Target validation using chemical probes

Nature Chemical Biology

Volumn 9, Issue 4, 2013, Pages 195-199

  Bunnage, Mark E ^a   Chekler, Eugene L Piatnitski ^a   Jones, Lyn H ^a  

^a PFIZER INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

APOLIPOPROTEIN A1; BENZODIAZEPINE;

ANALYTIC METHOD; BIOASSAY; CELL MEMBRANE PERMEABILITY; CHEMICAL PROBE; CHROMATIN; CYTOLOGY; DOSE RESPONSE; DRUG EFFICACY; DRUG RESEARCH; ENANTIOMER; GENE EXPRESSION; INTRACELLULAR SPACE; LIPOPHILICITY; MOLECULAR MECHANICS; MOLECULAR PROBE; NOTE; PHENOTYPE; PHYSICAL CHEMISTRY; PRIORITY JOURNAL; PROTEIN EXPRESSION; PROTEOMICS; STRUCTURE ACTIVITY RELATION;

BIOMARKERS, PHARMACOLOGICAL; CELL MEMBRANE PERMEABILITY; DRUG DISCOVERY; DRUG EVALUATION, PRECLINICAL; HUMANS; MOLECULAR PROBES; MOLECULAR TARGETED THERAPY; STRUCTURE-ACTIVITY RELATIONSHIP; VALIDATION STUDIES AS TOPIC;

EID: 84875476426     PISSN: 15524450     EISSN: 15524469     Source Type: Journal    
DOI: 10.1038/nchembio.1197     Document Type: Note

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