Isolation of the serotoninergic 5-HT(4(e)) receptor from human heart and comparative analysis of its pharmacological profile in C6-glial and CHO cell lines

British Journal of Pharmacology

Volumn 129, Issue 4, 2000, Pages 771-781

  Mialet, Jeanne ^a,b   Berque Bestel, Isabelle ^b   Eftekhari, Pierre ^c   Gastineau, Monique ^a,b   Giner, Mireille ^b   Dahmoune, Yamina ^b   Donzeau Gouge, Patrick ^d   Hoebeke, Johan ^c   Langlois, Michel ^b   Sicsic, Sames ^b   Fischmeister, Rodolphe ^a,b   Lezoualc'h, Frank ^a,b  

^a INSERM   (France)

^b UNIVERSITÉ PARIS SACLAY   (France)

^c INSTITUT DE BIOLOGIE MOLÉCULAIRE ET CELLULAIRE   (France)

^d INSTITUT HOSPITALIER JACQUES CARTIER   (France)

Author keywords

Adenylyl cyclase; Atrial arrhythmia; Benzamides; G protein coupled receptors; Human; Inverse agonism; Serotoninergic receptors

Indexed keywords

1 METHYL 3 INDOLECARBOXYLIC ACID [1 [2 (METHYLSULFONYLAMINO)ETHYL] 4 PIPERIDINYLMETHYL] ESTER; 4 AMINO 5 CHLORO 2 METHOXYBENZOIC ACID 2 (1 PIPERIDINYL)ETHYL ESTER; 4 AMINO 5 CHLORO 2 METHOXYBENZOIC ACID 2 (3,5 DIMETHYLPIPERIDINO)ETHYL ESTER; ADENYLATE CYCLASE; CISAPRIDE; RENZAPRIDE; SEROTONIN 4 AGONIST; SEROTONIN 4 RECEPTOR; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; CHO CELL; DRUG POTENCY; GLIA CELL; HEART ATRIUM; HUMAN; HUMAN TISSUE; IMMUNOBLOTTING; NONHUMAN; PRIORITY JOURNAL; RECEPTOR BINDING; REVERSE TRANSCRIPTION POLYMERASE CHAIN REACTION;

EID: 0034095536     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0703101     Document Type: Article

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