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Volumn 23, Issue 9, 2015, Pages 2195-2203

Structure-activity relationships of substituted 1H-indole-2-carboxamides as CB1 receptor allosteric modulators

(8) Nguyen, Thuy a German, Nadezhda a Decker, Ann M a Li, Jun Xu b Wiley, Jenny L a Thomas, Brian F a Kenakin, Terry P c Zhang, Yanan a

a RTI INTERNATIONAL (United States)

b UNIVERSITY AT BUFFALO (United States)

c UNIVERSITY OF NORTH CAROLINA SCHOOL OF MEDICINE (United States)

Author keywords

Allosteric modulators; CB1 receptor; Org compounds; Structure activity relationship

Indexed keywords

AMIDE; CANNABINOID 1 RECEPTOR; CANNABINOID 2 RECEPTOR; INDOLE DERIVATIVE;

ALLOSTERISM; ANIMAL; ANTAGONISTS AND INHIBITORS; CHEMICAL STRUCTURE; CHEMISTRY; CHO CELL LINE; CRICETULUS; DOSE RESPONSE; DRUG EFFECTS; HUMAN; METABOLISM; STRUCTURE ACTIVITY RELATION; SYNTHESIS;

ALLOSTERIC REGULATION; AMIDES; ANIMALS; CHO CELLS; CRICETULUS; DOSE-RESPONSE RELATIONSHIP, DRUG; HUMANS; INDOLES; MOLECULAR STRUCTURE; RECEPTOR, CANNABINOID, CB1; RECEPTOR, CANNABINOID, CB2; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84940006834 PISSN: 09680896 EISSN: 14643391 Source Type: Journal
DOI: 10.1016/j.bmc.2015.02.058 Document Type: Article

Times cited : (31)

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