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Volumn 21, Issue 24, 2013, Pages 7858-7873

Investigation of quinazolines as inhibitors of breast cancer resistance protein (ABCG2)

(3) Juvale, Kapil a Gallus, Jennifer a Wiese, Michael a

Author keywords

ATP binding cassette (ABC) transporter; Breast cancer resistance protein (BCRP ABCG2); Hoechst 33342 accumulation assay; Multidrug resistance; Quinazolines

Indexed keywords

1,2,3,4,6,7,12,12A OCTAHYDRO 6 ISOBUTYL 9 METHOXY 1,4 DIOXOPYRAZINO[1',2':1,6]PYRIDO[3,4 B]INDOLE 3 PROPANOIC ACID TERT BUTYL ESTER; 2 (3,4 DIMETHOXYPHENYL) N (3 NITROPHENYL)QUINAZOLIN 4 AMINE; 2 (3,4 DIMETHOXYPHENYL) N (4 NITROPHENYL)QUINAZOLIN 4 AMINE; 2 (3,4 DIMETHOXYPHENYL) N [3 (TRIFLUOROMETHYL)PHENYL]QUINAZOLIN 4 AMINE; 3 [(2 PHENYLQUINAZOLIN 4 YL)AMINO]PHENOL; 3 [[2 (3,4 DIMETHOXYPHENYL)QUINAZOLIN 4 YL]AMINO]PHENOL; 3,3' [(6,7 DIMETHOXYQUINAZOLINE 2,4 DIYL)BIS(AZANEDIYL)]DIBENZONITRILE; 6,7 DIMETHOXY N (3 NITROPHENYL)QUINAZOLIN 4 AMINE; 6,7 DIMETHOXY N2,N4 BIS (3 NITROPHENYL)QUINAZOLINE 2,4 DIAMINE; 6,7 DIMETHOXY N2,N4 BIS [3(TRIFLUOROMETHYL)PHENYL]QUINAZOLINE 2,4 DIAMINE; 6,7 DIMETHOXY N2,N4 BIS(3 NITROPHENYL)QUINAZOLINE 2,4 DIAMINE; BREAST CANCER RESISTANCE PROTEIN; CYCLOSPORIN A; GEFITINIB; MULTIDRUG RESISTANCE PROTEIN; MULTIDRUG RESISTANCE PROTEIN 1; N (3 BROMOPHENYL) 2 (3,4 DIMETHOXYPHENYL)QUINAZOLIN 4 AMINE; N (3 BROMOPHENYL) 2 PHENYLQUINAZOLIN 4 AMINE; N (3 NITROPHENYL) 2 PHENYLQUINAZOLIN 4 AMINE; N (3 NITROPHENYL)QUINAZOLIN 4 AMINE; N (3,4 DIMETHOXYPHENYL) 2 PHENYLQUINAZOLIN 4 AMINE; N,2 BIS (3,4 DIMETHOXYPHENYL)QUINAZOLIN 4 AMINE; N2,N4 BIS (3,4 DIMETHOXYPHENYL) 6,7 DIMETHOXYQUINAZOLINE 2,4 DIAMINE; N2,N4 BIS(3 BROMOPHENYL) 6,7 DIMETHOXYQUINAZOLINE 2,4 DIAMINE; PROTEIN INHIBITOR; QUINAZOLINE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CANCER CELL CULTURE; CANCER INHIBITION; CONTROLLED STUDY; DRUG CYTOTOXICITY; DRUG DETERMINATION; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; FEMALE; HUMAN; HUMAN CELL; IC 50; NONHUMAN; PROTEIN EXPRESSION; PROTEIN SYNTHESIS INHIBITION; STRUCTURE ACTIVITY RELATION; SUBSTITUTION REACTION;

ATP BINDING CASSETTE (ABC) TRANSPORTER; BREAST CANCER RESISTANCE PROTEIN (BCRP/ABCG2); HOECHST 33342 ACCUMULATION ASSAY; MULTIDRUG RESISTANCE; QUINAZOLINES;

ANIMALS; ATP-BINDING CASSETTE TRANSPORTERS; CELLS, CULTURED; DOGS; DOSE-RESPONSE RELATIONSHIP, DRUG; HUMANS; MOLECULAR STRUCTURE; NEOPLASM PROTEINS; QUINAZOLINES; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84888435947 PISSN: 09680896 EISSN: 14643391 Source Type: Journal
DOI: 10.1016/j.bmc.2013.10.007 Document Type: Article

Times cited : (91)

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