Pyrazole ligands: Structure - Affinity/activity relationships and estrogen receptor-α-selective agonists

Journal of Medicinal Chemistry

Volumn 43, Issue 26, 2000, Pages 4934-4947

  Stauffer, S R ^a   Coletta, C J ^a   Tedesco, R ^a   Nishiguchi, G ^a   Carlson, K ^a   Sun, J ^a   Katzenellenbogen, B S ^a   Katzenellenbogen, J A ^a  

^a UNIVERSITY OF ILLINOIS   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ESTRADIOL; ESTROGEN RECEPTOR ALPHA; ESTROGEN RECEPTOR BETA; HYDROXYL GROUP; PHENOL DERIVATIVE; PROPYLPYRAZOLE TRIOL; PYRAZOLE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; GENETIC TRANSCRIPTION; MOLECULAR INTERACTION; MOLECULAR MODEL; RECEPTOR BINDING; STRUCTURE ACTIVITY RELATION;

BINDING, COMPETITIVE; ESTROGEN RECEPTOR ALPHA; HUMANS; LIGANDS; MODELS, MOLECULAR; PHENOLS; PYRAZOLES; RADIOLIGAND ASSAY; RECEPTORS, ESTROGEN; STRUCTURE-ACTIVITY RELATIONSHIP; TRANS-ACTIVATION (GENETICS); TUMOR CELLS, CULTURED;

EID: 0034727853     PISSN: 00222623     EISSN: None     Source Type: Journal    
DOI: 10.1021/jm000170m     Document Type: Article

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