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Bioorganic and Medicinal Chemistry Letters

Volumn 26, Issue 11, 2016, Pages 2589-2593

Facile and efficient synthesis and biological evaluation of 4-anilinoquinazoline derivatives as EGFR inhibitors

(7) Wang, Zheng a Wu, Xue c Wang, Li a Zhang, Jiao a Liu, Jianli b Song, Zhongxing a Tang, Zhishu a

a SHAANXI UNIVERSITY OF CHINESE MEDICINE (China)

b NORTHWEST UNIVERSITY (China)

c FOURTH MILITARY MEDICAL UNIVERSITY (China)

Author keywords

4 Anilinoquinazoline; MTT assay; Synthesis; Western blotting analysis

Indexed keywords

4 ANILINOQUINAZOLINE DERIVATIVE; ANTINEOPLASTIC AGENT; GEFITINIB; METHYL GROUP; QUINAZOLINE; QUINAZOLINE DERIVATIVE; UNCLASSIFIED DRUG; VASCULOTROPIN INHIBITOR; EPIDERMAL GROWTH FACTOR RECEPTOR; PROTEIN KINASE INHIBITOR;

ANTINEOPLASTIC ACTIVITY; ARTICLE; CANCER CELL LINE; CONTROLLED STUDY; DRUG DESIGN; DRUG INHIBITION; DRUG POTENCY; DRUG SYNTHESIS; HEPG2 CELL LINE; HUMAN; HUMAN CELL; HUMAN CELL CULTURE; WESTERN BLOTTING; ANTAGONISTS AND INHIBITORS; CELL PROLIFERATION; CHEMICAL STRUCTURE; CHEMISTRY; DOSE RESPONSE; DRUG EFFECTS; DRUG SCREENING; METABOLISM; STRUCTURE ACTIVITY RELATION; SYNTHESIS; TUMOR CELL LINE;

ANTINEOPLASTIC AGENTS; CELL LINE, TUMOR; CELL PROLIFERATION; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG SCREENING ASSAYS, ANTITUMOR; HUMANS; MOLECULAR STRUCTURE; PROTEIN KINASE INHIBITORS; QUINAZOLINES; RECEPTOR, EPIDERMAL GROWTH FACTOR; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84964587681 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2016.04.032 Document Type: Article

Times cited : (21)

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