메뉴 건너뛰기




Volumn 2, Issue 11, 2015, Pages 1806-1813

The Sigma-2 Receptor and Progesterone Receptor Membrane Component 1 are Different Binding Sites Derived From Independent Genes

Author keywords

Clustered regularly interspaced short palindromic repeats (CRISPR) Cas9 knockout; Progesterone receptor membrane component 1 (PGRMC1); Sigma 2 receptor (S2R); 125I Iodoazido fenpropimorph ( 125I IAF); 3H 1,3 Di o tolylguanidine ( 3H DTG)

Indexed keywords

1,3 DI 2 TOLYLGUANIDINE; GUANIDINE DERIVATIVE; HALOPERIDOL; IODINE 125; LIPOFECTAMINE; PENTAZOCINE; PROGESTERONE BINDING PROTEIN; PROGESTERONE RECEPTOR; SIGMA 2 OPIATE RECEPTOR; UNCLASSIFIED DRUG; MEMBRANE PROTEIN; PGRMC1 PROTEIN, HUMAN; PROGESTERONE; PROTEIN BINDING; SIGMA OPIATE RECEPTOR; SIGMA-2 RECEPTOR;

EID: 84958834594     PISSN: None     EISSN: 23523964     Source Type: Journal    
DOI: 10.1016/j.ebiom.2015.10.017     Document Type: Article
Times cited : (82)

References (38)
  • 1
    • 84927556019 scopus 로고    scopus 로고
    • Elements in support of the 'non-identity' of the PGRMC1 protein with the sigma2 receptor
    • Abate C., Niso M., Infantino V., Menga A., Berardi F. Elements in support of the 'non-identity' of the PGRMC1 protein with the sigma2 receptor. Eur. J. Pharmacol. 2015, 758:16-23.
    • (2015) Eur. J. Pharmacol. , vol.758 , pp. 16-23
    • Abate, C.1    Niso, M.2    Infantino, V.3    Menga, A.4    Berardi, F.5
  • 2
    • 84879292172 scopus 로고    scopus 로고
    • Progesterone antagonism of neurite outgrowth depends on microglial activation via Pgrmc1/S2R
    • Bali N., Arimoto J.M., Morgan T.E., Finch C.E. Progesterone antagonism of neurite outgrowth depends on microglial activation via Pgrmc1/S2R. Endocrinology 2013, 154:2468-2480.
    • (2013) Endocrinology , vol.154 , pp. 2468-2480
    • Bali, N.1    Arimoto, J.M.2    Morgan, T.E.3    Finch, C.E.4
  • 3
    • 0024553608 scopus 로고
    • Evidence for a multi-site model of the rat brain sigma receptor
    • Bowen W.D., Hellewell S.B., Mcgarry K.A. Evidence for a multi-site model of the rat brain sigma receptor. Eur. J. Pharmacol. 1989, 163:309-318.
    • (1989) Eur. J. Pharmacol. , vol.163 , pp. 309-318
    • Bowen, W.D.1    Hellewell, S.B.2    Mcgarry, K.A.3
  • 4
    • 33646815696 scopus 로고    scopus 로고
    • The sigma-2 receptor agonist PB28 inhibits calcium release from the endoplasmic reticulum of SK-N-SH neuroblastoma cells
    • Cassano G., Gasparre G., Contino M., Niso M., Berardi F., Perrone R., Colabufo N.A. The sigma-2 receptor agonist PB28 inhibits calcium release from the endoplasmic reticulum of SK-N-SH neuroblastoma cells. Cell Calcium 2006, 40:23-28.
    • (2006) Cell Calcium , vol.40 , pp. 23-28
    • Cassano, G.1    Gasparre, G.2    Contino, M.3    Niso, M.4    Berardi, F.5    Perrone, R.6    Colabufo, N.A.7
  • 8
    • 0036141493 scopus 로고    scopus 로고
    • Sigma-2 receptor agonists activate a novel apoptotic pathway and potentiate antineoplastic drugs in breast tumor cell lines
    • Crawford K.W., Bowen W.D. Sigma-2 receptor agonists activate a novel apoptotic pathway and potentiate antineoplastic drugs in breast tumor cell lines. Cancer Res. 2002, 62:313-322.
    • (2002) Cancer Res. , vol.62 , pp. 313-322
    • Crawford, K.W.1    Bowen, W.D.2
  • 9
    • 84913594397 scopus 로고    scopus 로고
    • Genome editing. The new frontier of genome engineering with CRISPR-Cas9
    • Doudna J.A., Charpentier E. Genome editing. The new frontier of genome engineering with CRISPR-Cas9. Science 2014, 346:1258096.
    • (2014) Science , vol.346 , pp. 1258096
    • Doudna, J.A.1    Charpentier, E.2
  • 10
    • 46849119587 scopus 로고    scopus 로고
    • Probing the steroid binding domain-like I (SBDLI) of the sigma-1 receptor binding site using N-substituted photoaffinity labels
    • Fontanilla D., Hajipour A.R., Pal A., Chu U.B., Arbabian M., Ruoho A.E. Probing the steroid binding domain-like I (SBDLI) of the sigma-1 receptor binding site using N-substituted photoaffinity labels. Biochemistry 2008, 47:7205-7217.
    • (2008) Biochemistry , vol.47 , pp. 7205-7217
    • Fontanilla, D.1    Hajipour, A.R.2    Pal, A.3    Chu, U.B.4    Arbabian, M.5    Ruoho, A.E.6
  • 11
  • 12
    • 2942578089 scopus 로고    scopus 로고
    • Sigma-2 receptors are specifically localized to lipid rafts in rat liver membranes
    • Gebreselassie D., Bowen W.D. Sigma-2 receptors are specifically localized to lipid rafts in rat liver membranes. Eur. J. Pharmacol. 2004, 493:19-28.
    • (2004) Eur. J. Pharmacol. , vol.493 , pp. 19-28
    • Gebreselassie, D.1    Bowen, W.D.2
  • 13
  • 15
    • 0025180755 scopus 로고
    • A sigma-like binding site in rat pheochromocytoma (PC12) cells: decreased affinity for (+)-benzomorphans and lower molecular weight suggest a different sigma receptor form from that of guinea pig brain
    • Hellewell S.B., Bowen W.D. A sigma-like binding site in rat pheochromocytoma (PC12) cells: decreased affinity for (+)-benzomorphans and lower molecular weight suggest a different sigma receptor form from that of guinea pig brain. Brain Res. 1990, 527:244-253.
    • (1990) Brain Res. , vol.527 , pp. 244-253
    • Hellewell, S.B.1    Bowen, W.D.2
  • 16
    • 0028180570 scopus 로고
    • Rat liver and kidney contain high densities of sigma 1 and sigma 2 receptors: characterization by ligand binding and photoaffinity labeling
    • Hellewell S.B., Bruce A., Feinstein G., Orringer J., Williams W., Bowen W.D. Rat liver and kidney contain high densities of sigma 1 and sigma 2 receptors: characterization by ligand binding and photoaffinity labeling. Eur. J. Pharmacol. 1994, 268:9-18.
    • (1994) Eur. J. Pharmacol. , vol.268 , pp. 9-18
    • Hellewell, S.B.1    Bruce, A.2    Feinstein, G.3    Orringer, J.4    Williams, W.5    Bowen, W.D.6
  • 18
    • 0023161247 scopus 로고
    • 3H]SKF 10047 binding sites in rat brain membranes: evidence of multiplicity
    • 3H]SKF 10047 binding sites in rat brain membranes: evidence of multiplicity. Eur. J. Pharmacol. 1987, 136:231-234.
    • (1987) Eur. J. Pharmacol. , vol.136 , pp. 231-234
    • Itzhak, Y.1
  • 19
    • 0025099110 scopus 로고
    • Clorgyline displays high affinity for sigma binding sites in C57BL/6 mouse brain
    • Itzhak Y., Kassim C.O. Clorgyline displays high affinity for sigma binding sites in C57BL/6 mouse brain. Eur. J. Pharmacol. 1990, 176:107-108.
    • (1990) Eur. J. Pharmacol. , vol.176 , pp. 107-108
    • Itzhak, Y.1    Kassim, C.O.2
  • 22
    • 0017064976 scopus 로고
    • The effects of morphine- and nalorphine-like drugs in the nondependent and morphine-dependent chronic spinal dog
    • Martin W.R., Eades C.G., Thompson J.A., Huppler R.E., Gilbert P.E. The effects of morphine- and nalorphine-like drugs in the nondependent and morphine-dependent chronic spinal dog. J. Pharmacol. Exp. Ther. 1976, 197:517-532.
    • (1976) J. Pharmacol. Exp. Ther. , vol.197 , pp. 517-532
    • Martin, W.R.1    Eades, C.G.2    Thompson, J.A.3    Huppler, R.E.4    Gilbert, P.E.5
  • 23
    • 84893187276 scopus 로고    scopus 로고
    • Sigma (sigma) receptors as potential therapeutic targets to mitigate psychostimulant effects
    • Matsumoto R.R., Nguyen L., Kaushal N., Robson M.J. Sigma (sigma) receptors as potential therapeutic targets to mitigate psychostimulant effects. Adv. Pharmacol. 2014, 69:323-386.
    • (2014) Adv. Pharmacol. , vol.69 , pp. 323-386
    • Matsumoto, R.R.1    Nguyen, L.2    Kaushal, N.3    Robson, M.J.4
  • 24
    • 84885646346 scopus 로고    scopus 로고
    • Progesterone receptor membrane component 1/Sigma-2 receptor associates with MAP1LC3B and promotes autophagy
    • Mir S.U., Schwarze S.R., Jin L., Zhang J., Friend W., Miriyala S., St Clair D., Craven R.J. Progesterone receptor membrane component 1/Sigma-2 receptor associates with MAP1LC3B and promotes autophagy. Autophagy 2013, 9:1566-1578.
    • (2013) Autophagy , vol.9 , pp. 1566-1578
    • Mir, S.U.1    Schwarze, S.R.2    Jin, L.3    Zhang, J.4    Friend, W.5    Miriyala, S.6    St Clair, D.7    Craven, R.J.8
  • 25
    • 0025951663 scopus 로고
    • Interaction of forskolin with the P-glycoprotein multidrug transporter
    • Morris D.I., Speicher L.A., Ruoho A.E., Tew K.D., Seamon K.B. Interaction of forskolin with the P-glycoprotein multidrug transporter. Biochemistry 1991, 30:8371-8379.
    • (1991) Biochemistry , vol.30 , pp. 8371-8379
    • Morris, D.I.1    Speicher, L.A.2    Ruoho, A.E.3    Tew, K.D.4    Seamon, K.B.5
  • 26
    • 84941564384 scopus 로고    scopus 로고
    • Characterization of CM572, a selective irreversible partial agonist of the Sigma-2 receptor with antitumor activity
    • Nicholson H., Comeau A., Mesangeau C., McCurdy C.R., Bowen W.D. Characterization of CM572, a selective irreversible partial agonist of the Sigma-2 receptor with antitumor activity. J. Pharmacol. Exp. Ther. 2015.
    • (2015) J. Pharmacol. Exp. Ther.
    • Nicholson, H.1    Comeau, A.2    Mesangeau, C.3    McCurdy, C.R.4    Bowen, W.D.5
  • 28
    • 38549114147 scopus 로고    scopus 로고
    • Progesterone receptor membrane component-1 (PGRMC1) is the mediator of progesterone's antiapoptotic action in spontaneously immortalized granulosa cells as revealed by PGRMC1 small interfering ribonucleic acid treatment and functional analysis of PGRMC1 mutations
    • Peluso J.J., Romak J., LIU X. Progesterone receptor membrane component-1 (PGRMC1) is the mediator of progesterone's antiapoptotic action in spontaneously immortalized granulosa cells as revealed by PGRMC1 small interfering ribonucleic acid treatment and functional analysis of PGRMC1 mutations. Endocrinology 2008, 149:534-543.
    • (2008) Endocrinology , vol.149 , pp. 534-543
    • Peluso, J.J.1    Romak, J.2    LIU, X.3
  • 31
    • 84905262730 scopus 로고    scopus 로고
    • Improved vectors and genome-wide libraries for CRISPR screening
    • Sanjana N.E., Shalem O., Zhang F. Improved vectors and genome-wide libraries for CRISPR screening. Nat. Methods 2014, 11:783-784.
    • (2014) Nat. Methods , vol.11 , pp. 783-784
    • Sanjana, N.E.1    Shalem, O.2    Zhang, F.3
  • 32
    • 0027471841 scopus 로고
    • Sigma receptor-active neuroleptics are cytotoxic to C6 glioma Cells in culture
    • Vilner B.J., Bowen W.D. Sigma receptor-active neuroleptics are cytotoxic to C6 glioma Cells in culture. Eur. J. Pharmacol. 1993, 244:199-201.
    • (1993) Eur. J. Pharmacol. , vol.244 , pp. 199-201
    • Vilner, B.J.1    Bowen, W.D.2
  • 33
    • 0034053453 scopus 로고    scopus 로고
    • Modulation of cellular calcium by sigma-2 receptors: release from intracellular stores in human SK-N-SH neuroblastoma cells
    • Vilner B.J., Bowen W.D. Modulation of cellular calcium by sigma-2 receptors: release from intracellular stores in human SK-N-SH neuroblastoma cells. J. Pharmacol. Exp. Ther. 2000, 292:900-911.
    • (2000) J. Pharmacol. Exp. Ther. , vol.292 , pp. 900-911
    • Vilner, B.J.1    Bowen, W.D.2
  • 34
    • 0028795145 scopus 로고
    • Sigma-1 and sigma-2 receptors are expressed in a wide variety of human and rodent tumor cell lines
    • Vilner B.J., John C.S., Bowen W.D. Sigma-1 and sigma-2 receptors are expressed in a wide variety of human and rodent tumor cell lines. Cancer Res. 1995, 55:408-413.
    • (1995) Cancer Res. , vol.55 , pp. 408-413
    • Vilner, B.J.1    John, C.S.2    Bowen, W.D.3
  • 35
    • 0011190242 scopus 로고
    • 1,3-Di(2-[5-3H]tolyl)guanidine: a selective ligand that labels sigma-type receptors for psychotomimetic opiates and antipsychotic drugs
    • Weber E., Sonders M., Quarum M., Mclean S., Pou S., Keana J.F. 1,3-Di(2-[5-3H]tolyl)guanidine: a selective ligand that labels sigma-type receptors for psychotomimetic opiates and antipsychotic drugs. Proc. Natl. Acad. Sci. U. S. A. 1986, 83:8784-8788.
    • (1986) Proc. Natl. Acad. Sci. U. S. A. , vol.83 , pp. 8784-8788
    • Weber, E.1    Sonders, M.2    Quarum, M.3    Mclean, S.4    Pou, S.5    Keana, J.F.6


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.