Analogs of lactam derivatives of α-melanotropin with basic and acidic residues

Biochemical and Biophysical Research Communications

Volumn 272, Issue 1, 2000, Pages 23-28

  Bednarek, Maria A ^a   MacNeil, Tanya ^a   Kalyani, Rubana N ^a   Tang, Rui ^a   Van Der Ploeg, Lex H T ^a   Weinberg, David H ^a  

^a MERCK RESEARCH LABORATORIES   (United States)

Author keywords

Binding affinity; cAMP accumulation assay; Glutamic acid scan; Lysine scan; Melanocortin receptor; Melanotropin

Indexed keywords

ALPHA INTERMEDIN DERIVATIVE; DRUG RESIDUE; GLUTAMIC ACID; LACTAM DERIVATIVE; LIGAND; MELANOCORTIN RECEPTOR; N ACETYL ALPHA INTERMEDIN[4-10]CYCLO[4 NORLEUCINE 5 ASPARTIC ACID 7 [3 (2 NAPHTHYL)ALANINE] 10 LYSINAMIDE]; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; LIGAND BINDING; PRIORITY JOURNAL;

EID: 0034720468     PISSN: 0006291X     EISSN: None     Source Type: Journal    
DOI: 10.1006/bbrc.2000.2589     Document Type: Article

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