SCOPUS 정보 검색 플랫폼

Volumn 23, Issue 10, 2015, Pages 2480-2488

Structure activity relationship of selective GABA uptake inhibitors

(10) Vogensen, Stine B a Jørgensen, Lars a Madsen, Karsten K a Jurik, Andreas b Borkar, Nrupa a Rosatelli, Emiliano c Nielsen, Birgitte a Ecker, Gerhard F b Schousboe, Arne a Clausen, Rasmus P a

a UNIVERSITY OF COPENHAGEN (Denmark)

b UNIVERSITY OF VIENNA (Austria)

c UNIVERSITY OF PERUGIA (Italy)

Author keywords

BGT 1; GABA uptake; Inhibitors; mGAT2; Tiagabine

Indexed keywords

4 AMINOBUTYRIC ACID CARRIER; 4 AMINOBUTYRIC ACID RECEPTOR STIMULATING AGENT; 4 AMINOBUTYRIC ACID UPTAKE INHIBITOR; AMINO ACID; BETAINE PLASMA MEMBRANE TRANSPORT PROTEINS; CARRIER PROTEIN; ISOPROTEIN; LIGAND; NIPECOTIC ACID DERIVATIVE; TIAGABINE;

ANIMAL; ANTAGONISTS AND INHIBITORS; CHEMICAL STRUCTURE; CHEMISTRY; HEK293 CELL LINE; HUMAN; MOLECULAR DOCKING; MOUSE; STRUCTURE ACTIVITY RELATION; SYNTHESIS;

AMINO ACIDS; ANIMALS; CARRIER PROTEINS; GABA AGONISTS; GABA PLASMA MEMBRANE TRANSPORT PROTEINS; GABA UPTAKE INHIBITORS; HEK293 CELLS; HUMANS; LIGANDS; MICE; MOLECULAR DOCKING SIMULATION; MOLECULAR STRUCTURE; NIPECOTIC ACIDS; PROTEIN ISOFORMS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84937760304 PISSN: 09680896 EISSN: 14643391 Source Type: Journal
DOI: 10.1016/j.bmc.2015.03.060 Document Type: Article

Times cited : (30)

References (33)

1
- 84937772561
- Elsevier
- S.J. Enna GABA, Adv. Pharmacol. Vol. 54 2006 Elsevier
- (2006) GABA, Adv. Pharmacol. , vol.54
- Enna, S.J.¹

2
- 0011148741
- Raven Press New York
- G. Nistico, P.L. Morselli, K.G. Lloyd, R.G. Fariello, and J. Engel Neurotransmitters, Seizures, and Epilepsy III 1986 Raven Press New York
- (1986) Neurotransmitters, Seizures, and Epilepsy III
- Nistico, G.¹ Morselli, P.L.² Lloyd, K.G.³ Fariello, R.G.⁴ Engel, J.⁵

3
- 0038677031
- H. Ashton, and A.H. Young J. Psychopharmacol. 17 2003 174
- (2003) J. Psychopharmacol. , vol.17 , pp. 174
- Ashton, H.¹ Young, A.H.²

4
- 79959525532
- K.K. Madsen, B. Ebert, O.M. Larsson, R.P. Clausen, A. Schousboe, and H.S. White J. Pharmacol. Exp. Ther. 338 2011 214
- (2011) J. Pharmacol. Exp. Ther. , vol.338 , pp. 214
- Madsen, K.K.¹ Ebert, B.² Larsson, O.M.³ Clausen, R.P.⁴ Schousboe, A.⁵ White, H.S.⁶

5
- 64349115311
- K.K. Madsen, R.P. Clausen, O.M. Larsson, P. Krogsgaard-Larsen, A. Schousboe, and H. Steve White J. Neurochem. 109 2009 139
- (2009) J. Neurochem. , vol.109 , pp. 139
- Madsen, K.K.¹ Clausen, R.P.² Larsson, O.M.³ Krogsgaard-Larsen, P.⁴ Schousboe, A.⁵ Steve White, H.⁶

6
- 0030272426
- L.A. Borden Neurochem. Int. 29 1996 335
- (1996) Neurochem. Int. , vol.29 , pp. 335
- Borden, L.A.¹

7
- 33748658838
- S. Hog, J.R. Greenwood, K.B. Madsen, O.M. Larsson, B. Frolund, A. Schousboe, P. Krogsgaard-Larsen, and R.P. Clausen Curr. Top. Med. Chem. 6 2006 1861
- (2006) Curr. Top. Med. Chem. , vol.6 , pp. 1861
- Hog, S.¹ Greenwood, J.R.² Madsen, K.B.³ Larsson, O.M.⁴ Frolund, B.⁵ Schousboe, A.⁶ Krogsgaard-Larsen, P.⁷ Clausen, R.P.⁸

8
- 0023577566
- P. Krogsgaard-Larsen, E. Falch, O.M. Larsson, and A. Schousboe Epilepsy Res. 1 1987 77
- (1987) Epilepsy Res. , vol.1 , pp. 77
- Krogsgaard-Larsen, P.¹ Falch, E.² Larsson, O.M.³ Schousboe, A.⁴

9
- 0033864480
- P. Krogsgaard-Larsen, B. Frolund, and K. Frydenvang Curr. Pharm. Des. 6 2000 1193
- (2000) Curr. Pharm. Des. , vol.6 , pp. 1193
- Krogsgaard-Larsen, P.¹ Frolund, B.² Frydenvang, K.³

10
- 84875137124
- S.B. Vogensen, L. Jørgensen, K.K. Madsen, N. Borkar, P. Wellendorph, J. Skovgaard-Petersen, A. Schousboe, H.S. White, P. Krogsgaard-Larsen, and R.P. Clausen J. Med. Chem. 56 2013 2160
- (2013) J. Med. Chem. , vol.56 , pp. 2160
- Vogensen, S.B.¹ Jørgensen, L.² Madsen, K.K.³ Borkar, N.⁴ Wellendorph, P.⁵ Skovgaard-Petersen, J.⁶ Schousboe, A.⁷ White, H.S.⁸ Krogsgaard-Larsen, P.⁹ Clausen, R.P.¹⁰

11
- 33744462712
- R.P. Clausen, K. Madsen, O.M. Larsson, B. Frølund, P. Krogsgaard-Larsen, and A. Schousboe Adv. Pharmacol. 54 2006 265
- (2006) Adv. Pharmacol. , vol.54 , pp. 265
- Clausen, R.P.¹ Madsen, K.² Larsson, O.M.³ Frølund, B.⁴ Krogsgaard-Larsen, P.⁵ Schousboe, A.⁶

12
- 19944428485
- R.P. Clausen, E.K. Moltzen, J. Perregaard, S.M. Lenz, C. Sanchez, E. Falch, B. Frolund, T. Bolvig, A. Sarup, O.M. Larsson, A. Schousboe, and P. Krogsgaard-Larsen Bioorg. Med. Chem. 13 2005 895
- (2005) Bioorg. Med. Chem. , vol.13 , pp. 895
- Clausen, R.P.¹ Moltzen, E.K.² Perregaard, J.³ Lenz, S.M.⁴ Sanchez, C.⁵ Falch, E.⁶ Frolund, B.⁷ Bolvig, T.⁸ Sarup, A.⁹ Larsson, O.M.¹⁰ Schousboe, A.¹¹ Krogsgaard-Larsen, P.¹²

13
- 33645885629
- R.P. Clausen, B. Frolund, O.M. Larsson, A. Schousboe, P. Krogsgaard-Larsen, and H.S. White Neurochem. Int. 48 2006 637
- (2006) Neurochem. Int. , vol.48 , pp. 637
- Clausen, R.P.¹ Frolund, B.² Larsson, O.M.³ Schousboe, A.⁴ Krogsgaard-Larsen, P.⁵ White, H.S.⁶

14
- 0030760706
- M. Nakashita, K. Sasaki, N. Sakai, and N. Saito Neurosci. Res. 29 1997 87
- (1997) Neurosci. Res. , vol.29 , pp. 87
- Nakashita, M.¹ Sasaki, K.² Sakai, N.³ Saito, N.⁴

15
- 0036713897
- A. Berkessel, K. Glaubitz, and J. Lex Eur. J. Org. Chem. 2002 2948
- (2002) Eur. J. Org. Chem. , pp. 2948
- Berkessel, A.¹ Glaubitz, K.² Lex, J.³

16
- 0033539049
- L.J.S. Knutsen, K.E. Andersen, J. Lau, B.F. Lundt, R.F. Henry, H.E. Morton, L. Nærum, H. Petersen, H. Stephensen, P.D. Suzdak, M.D.B. Swedberg, C. Thomsen, and P.O. Sørensen J. Med. Chem. 42 1999 3447
- (1999) J. Med. Chem. , vol.42 , pp. 3447
- Knutsen, L.J.S.¹ Andersen, K.E.² Lau, J.³ Lundt, B.F.⁴ Henry, R.F.⁵ Morton, H.E.⁶ Nærum, L.⁷ Petersen, H.⁸ Stephensen, H.⁹ Suzdak, P.D.¹⁰ Swedberg, M.D.B.¹¹ Thomsen, C.¹² Sørensen, P.O.¹³

17
- 0026498594
- M.R. Pavia, S.J. Lobbestael, D. Nugiel, D.R. Mayhugh, V.E. Gregor, C.P. Taylor, R.D. Schwarz, L. Brahce, and M.G. Vartanian J. Med. Chem. 35 1992 4238
- (1992) J. Med. Chem. , vol.35 , pp. 4238
- Pavia, M.R.¹ Lobbestael, S.J.² Nugiel, D.³ Mayhugh, D.R.⁴ Gregor, V.E.⁵ Taylor, C.P.⁶ Schwarz, R.D.⁷ Brahce, L.⁸ Vartanian, M.G.⁹

18
- 0015379982
- S. Umio, I. Ueda, and H. Nojima J. Med. Chem. 15 1972 855
- (1972) J. Med. Chem. , vol.15 , pp. 855
- Umio, S.¹ Ueda, I.² Nojima, H.³

19
- 27944451724
- L.G. Ma, D.M. Du, and J.X. Xu J. Org. Chem. 70 2005 10155
- (2005) J. Org. Chem. , vol.70 , pp. 10155
- Ma, L.G.¹ Du, D.M.² Xu, J.X.³

20
- 0037324997
- M. Schinnerl, J.K. Murray, J.M. Langenhan, and S.H. Gellman Eur. J. Org. Chem. 2003 721
- (2003) Eur. J. Org. Chem. , pp. 721
- Schinnerl, M.¹ Murray, J.K.² Langenhan, J.M.³ Gellman, S.H.⁴

21
- 19944433063
- H.S. White, W.P. Watson, S.L. Hansen, S. Slough, J. Perregaard, A. Sarup, T. Bolvig, G. Petersen, O.M. Larsson, R.P. Clausen, B. Frølund, E. Falch, P. Krogsgaard-Larsen, and A. Schousboe J. Pharmacol. Exp. Ther. 312 2005 866
- (2005) J. Pharmacol. Exp. Ther. , vol.312 , pp. 866
- White, H.S.¹ Watson, W.P.² Hansen, S.L.³ Slough, S.⁴ Perregaard, J.⁵ Sarup, A.⁶ Bolvig, T.⁷ Petersen, G.⁸ Larsson, O.M.⁹ Clausen, R.P.¹⁰ Frølund, B.¹¹ Falch, E.¹² Krogsgaard-Larsen, P.¹³ Schousboe, A.¹⁴

22
- 0030955132
- C. Thomsen, P.O. Sørensen, and J. Egebjerg Br. J. Pharmacol. 120 1997 983
- (1997) Br. J. Pharmacol. , vol.120 , pp. 983
- Thomsen, C.¹ Sørensen, P.O.² Egebjerg, J.³

23
- 84973243729
- J.A. Murphy, K.A. Scott, R.S. Sinclair, C.G. Martin, A.R. Kennedy, and N. Lewis J. Chem. Soc., Perkin Trans. 1 2000 2385
- (2000) J. Chem. Soc., Perkin Trans. 1 , pp. 2385
- Murphy, J.A.¹ Scott, K.A.² Sinclair, R.S.³ Martin, C.G.⁴ Kennedy, A.R.⁵ Lewis, N.⁶

24
- 0033531676
- B.M. Trost, and J.D.J. Oslob Am. Chem. Soc. 121 1999 3057
- (1999) Am. Chem. Soc. , vol.121 , pp. 3057
- Trost, B.M.¹ Oslob, J.D.J.²

25
- 85077864655
- H.H. Massoudi, D. Cantacuzène, C. Wakselman, and C. Bouthier de la Tour Synthesis 1983 1010
- (1983) Synthesis , pp. 1010
- Massoudi, H.H.¹ Cantacuzène, D.² Wakselman, C.³ Bouthier De La Tour, C.⁴

26
- 84973230858
- R.A. Laskowski, M.W. MacArthur, D.S. Moss, and J.M. Thornton J. Appl. Cryst. 26 1993 283
- (1993) J. Appl. Cryst. , vol.26 , pp. 283
- Laskowski, R.A.¹ Macarthur, M.W.² Moss, D.S.³ Thornton, J.M.⁴

27
- 84887404259
- A. Penmatsa, K.H. Wang, and E. Gouaux Nature 503 2013 85
- (2013) Nature , vol.503 , pp. 85
- Penmatsa, A.¹ Wang, K.H.² Gouaux, E.³

28
- 79951747486
- A. Ray, E. Lindahl, and B. Wallner Bioinformatics 26 2010 3067
- (2010) Bioinformatics , vol.26 , pp. 3067
- Ray, A.¹ Lindahl, E.² Wallner, B.³

29
- 77954125609
- S. Skovstrup, O. Taboureau, H. Bräuner-Osborne, and F.S. Jørgensen ChemMedChem 5 2010 986
- (2010) ChemMedChem , vol.5 , pp. 986
- Skovstrup, S.¹ Taboureau, O.² Bräuner-Osborne, H.³ Jørgensen, F.S.⁴

30
- 84906282999
- T. Kobayashi, A. Suemasa, A. Igawa, S. Ide, H. Fukuda, H. Abe, M. Arisawa, M. Minami, and S. Shuto ACS Med. Chem. Lett. 5 2014 889
- (2014) ACS Med. Chem. Lett. , vol.5 , pp. 889
- Kobayashi, T.¹ Suemasa, A.² Igawa, A.³ Ide, S.⁴ Fukuda, H.⁵ Abe, H.⁶ Arisawa, M.⁷ Minami, M.⁸ Shuto, S.⁹

31
- 84918775764
- A. Al-Khawaja, J.G. Petersen, M. Damgaard, M.H. Jensen, S.B. Vogensen, M.E. Lie, B. Kragholm, H. Bräuner-Osborne, R.P. Clausen, B. Frølund, and P. Wellendorph Neurochem. Res. 39 2014 1988
- (2014) Neurochem. Res. , vol.39 , pp. 1988
- Al-Khawaja, A.¹ Petersen, J.G.² Damgaard, M.³ Jensen, M.H.⁴ Vogensen, S.B.⁵ Lie, M.E.⁶ Kragholm, B.⁷ Bräuner-Osborne, H.⁸ Clausen, R.P.⁹ Frølund, B.¹⁰ Wellendorph, P.¹¹

32
- 0036077331
- H.S. White, A. Sarup, T. Bolvig, A.S. Kristensen, G. Petersen, N. Nelson, D.S. Pickering, O.M. Larsson, B. Frolund, P. Krogsgaard-Larsen, and A. Schousboe J. Pharmacol. Exp. Ther. 302 2002 636
- (2002) J. Pharmacol. Exp. Ther. , vol.302 , pp. 636
- White, H.S.¹ Sarup, A.² Bolvig, T.³ Kristensen, A.S.⁴ Petersen, G.⁵ Nelson, N.⁶ Pickering, D.S.⁷ Larsson, O.M.⁸ Frolund, B.⁹ Krogsgaard-Larsen, P.¹⁰ Schousboe, A.¹¹

33
- 0019781092
- O.M. Larsson, P. Thorbek, P. Krogsgaard-Larsen, and A. Schousboe J. Neurochem. 37 1981 1509
- (1981) J. Neurochem. , vol.37 , pp. 1509
- Larsson, O.M.¹ Thorbek, P.² Krogsgaard-Larsen, P.³ Schousboe, A.⁴

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.