Pharmacological comparison between [3H]GR 113808 binding sites and functional 5-HT4 receptors in neurons

European Journal of Pharmacology

Volumn 298, Issue 2, 1996, Pages 165-174

  Ansanay, Hervé ^a   Sebben, Michèle ^a   Bockaert, Joël ^a   Dumuis, Aline ^a  

^a CNRS UPR 9023   (France)

Author keywords

5 HT4 receptor; Desensitization; Radioligand binding; 3H GR 113808

Indexed keywords

1 METHYL 3 INDOLECARBOXYLIC ACID [1 [2 (METHYLSULFONYLAMINO)ETHYL] 4 PIPERIDINYLMETHYL] ESTER; 2,3 DIHYDRO 2 OXO 1 BENZIMIDAZOLECARBOXYLIC ACID 6 METHOXY 3ALPHA TROPANYL ESTER; 2,3 DIHYDRO 3 ISOPROPYL 2 OXO 1 BENZIMIDAZOLECARBOXYLIC ACID 3ALPHA TROPANYLAMIDE; 3 ETHYL 2,3 DIHYDRO 2 OXO 1 BENZIMIDAZOLECARBOXYLIC ACID 3ALPHA TROPANYLAMIDE; 4 AMINO 5 CHLORO 2 METHOXYBENZOIC ACID 2 (1 PIPERIDINYL)ETHYL ESTER; 4 AMINO 5 CHLORO 2 METHOXYBENZOIC ACID 2 (DIETHYLAMINO)ETHYL ESTER; 4 AMINO 5 CHLORO N [(HEXAHYDRO 1H PYRROLIZIN 1 YL)METHYL] 2 METHOXYBENZAMIDE; 5 CARBAMOYLTRYPTAMINE; 5 METHOXY 3 (1,2,3,6 TETRAHYDRO 5 PYRIDYL) 1H INDOLE; 5 METHOXYTRYPTAMINE; ADENYLATE CYCLASE; BENZAMIDE DERIVATIVE; BENZIMIDAZOLONE DERIVATIVE; CISAPRIDE; CLEBOPRIDE; CYCLIC AMP; GR 127487; INDOLE DERIVATIVE; ITASETRON; METOCLOPRAMIDE; RADIOLIGAND; RENZAPRIDE; RN 76186; SB 205149; SC 49515; SEROTONIN; SEROTONIN 4 ANTAGONIST; SEROTONIN 4 RECEPTOR; SEROTONIN AGONIST; SEROTONIN ANTAGONIST; TROPISETRON; UNCLASSIFIED DRUG; ZACOPRIDE; SEROTONIN RECEPTOR; SULFONAMIDE;

ANIMAL CELL; ARTICLE; BINDING COMPETITION; BINDING SITE; BRAIN NERVE CELL; CONCENTRATION RESPONSE; CONTROLLED STUDY; DESENSITIZATION; DRUG SPECIFICITY; EMBRYO; LIGAND BINDING; MOUSE; NERVE CELL CULTURE; NONHUMAN; PRIORITY JOURNAL; RECEPTOR AFFINITY; ANIMAL; CELL CULTURE; DOSE RESPONSE; DRUG EFFECT; MOUSE STRAIN; NERVE CELL;

ANIMALS; BINDING SITES; CELLS, CULTURED; DOSE-RESPONSE RELATIONSHIP, DRUG; INDOLES; MICE; MICE, INBRED STRAINS; NEURONS; RECEPTORS, SEROTONIN; SEROTONIN ANTAGONISTS; SULFONAMIDES;

EID: 0029670468     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/0014-2999(95)00786-5     Document Type: Article

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