[3H]5-hydroxytryptamine labels the agonist high affinity state of the cloned rat 5-HT4 receptor

European Journal of Pharmacology

Volumn 304, Issue 1-3, 1996, Pages 231-235

  Adham, Nika ^a   Gerald, Christophe ^a   Schechter, Lee ^b   Vaysse, Pierre ^a   Weinshank, Richard ^a   Branchek, Theresa ^a  

^a H LUNDBECK A S   (Denmark)

^b PFIZER INC   (United States)

Author keywords

5 HT4 receptor; affinity state; radioligand binding; splice variant

Indexed keywords

1 METHYL 3 INDOLECARBOXYLIC ACID [1 [2 (METHYLSULFONYLAMINO)ETHYL] 4 PIPERIDINYLMETHYL] ESTER; 2 DIPROPYLAMINO 8 HYDROXYTETRALIN; 5 CARBAMOYLTRYPTAMINE; 5 METHOXYTRYPTAMINE; ALPHA METHYLSEROTONIN; GUANINE NUCLEOTIDE; GUANINE NUCLEOTIDE BINDING PROTEIN; GUANOSINE 5' O (3 THIOTRIPHOSPHATE); KETANSERIN; RADIOLIGAND; RECEPTOR PROTEIN; RENZAPRIDE; SEROTONIN; SEROTONIN 4 RECEPTOR; SEROTONIN AGONIST; SEROTONIN ANTAGONIST; TROPISETRON; ZACOPRIDE; DIAGNOSTIC AGENT; INDOLE DERIVATIVE; SEROTONIN RECEPTOR; SULFONAMIDE;

ANIMAL CELL; ARTICLE; CELL LINE; CONCENTRATION RESPONSE; CONTROLLED STUDY; MOLECULAR CLONING; NONHUMAN; PRIORITY JOURNAL; RAT; RECEPTOR AFFINITY; RECEPTOR BINDING; AFFINITY LABELING; ANIMAL; BINDING COMPETITION; CELL STRAIN COS1; GENETIC TRANSFECTION; GENETICS; METABOLISM; RADIOASSAY;

AFFINITY LABELS; ANIMALS; BINDING, COMPETITIVE; CLONING, MOLECULAR; COS CELLS; INDOLES; RADIOLIGAND ASSAY; RATS; RECEPTORS, SEROTONIN; RECEPTORS, SEROTONIN, 5-HT4; SEROTONIN; SEROTONIN AGONISTS; SEROTONIN ANTAGONISTS; SULFONAMIDES; TRANSFECTION;

EID: 0030598576     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/0014-2999(96)00122-7     Document Type: Article

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