Characterization of non-peptide antagonist and peptide agonist binding sites of the NK1 receptor with fluorescent ligands

Journal of Biological Chemistry

Volumn 272, Issue 34, 1997, Pages 21167-21175

  Turcatti, Gerardo ^a   Zoffmann, Sannah ^b   Lowe III, John A ^c   Drozda, Susan E ^c   Chassaing, Gérard ^d   Schwartz, Thue W ^b   Chollet, André ^a  

^a GLAXOSMITHKLINE   (United States)

^b UNIVERSITY OF COPENHAGEN   (Denmark)

^c PFIZER GLOBAL RESEARCH AND DEVELOPMENT   (United States)

^d SORBONNE UNIVERSITÉ   (France)

Author keywords

[No Author keywords available]

Indexed keywords

SUBSTANCE P RECEPTOR;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; BINDING SITE; CARBOXY TERMINAL SEQUENCE; CHO CELL; HORMONE RECEPTOR INTERACTION; LIGAND BINDING; NONHUMAN; PRIORITY JOURNAL;

ANIMALS; BINDING SITES; BINDING, COMPETITIVE; BIPHENYL COMPOUNDS; CHO CELLS; COS CELLS; CRICETINAE; DANSYL COMPOUNDS; FLUORESCENCE POLARIZATION; FLUORESCENT DYES; HUMANS; LIGANDS; MEMBRANE GLYCOPROTEINS; MUTAGENESIS, SITE-DIRECTED; PROTEIN STRUCTURE, SECONDARY; RECEPTORS, NEUROKININ-1; RECOMBINANT PROTEINS; SOLUBILITY; SPECTROMETRY, FLUORESCENCE; SUBSTANCE P;

ANIMALIA;

EID: 0030826420     PISSN: 00219258     EISSN: None     Source Type: Journal    
DOI: 10.1074/jbc.272.34.21167     Document Type: Article

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