Identification of residues involved in neurotensin binding and modeling of the agonist binding site in neurotensin receptor 1

Journal of Biological Chemistry

Volumn 275, Issue 1, 2000, Pages 328-336

  Barroso, Séverine ^a   Richard, Françoise ^a   Nicolas Ethève, Delphine ^a   Reversat, Jean Louis ^b   Bernassau, Jean Marie ^b   Kitabgi, Patrick ^a   Labbé Jullié, Catherine ^a  

^a INSTITUT DE PHARMACOLOGIE MOLÉCULAIRE ET CELLULAIRE   (France)

^b SANOFI   (France)

Author keywords

[No Author keywords available]

Indexed keywords

2 [[1 (7 CHLORO 4 QUINOLINYL) 5 (2,6 DIMETHOXYPHENYL) 3 PYRAZOLYL]CARBONYLAMINO] 2 ADAMANTANECARBOXYLIC ACID; COMPLEMENTARY DNA; IODINE 125; NEUROPEPTIDE; NEUROTENSIN; NEUROTENSIN RECEPTOR; RECEPTOR SUBTYPE; TRITIUM;

ANIMAL CELL; ARTICLE; BINDING SITE; DOPAMINERGIC SYSTEM; HORMONE RECEPTOR INTERACTION; MOLECULAR MODEL; NEUROTRANSMISSION; NONHUMAN; PEPTIDE ANALYSIS; PRIORITY JOURNAL; SITE DIRECTED MUTAGENESIS; STRUCTURE ACTIVITY RELATION;

AMINO ACIDS; ANIMALS; BINDING SITES; BINDING, COMPETITIVE; COMPUTER SIMULATION; DOSE-RESPONSE RELATIONSHIP, DRUG; INOSITOL PHOSPHATES; MODELS, MOLECULAR; MUTAGENESIS; NEUROTENSIN; PYRAZOLES; QUINOLINES; RATS; RECEPTORS, NEUROTENSIN; STRUCTURE-ACTIVITY RELATIONSHIP;

ANIMALIA; TRITIUM;

EID: 0034614509     PISSN: 00219258     EISSN: None     Source Type: Journal    
DOI: 10.1074/jbc.275.1.328     Document Type: Article

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