Activity of cytisine and its brominated isosteres on recombinant human α7, α4β2 and α4β4 nicotinic acetylcholine receptors

Journal of Neurochemistry

Volumn 78, Issue 5, 2001, Pages 1029-1043

  Houlihan, Lee M ^a   Slater, Yvonne ^a   Guerra, Doris L ^b   Peng, Jian Hong ^c   Kuo, Yen Ping ^c   Lukas, Ronald J ^c   Cassels, Bruce K ^b   Bermudez, Isabel ^a  

^a OXFORD BROOKES UNIVERSITY   (United Kingdom)

^b UNIVERSITY OF CHILE   (Chile)

^c BARROW NEUROLOGICAL INSTITUTE   (United States)

Author keywords

Cytisine; Neuronal nicotinic acetylcholine receptor; Two site receptor occupation model; Xenopus oocyte

Indexed keywords

BUNGAROTOXIN; CYTISINE; NICOTINIC RECEPTOR; RECEPTOR SUBTYPE;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; BROMINATION; CONTROLLED STUDY; ENZYME ACTIVITY; ENZYME BINDING; ENZYME INHIBITION; HUMAN; HUMAN CELL; NONHUMAN; OOCYTE; PRIORITY JOURNAL; XENOPUS;

ACETYLCHOLINE; ANIMALS; BINDING, COMPETITIVE; BUNGAROTOXINS; CYTOSINE; ELECTROPHYSIOLOGY; GENE EXPRESSION; HUMANS; IODINE RADIOISOTOPES; OOCYTES; RECEPTORS, NICOTINIC; RECOMBINANT PROTEINS; RNA, MESSENGER; TRITIUM; XENOPUS LAEVIS;

ANIMALIA;

EID: 0034839206     PISSN: 00223042     EISSN: None     Source Type: Journal    
DOI: 10.1046/j.1471-4159.2001.00481.x     Document Type: Article

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