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Bioorganic and Medicinal Chemistry Letters

Volumn 25, Issue 16, 2015, Pages 3213-3216

Synthesis and biological evaluation of novel m-carborane-containing estrogen receptor partial agonists as SERM candidates

(4) Ohta, Kiminori a Ogawa, Takumi a Kaise, Asako a Endo, Yasuyuki a

a TOHOKU PHARMACEUTICAL UNIVERSITY (Japan)

Author keywords

Carborane; Estrogen receptor; Partial agonist; SERM

Indexed keywords

CARBORANE DERIVATIVE; ESTRADIOL; ESTROGEN RECEPTOR ALPHA; HORMONE RECEPTOR AFFECTING AGENT; METHYL GROUP; N,N DIMETHYLAMINOETHYLOXY; SELECTIVE ESTROGEN RECEPTOR MODULATOR; UNCLASSIFIED DRUG; BORON DERIVATIVE; RECOMBINANT PROTEIN;

ARTICLE; BINDING AFFINITY; BIOLOGICAL ACTIVITY; CELL PROLIFERATION; COMPETITIVE BINDING ASSAY; DRUG POTENCY; DRUG SYNTHESIS; HUMAN; HUMAN CELL; MCF 7 CELL LINE; RECEPTOR BINDING; ANTAGONISTS AND INHIBITORS; CHEMICAL STRUCTURE; CONFORMATION; DRUG DESIGN; DRUG EFFECTS; METABOLISM; STRUCTURE ACTIVITY RELATION; SYNTHESIS;

BORON COMPOUNDS; CELL PROLIFERATION; DRUG DESIGN; ESTROGEN RECEPTOR ALPHA; HUMANS; MCF-7 CELLS; MODELS, MOLECULAR; MOLECULAR CONFORMATION; RECOMBINANT PROTEINS; SELECTIVE ESTROGEN RECEPTOR MODULATORS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84934807680 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2015.05.083 Document Type: Article

Times cited : (13)

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