Effect of the amide fragment on 5-HT(1A) receptor activity of some analogs of MP 3022

Polish Journal of Pharmacology

Volumn 51, Issue 5, 1999, Pages 415-421

  Paluchowska, Maria H ^a   Charakchieva Minol, Sijka ^a   Tatarczyńska, Ewa ^a   Kłodzińska, Aleksandra ^a  

^a INSTITUTE OF PHARMACOLOGY   (Poland)

Author keywords

5 HT(1A) ligands; Structure activity relationship

Indexed keywords

1 [3 (1 BENZOTRIAZOLYL)PROPYL] 4 (2 METHOXYPHENYL)PIPERAZINE; 2 DIPROPYLAMINO 8 HYDROXYTETRALIN; AMIDE; SEROTONIN 1A AGONIST; SEROTONIN 1A ANTAGONIST; SEROTONIN 1A RECEPTOR; SEROTONIN 2A AGONIST; SEROTONIN 2A ANTAGONIST; SEROTONIN 2A RECEPTOR; SEROTONIN AGONIST; SEROTONIN ANTAGONIST; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ARTICLE; BINDING AFFINITY; CHEMICAL STRUCTURE; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; DRUG SYNTHESIS; IN VITRO STUDY; IN VIVO STUDY; INTRAPERITONEAL DRUG ADMINISTRATION; MALE; NONHUMAN; RADIOASSAY; RAT; RECEPTOR AFFINITY; STRUCTURE ACTIVITY RELATION; SUBCUTANEOUS DRUG ADMINISTRATION;

AMIDES; ANIMALS; BEHAVIOR, ANIMAL; BRAIN; MALE; PIPERAZINES; RATS; RATS, WISTAR; RECEPTOR, SEROTONIN, 5-HT2A; RECEPTORS, SEROTONIN; RECEPTORS, SEROTONIN, 5-HT1; SEROTONIN AGENTS; SEROTONIN ANTAGONISTS; STRUCTURE-ACTIVITY RELATIONSHIP; TRIAZOLES;

EID: 0032708560     PISSN: 12306002     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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