Inhibitors of kinesin activity from structure-based computer screening

Biochemistry

Volumn 39, Issue 10, 2000, Pages 2805-2814

  Hopkins, Seth C ^a,c   Vale, Ronald D ^a,b   Kuntz, Irwin D ^a  

^a UNIVERSITY OF CALIFORNIA   (United States)

^b UNIVERSITY OF CALIFORNIA   (United States)

^c SUNOVION PHARMACEUTICALS INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ANTHRAQUINONE DERIVATIVE; ENZYME INHIBITOR; FLUORESCEIN DERIVATIVE; KINESIN; NAPHTHALENE DERIVATIVE; PHENOLPHTHALEIN;

ARTICLE; BINDING SITE; COMPUTER ANALYSIS; CONTROLLED STUDY; DISSOCIATION CONSTANT; ENZYME INHIBITOR INTERACTION; HUMAN; INHIBITION KINETICS; MOLECULAR DYNAMICS; PRIORITY JOURNAL;

ADENOSINE TRIPHOSPHATASES; BINDING SITES; COMPUTATIONAL BIOLOGY; COMPUTER SIMULATION; ENZYME INHIBITORS; FLUORESCENT DYES; HUMANS; KINESIN; MODELS, MOLECULAR; ROSE BENGAL; SOFTWARE; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0034646180     PISSN: 00062960     EISSN: None     Source Type: Journal    
DOI: 10.1021/bi992474k     Document Type: Article

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