTIATION; DRUG STABILITY; DRUG STRUCTURE; ENZYME BINDING; ENZYME STRUCTURE; HUMAN; HUMAN IMMUNODEFICIENCY VIRUS 1; HYPERTENSION; MOLECULAR MIMICRY; MOLECULAR RECOGNITION; PROTEIN CONFORMATION; STRUCTURE ACTIVITY RELATION;

EID: 0034929804 PISSN: 09298673 EISSN: None Source Type: Journal
DOI: 10.2174/0929867013372715 Document Type: Article

Times cited : (95)

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