Molecular basis for the interaction of [Nle4,D-Phe7]melanocyte stimulating hormone with the human melanocortin-1 receptor (melanocyte α- MSH receptor)

Journal of Biological Chemistry

Volumn 272, Issue 37, 1997, Pages 23000-23010

  Yang, Ying Kui ^a   Dickinson, Chris ^a   Haskell Luevano, Carrie ^a   Gantz, Ira ^a,b  

^a UNIVERSITY OF MICHIGAN MEDICAL SCHOOL   (United States)

^b 1150 W Medical Center Dr ^*  (United States)

Author keywords

[No Author keywords available]

Indexed keywords

GUANINE NUCLEOTIDE BINDING PROTEIN; INTERMEDIN; IODINE 125; MEMBRANE RECEPTOR;

AMINO ACID SUBSTITUTION; ARTICLE; BINDING AFFINITY; HORMONE RECEPTOR INTERACTION; HUMAN; HUMAN CELL; LIGAND BINDING; MOLECULAR MODEL; PRIORITY JOURNAL; SITE DIRECTED MUTAGENESIS;

EID: 0030761093     PISSN: 00219258     EISSN: None     Source Type: Journal    
DOI: 10.1074/jbc.272.37.23000     Document Type: Article

References (23)

1. De Wied, D., and Jolies, J. (1982) Physiol. Rev. 62 976-1059
2. Tatro, J. B. (1997) Neuroimmunomodulation, in press
3. Fan, W., Boston, B. A., Kesterson, R. A., Hruby, V. J., and Cone, R. D. (1997) Nature 385, 165-168
4. Sawyer, T. K., Sanfillippo, P. J., Hruby, V. J., Engel, M. H., Howard, C. B., Burnett, J. B., and Hadley, M. E. (1980) Proc. Natl. Acad. Sci. U. S. A. 77, 5754-5758
5. Hruby, V. J., Wilkes, B. C., Cody, W. L., Sawyer, T. K., and Hadley, M. E. (1984) Peptide Protein Rev. 3, 1-64
6. Haskell-Luevano, C., Miwa, H., Dickinson, C., Hadley, M. E., Hruby, V. J., Yamada, T., and Gantz, I. (1996) J. Med. Chem. 39, 432-435
7. Mountjoy, K G. (1994) Mol. Cell. Endocrinol. 102, R7-R11
8. Haskell-Luevano, C., Sawyer, T. K., Trumpp-Kallmeyer, S., Bikker, J. A., Humblet, C., Gantz, I., and Hruby, V. J. (1996) Drug Design and Discovery 14, 197-211
9. Sawyer, T. K., Castrucci, A. M., Staples, D. J., Affholter, J. A., DeVaux, A. E., Hruby, V. J., and Hadley, M. E. (1993) Ann. N. Y. Acad. Sci. 680, 597-399
10. Chhajlani, V., Xu, X., Blauw, J., and Sudarshi, S. (1996) Biochem. Biophys. Res. Commun. 219, 521-525
11. Al-Obeidi, F., Hadley, M. E., Pettitt, B. M., and Hruby, V. J. (1989) J. Am. Chem. Soc. 111, 3413-3416
12. Al-Obeidi, F., Castrucci, A. M., Hadley, M. E., and Hruby, V. J. (1989) J. Med. Chem. 32, 2555-2561
13. Henderson, R., Baldwin, J. M., Ceska, T. A., Zemlin, F., Beckmann, E., and Downing, K. H. (1990) J. Mol. Biol. 213, 899-929
14. Schertler, G. F. X., Villa, C., and Henderson, R. (1993) Nature 362, 770-772
15. Sambrook, J., Fritsch, E. F., and Maniatis, T. (1989) Molecular Cloning: A Laboratory Manual, 2nd Ed., Cold Spring Harbor Laboratory, Cold Sring Harbor, NY
16. Tatro, J. B., and Reichlin, S. (1987) Endocrinology 121, 1900-1907
17. Haskell-Luevano, C., Miwa, H., Dickinson, C., Hruby, V. J., Yamada, T., and Gantz, I. (1994) Biochem. Biophys. Res. Commun. 204, 1137-1142
18. Prusis, P., Frändberg, P-A., Kalvinsh, I., Muceniece, R., and Wikberg, J. E. S. (1995) Biochem. Biophys. Res. Commun. 210, 205-210
19. Frändberg, P-A., Muceniece, R., Prusis, P., Wikberg, J., and Chhajlani, V. (1994) Biochem. Biophys. Res. Commun. 207, 1266-1271
20. Strader, C. D., Sigal, I. S., Candelore, M. R., Rands, E., Hill, W. S., and Dixon, R. A. F. (1988) J. Biol. Chem. 263, 10267-10271
21. Robbins L. S., Nadeau, J. H., Johnson, K R., Kelly, M. A., Roselli-Rehfuss, L., Baack, E., Mountjoy, K. G., and Cone, R. (1993) Cell 72, 827-834
22. Cone, R. (1995) Endocrine Society Meeting, Washington, D. C., June 14, 1995
23. Mitchell, J. B. O., Nandi, C. L., McDonald, I. K., Thomton, J. M., and Price, S. L. (1994) J. Mol. Biol. 239, 315-331