An Advanced Tool to Interrogate BRD9

Journal of Medicinal Chemistry

Volumn 59, Issue 10, 2016, Pages 4459-4461

  Karim, Rezaul M ^a,b   Schönbrunn, Ernst ^a,b  

^a H LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE   (United States)

^b UNIVERSITY OF SOUTH FLORIDA   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

BI 9564; BROMODOMAIN CONTAINING PROTEIN 9; BROMODOMAIN INHIBITOR; PROTEIN; UNCLASSIFIED DRUG; BENZYLAMINE DERIVATIVE; BI-9564; BRD9 PROTEIN, HUMAN; MOLECULAR LIBRARY; NAPHTHYRIDINE DERIVATIVE; TRANSCRIPTION FACTOR;

CHROMATIN ASSEMBLY AND DISASSEMBLY; CONFORMATIONAL TRANSITION; DRUG TOLERANCE; GENETIC TRANSCRIPTION; HUMAN; NONHUMAN; PHARMACOPHORE; PROTEIN BINDING; PROTEIN FUNCTION; REVIEW; STRUCTURE ACTIVITY RELATION; ANTAGONISTS AND INHIBITORS; CHEMICAL STRUCTURE; CHEMISTRY; METABOLISM; MOLECULAR LIBRARY; MOLECULAR MODEL; PHARMACOLOGY;

BENZYLAMINES; HUMANS; MODELS, MOLECULAR; MOLECULAR STRUCTURE; NAPHTHYRIDINES; SMALL MOLECULE LIBRARIES; TRANSCRIPTION FACTORS;

EID: 84971597928     PISSN: 00222623     EISSN: 15204804     Source Type: Journal    
DOI: 10.1021/acs.jmedchem.6b00550     Document Type: Review

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