The design of non-peptide human Bradykinin B2 receptor antagonists employing the benzodiazepine peptidomimetic scaffold

Bioorganic and Medicinal Chemistry Letters

Volumn 9, Issue 3, 1999, Pages 463-468

  Dziadulewicz, Edward K ^a   Brown, Michael C ^a,c   Dunstan, Andrew R ^a,d   Lee, Wai ^a   Said, Najeeb B ^b,e   Garratt, Peter J ^b  

^a Novatis Inst for Medical Sciences   (United Kingdom)

^b UNIVERSITY COLLEGE LONDON   (United Kingdom)

^c DUPONT COMPANY   (United States)

^d NOVARTIS HORSHAM RESEARCH CENTRE   (United Kingdom)

^e INSTITUTO DE QUÍMICA ORGÁNICA GENERAL   (Spain)

Author keywords

[No Author keywords available]

Indexed keywords

BENZODIAZEPINE; BRADYKININ B2 RECEPTOR AGONIST; ICATIBANT;

ARTICLE; DRUG DESIGN; DRUG MECHANISM; DRUG RECEPTOR BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; STRUCTURE ANALYSIS;

BRADYKININ; DRUG DESIGN; HUMANS; MOLECULAR MIMICRY; RECEPTOR, BRADYKININ B2; RECEPTORS, BRADYKININ;

EID: 0033535143     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(99)00015-3     Document Type: Article

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