Novel series of O-substituted 8-quinolines and 4-benzothiazoles as potent antagonists of the bradykinin B2 receptors

Bioorganic and Medicinal Chemistry Letters

Volumn 9, Issue 3, 1999, Pages 327-332

  Heitsch, Holger ^a   Wagner, Adalbert ^a   Schölkens, Bernward A ^a   Wirth, Klaus ^a  

^a SANOFI   (France)

Author keywords

[No Author keywords available]

Indexed keywords

BENZOTHIAZOLE DERIVATIVE; BRADYKININ B2 RECEPTOR ANTAGONIST; QUINOLINE DERIVATIVE;

ARTICLE; BINDING AFFINITY; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; HUMAN; NONHUMAN; STRUCTURE ACTIVITY RELATION;

BENZOTHIAZOLES; QUINOLINES; RECEPTOR, BRADYKININ B2; RECEPTORS, BRADYKININ; STRUCTURE-ACTIVITY RELATIONSHIP; THIAZOLES;

EID: 0033535065     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(98)00736-7     Document Type: Article

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