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MedChemComm

Volumn 6, Issue 7, 2015, Pages 1267-1271

Fragment growing exploiting dynamic combinatorial chemistry of inhibitors of the aspartic protease endothiapepsin

(3) Mondal, Milon a Groothuis, Daphne E a Hirsch, Anna K H a

a UNIVERSITY OF GRONINGEN (Netherlands)

Author keywords

[No Author keywords available]

Indexed keywords

ACYLHYDRAZONE DERIVATIVE; ASPARTIC PROTEINASE INHIBITOR; ENDOTHIAPEPSIN; HYDRAZONE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; COMBINATORIAL CHEMISTRY; DRUG DESIGN; DRUG SYNTHESIS; DRUG TARGETING; ENZYME ACTIVITY; ENZYME INHIBITION; ENZYME STRUCTURE; FLUORESCENCE ANALYSIS; FRAGMENT BASED DRUG DESIGN; HYDROGEN BOND; PRIORITY JOURNAL; PROCESS OPTIMIZATION;

EID: 84936870389 PISSN: 20402503 EISSN: 20402511 Source Type: Journal
DOI: 10.1039/c5md00157a Document Type: Article

Times cited : (17)

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