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Volumn 6, Issue 7, 2015, Pages 1381-1386

Design and synthesis of potent and selective inhibitors of BRD7 and BRD9 bromodomains

(10) Hay, Duncan A a,b Rogers, Catherine M b,c Fedorov, Oleg b,c Tallant, Cynthia b,c Martin, Sarah b,c Monteiro, Octovia P b,c Müller, Susanne b,c Knapp, Stefan b,c Schofield, Christopher J a Brennan, Paul E b,c

a UNIVERSITY OF OXFORD (United Kingdom)

b UNIVERSITY OF OXFORD (United Kingdom)

c UNIVERSITY OF OXFORD (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

BARRIER TO AUTOINTEGRATION FACTOR; BRD7 PROTEIN; BRD9 PROTEIN; BROMODOMAIN INHIBITOR; GSK 2801; HISTONE ACETYLTRANSFERASE PCAF; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; BINDING SITE; CELL MEMBRANE PERMEABILITY; CHEMICAL STRUCTURE; CYCLOADDITION; ENANTIOSELECTIVITY; ENTROPY; HUMAN; HYDROPHILICITY; IC50; LIPOPHILICITY; PRIORITY JOURNAL; PROTEIN BINDING; PROTEIN PROTEIN INTERACTION; SYNTHESIS;

EID: 84936874034 PISSN: 20402503 EISSN: 20402511 Source Type: Journal
DOI: 10.1039/c5md00152h Document Type: Article

Times cited : (63)

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