6-[18F]fluoro-A-85380, a novel radioligand for in vivo imaging of central nicotinic acetylcholine receptors

Life Sciences

Volumn 67, Issue 4, 2000, Pages 463-469

  Horti, Andrew G ^a   Chefer, Svetlana I ^a   Mukhin, Alexey G ^a   Koren, Andrei O ^a   Gündisch, Daniela ^a   Links, Jonathan M ^a,b   Kurian, Varughese ^a   Dannals, Robert F ^b   London, Edythe D ^a  

^a NATIONAL INSTITUTE ON DRUG ABUSE   (United States)

^b DEPARTMENT OF PATHOLOGY   (United States)

Author keywords

6 18F fluoro 3 (2(S)azetidinyl methoxy)pyridine (6 18F fluoro A 85380, 6 18F FA); Nicotinic acetylcholine receptor; Positron emission tomography (nAChRs)

Indexed keywords

3 (2 AZETIDINYLMETHOXY)PYRIDINE F 18; CHOLINERGIC RECEPTOR; RADIOLIGAND; UNCLASSIFIED DRUG; 3 (2 AZETIDINYLMETHOXY)PYRIDINE; AZETIDINE DERIVATIVE; DIAGNOSTIC AGENT; FLUORINE; NICOTINIC RECEPTOR;

ANIMAL TISSUE; ARTICLE; BRAIN SCINTISCANNING; CHEMICAL STRUCTURE; CHOLINERGIC SYSTEM; CONTROLLED STUDY; FLUORINATION; IN VITRO STUDY; NONHUMAN; POSITRON EMISSION TOMOGRAPHY; RADIOACTIVITY; RHESUS MONKEY; ANIMAL; BRAIN; COMPUTER ASSISTED EMISSION TOMOGRAPHY; FISCHER 344 RAT; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; MACACA; MALE; METABOLISM; RAT; SCINTISCANNING; SYNTHESIS; TISSUE DISTRIBUTION;

ANIMALS; AZETIDINES; BRAIN; CHROMATOGRAPHY, HIGH PRESSURE LIQUID; FLUORINE RADIOISOTOPES; MACACA MULATTA; MALE; RATS; RATS, INBRED F344; RECEPTORS, NICOTINIC; TISSUE DISTRIBUTION; TOMOGRAPHY, EMISSION-COMPUTED;

EID: 0034674053     PISSN: 00243205     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0024-3205(00)00635-4     Document Type: Article

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