SCOPUS 정보 검색 플랫폼

Volumn 21, Issue 18, 2015, Pages 6921-6929

Synthesis and biological evaluation of RGD peptidomimetic-paclitaxel conjugates bearing lysosomally cleavable linkers

(14) Dal Corso, Alberto a Caruso, Michele b Belvisi, Laura a Arosio, Daniela c Piarulli, Umberto d Albanese, Clara b Gasparri, Fabio b Marsiglio, Aurelio b Sola, Francesco b Troiani, Sonia b Valsasina, Barbara b Pignataro, Luca a Donati, Daniele b Gennari, Cesare a

a UNIVERSITY OF MILAN (Italy)

b NERVIANO MEDICAL SCIENCES (Italy)

c CNR Consiglio Nazionale delle Ricerche (Italy)

d UNIVERSITY OF INSUBRIA (Italy)

Author keywords

antitumor agents; drug delivery; integrins; peptidomimetics; prodrugs

Indexed keywords

ANTIGENS; CELL CULTURE; COMPUTATIONAL ELECTROMAGNETICS; DRUG DELIVERY; PEPTIDES;

ACUTE LYMPHOBLASTIC LEUKEMIA; ANTI-PROLIFERATIVE ACTIVITIES; ANTI-TUMOR AGENTS; BIOLOGICAL EVALUATION; INTEGRINS; NANOMOLAR CONCENTRATION; PEPTIDOMIMETICS; PRODRUGS;

SYNTHESIS (CHEMICAL);

ANTINEOPLASTIC AGENT; ARGINYL-GLYCYL-ASPARTIC ACID; CYCLOPEPTIDE; LIGAND; OLIGOPEPTIDE; PACLITAXEL; PEPTIDOMIMETIC AGENT; PHARMACOLOGY; PIPERAZINEDIONE; VITRONECTIN RECEPTOR;

ANALOGS AND DERIVATIVES; BINDING COMPETITION; CELL PROLIFERATION; CELL SURVIVAL; CHEMICAL STRUCTURE; CHEMISTRY; DRUG EFFECTS; DRUG RELEASE; DRUG STABILITY; HUMAN; LYSOSOME; METABOLISM; SYNTHESIS; TUMOR CELL LINE;

ANALOGS AND DERIVATIVES; ANTINEOPLASTIC AGENTS; BINDING, COMPETITIVE; CELL LINE, TUMOR; CELL PROLIFERATION; CELL SURVIVAL; CHEMICAL SYNTHESIS; CHEMISTRY; DIKETOPIPERAZINES; DRUG EFFECTS; DRUG LIBERATION; DRUG STABILITY; HUMANS; INTEGRIN ALPHAVBETA3; LIGANDS; LYSOSOMES; METABOLISM; MOLECULAR STRUCTURE; OLIGOPEPTIDES; PACLITAXEL; PEPTIDES, CYCLIC; PEPTIDOMIMETICS; PHARMACOLOGY;

EID: 84927616502 PISSN: 09476539 EISSN: 15213765 Source Type: Journal
DOI: 10.1002/chem.201500158 Document Type: Article

Times cited : (52)

References (38)

1
- 84862698355
- T. Lammers, F. Kiessling, W. E. Hennink, G. Storm, J. Controlled Release 2012, 161, 175-187
- (2012) J. Controlled Release , vol.161 , pp. 175-187
- Lammers, T.¹ Kiessling, F.² Hennink, W.E.³ Storm, G.⁴

2
- 84999317594
- U. K. Marelli, F. Rechenmacher, T. R. Ali Sobahi, C. Mas-Moruno, H. Kessler, Front. Oncol. 2013, 3, 1-12.
- (2013) Front. Oncol. , vol.3 , pp. 1-12
- Marelli, U.K.¹ Rechenmacher, F.² Ali Sobahi, T.R.³ Mas-Moruno, C.⁴ Kessler, H.⁵

3
- 84898066972
- R. V. J. Chari, M. L. Miller, W. C. Widdison, Angew. Chem. Int. Ed. 2014, 53, 3796-3827
- (2014) Angew. Chem. Int. Ed. , vol.53 , pp. 3796-3827
- Chari, R.V.J.¹ Miller, M.L.² Widdison, W.C.³

4
- 84905368754
- Angew. Chem. 2014, 126, 3872-3904.
- (2014) Angew. Chem. , vol.126 , pp. 3872-3904

5
- 85050579641
- A. M. Thayer, C&EN 2014, 92/3, 13-21.
- (2014) C&EN , vol.923 , pp. 13-21
- Thayer, A.M.¹

6
- 84872866038
- N. Krall, J. Scheuermann, D. Neri, Angew. Chem. Int. Ed. 2013, 52, 1384-1402
- (2013) Angew. Chem. Int. Ed. , vol.52 , pp. 1384-1402
- Krall, N.¹ Scheuermann, J.² Neri, D.³

7
- 84874631707
- Angew. Chem. 2013, 125, 1424-1443.
- (2013) Angew. Chem. , vol.125 , pp. 1424-1443

8
- 84868563717
- F. Danhier, A. Le Breton, V. Préat, Mol. Pharm. 2012, 9, 2961-2973.
- (2012) Mol. Pharm. , vol.9 , pp. 2961-2973
- Danhier, F.¹ Le Breton, A.² Préat, V.³

9
- 0021271957
- M. D. Pierschbacher, E. Ruoslahti, Nature 1984, 309, 30-33.
- (1984) Nature , vol.309 , pp. 30-33
- Pierschbacher, M.D.¹ Ruoslahti, E.²

10
- 77950674729
- L. Auzzas, F. Zanardi, L. Battistini, P. Burreddu, P. Carta, G. Rassu, C. Curti, G. Casiraghi, Curr. Med. Chem. 2010, 17, 1255-1299.
- (2010) Curr. Med. Chem. , vol.17 , pp. 1255-1299
- Auzzas, L.¹ Zanardi, F.² Battistini, L.³ Burreddu, P.⁴ Carta, P.⁵ Rassu, G.⁶ Curti, C.⁷ Casiraghi, G.⁸

11
- 0037023363
- J. P. Xiong, T. Stehle, R. Zhang, A. Joachimiak, M. Frech, S. L. Goodman, M. A. Arnaout, Science 2002, 296, 151-155
- (2002) Science , vol.296 , pp. 151-155
- Xiong, J.P.¹ Stehle, T.² Zhang, R.³ Joachimiak, A.⁴ Frech, M.⁵ Goodman, S.L.⁶ Arnaout, M.A.⁷

12
- 0037131442
- K. E. Gottschalk, H. Kessler, Angew. Chem. Int. Ed. 2002, 41, 3767-3774
- (2002) Angew. Chem. Int. Ed. , vol.41 , pp. 3767-3774
- Gottschalk, K.E.¹ Kessler, H.²

13
- 0037556057
- Angew. Chem. 2002, 114, 3919-3927.
- (2002) Angew. Chem. , vol.114 , pp. 3919-3927

14
- 0032535999
- W. Arap, R. Pasqualini, E. Ruoslahti, Science 1998, 279, 377-380.
- (1998) Science , vol.279 , pp. 377-380
- Arap, W.¹ Pasqualini, R.² Ruoslahti, E.³

15
- 0036725452
- F. M. H. de Groot, H. J. Broxterman, H. P. H. M. Adams, A. van Vliet, G. I. Tesser, Y. W. Elderkamp, A. J. Schraa, R. J. Kok, G. Molema, H. M. Pinedo, H. W. Scheeren, Mol. Cancer Ther. 2002, 1, 901-911.
- (2002) Mol. Cancer Ther. , vol.1 , pp. 901-911
- De Groot, F.M.H.¹ Broxterman, H.J.² Adams, H.P.H.M.³ Van Vliet, A.⁴ Tesser, G.I.⁵ Elderkamp, Y.W.⁶ Schraa, A.J.⁷ Kok, R.J.⁸ Molema, G.⁹ Pinedo, H.M.¹⁰ Scheeren, H.W.¹¹

16
- 12344253955
- D. J. Burkhart, B. T. Kalet, M. P. Coleman, G. C. Post, T. H. Koch, Mol. Cancer Ther. 2004, 3, 1593-1604.
- (2004) Mol. Cancer Ther. , vol.3 , pp. 1593-1604
- Burkhart, D.J.¹ Kalet, B.T.² Coleman, M.P.³ Post, G.C.⁴ Koch, T.H.⁵

17
- 84902655584
- J. L. Crisp, E. N. Savariar, H. L. Glasgow, L. G. Ellies, M. A. Whitney, R. Y. Tsien, Mol. Cancer Ther. 2014, 13, 1514-1525.
- (2014) Mol. Cancer Ther. , vol.13 , pp. 1514-1525
- Crisp, J.L.¹ Savariar, E.N.² Glasgow, H.L.³ Ellies, L.G.⁴ Whitney, M.A.⁵ Tsien, R.Y.⁶

18
- 84864456950
- M. H. Lee, J. Y. Kim, J. H. Han, S. Bhuniya, J. L. Sessler, C. Kang, J. S. Kim, J. Am. Chem. Soc. 2012, 134, 12668-12674.
- (2012) J. Am. Chem. Soc. , vol.134 , pp. 12668-12674
- Lee, M.H.¹ Kim, J.Y.² Han, J.H.³ Bhuniya, S.⁴ Sessler, J.L.⁵ Kang, C.⁶ Kim, J.S.⁷

19
- 38949103712
- S. Mukhopadhyay, C. M. Barnés, A. Haskel, S. M. Short, K. R. Barnes, S. J. Lippard, Bioconjugate Chem. 2008, 19, 39-49.
- (2008) Bioconjugate Chem. , vol.19 , pp. 39-49
- Mukhopadhyay, S.¹ Barnés, C.M.² Haskel, A.³ Short, S.M.⁴ Barnes, K.R.⁵ Lippard, S.J.⁶

20
- 13944278751
- X. Chen, C. Plasencia, Y. Hou, N. Neamati, J. Med. Chem. 2005, 48, 1098-1106
- (2005) J. Med. Chem. , vol.48 , pp. 1098-1106
- Chen, X.¹ Plasencia, C.² Hou, Y.³ Neamati, N.⁴

21
- 48149102140
- Q. Cao, Z. B. Li, K. Chen, Z. Wu, L. He, N. Neamati, X. Chen, Eur. J. Nucl. Med. Mol. Imaging 2008, 35, 1489-1498
- (2008) Eur. J. Nucl. Med. Mol. Imaging , vol.35 , pp. 1489-1498
- Cao, Q.¹ Li, Z.B.² Chen, K.³ Wu, Z.⁴ He, L.⁵ Neamati, N.⁶ Chen, X.⁷

22
- 84865138567
- M. Pilkington-Miksa, D. Arosio, L. Battistini, L. Belvisi, M. De Matteo, F. Vasile, P. Burreddu, P. Carta, G. Rassu, P. Perego, N. Carenini, F. Zunino, M. De Cesare, V. Castiglioni, E. Scanziani, C. Scolastico, G. Casiraghi, F. Zanardi, L. Manzoni, Bioconjugate Chem. 2012, 23, 1610-1622.
- (2012) Bioconjugate Chem. , vol.23 , pp. 1610-1622
- Pilkington-Miksa, M.¹ Arosio, D.² Battistini, L.³ Belvisi, L.⁴ De Matteo, M.⁵ Vasile, F.⁶ Burreddu, P.⁷ Carta, P.⁸ Rassu, G.⁹ Perego, P.¹⁰ Carenini, N.¹¹ Zunino, F.¹² De Cesare, M.¹³ Castiglioni, V.¹⁴ Scanziani, E.¹⁵ Scolastico, C.¹⁶ Casiraghi, G.¹⁷ Zanardi, F.¹⁸ Manzoni, L.¹⁹

23
- 0032819838
- H. M. Ellerby, W. Arap, L. M. Ellerby, R. Kain, R. Andrusiak, G. Del Rio, S. Krajewsky, C. R. Lombardo, R. Rao, E. Ruoslahti, D. E. Bredesen, R. Pasqualini, Nat. Med. 1999, 5, 1032-1038.
- (1999) Nat. Med. , vol.5 , pp. 1032-1038
- Ellerby, H.M.¹ Arap, W.² Ellerby, L.M.³ Kain, R.⁴ Andrusiak, R.⁵ Del Rio, G.⁶ Krajewsky, S.⁷ Lombardo, C.R.⁸ Rao, R.⁹ Ruoslahti, E.¹⁰ Bredesen, D.E.¹¹ Pasqualini, R.¹²

24
- 84899090315
- M. Mingozzi, L. Manzoni, D. Arosio, A. Dal Corso, M. Manzotti, F. Innamorati, L. Pignataro, D. Lecis, D. Delia, P. Seneci, C. Gennari, Org. Biomol. Chem. 2014, 12, 3288-3302.
- (2014) Org. Biomol. Chem. , vol.12 , pp. 3288-3302
- Mingozzi, M.¹ Manzoni, L.² Arosio, D.³ Dal Corso, A.⁴ Manzotti, M.⁵ Innamorati, F.⁶ Pignataro, L.⁷ Lecis, D.⁸ Delia, D.⁹ Seneci, P.¹⁰ Gennari, C.¹¹

25
- 84860773239
- M. Marchini, M. Mingozzi, R. Colombo, I. Guzzetti, L. Belvisi, F. Vasile, D. Potenza, U. Piarulli, D. Arosio, C. Gennari, Chem. Eur. J. 2012, 18, 6195-6207.
- (2012) Chem. Eur. J. , vol.18 , pp. 6195-6207
- Marchini, M.¹ Mingozzi, M.² Colombo, R.³ Guzzetti, I.⁴ Belvisi, L.⁵ Vasile, F.⁶ Potenza, D.⁷ Piarulli, U.⁸ Arosio, D.⁹ Gennari, C.¹⁰

26
- 84870974922
- R. Colombo, M. Mingozzi, L. Belvisi, D. Arosio, U. Piarulli, N. Carenini, P. Perego, N. Zaffaroni, M. De Cesare, V. Castiglioni, E. Scanziani, C. Gennari, J. Med. Chem. 2012, 55, 10460-10474.
- (2012) J. Med. Chem. , vol.55 , pp. 10460-10474
- Colombo, R.¹ Mingozzi, M.² Belvisi, L.³ Arosio, D.⁴ Piarulli, U.⁵ Carenini, N.⁶ Perego, P.⁷ Zaffaroni, N.⁸ De Cesare, M.⁹ Castiglioni, V.¹⁰ Scanziani, E.¹¹ Gennari, C.¹²

27
- 33644827912
- K. Temming, R. M. Schiffelers, G. Molemad, R. J. Kok, Drug Resist. Updates 2005, 8, 381-402
- (2005) Drug Resist. Updates , vol.8 , pp. 381-402
- Temming, K.¹ Schiffelers, R.M.² Molemad, G.³ Kok, R.J.⁴

28
- 58949095768
- C. Ryppa, H. Mann-Steinberg, M. L. Biniossek, R. Satchi-Fainaro, F. Kratz, Int. J. Pharm. 2009, 368, 89-97.
- (2009) Int. J. Pharm. , vol.368 , pp. 89-97
- Ryppa, C.¹ Mann-Steinberg, H.² Biniossek, M.L.³ Satchi-Fainaro, R.⁴ Kratz, F.⁵

29
- 3042779899
- M. Dyba, N. I. Tarasova, C. J. Michejda, Curr. Pharm. Des. 2004, 10, 2311-2334.
- (2004) Curr. Pharm. Des. , vol.10 , pp. 2311-2334
- Dyba, M.¹ Tarasova, N.I.² Michejda, C.J.³

30
- 84864572139
- K. Y. Choi, M. Swierczewska, S. Lee, X. Chen, Theranostics 2012, 2, 156-178.
- (2012) Theranostics , vol.2 , pp. 156-178
- Choi, K.Y.¹ Swierczewska, M.² Lee, S.³ Chen, X.⁴

31
- 84875140978
- M. Nahrwold, C. Weiß, T. Bogner, F. Mertink, J. Conradi, B. Sammet, R. Palmisano, S. Royo Gracia, T. Preuße, N. Sewald, J. Med. Chem. 2013, 56, 1853-1864.
- (2013) J. Med. Chem. , vol.56 , pp. 1853-1864
- Nahrwold, M.¹ Weiß, C.² Bogner, T.³ Mertink, F.⁴ Conradi, J.⁵ Sammet, B.⁶ Palmisano, R.⁷ Royo Gracia, S.⁸ Preuße, T.⁹ Sewald, N.¹⁰

32
- 0035966194
- F. M. H. de Groot, W. J. Loos, R. Koekkoek, L. W. A. van Berkom, G. F. Busscher, A. E. Seelen, C. Albrecht, P. de Bruijn, H. W. Scheeren, J. Org. Chem. 2001, 66, 8815-8830.
- (2001) J. Org. Chem. , vol.66 , pp. 8815-8830
- De Groot, F.M.H.¹ Loos, W.J.² Koekkoek, R.³ Van Berkom, L.W.A.⁴ Busscher, G.F.⁵ Seelen, A.E.⁶ Albrecht, C.⁷ De Bruijn, P.⁸ Scheeren, H.W.⁹

33
- 84866334630
- K. Hochdörffer, K. Abu Ajaj, C. Schäfer-Obodozie, F. Kratz, J. Med. Chem. 2012, 55, 7502-7515.
- (2012) J. Med. Chem. , vol.55 , pp. 7502-7515
- Hochdörffer, K.¹ Abu Ajaj, K.² Schäfer-Obodozie, C.³ Kratz, F.⁴

34
- 84855427940
- Y. Liu, K. M. Bajjuri, C. Liu, S. C. Sinha, Mol. Pharm. 2012, 9, 168-175.
- (2012) Mol. Pharm. , vol.9 , pp. 168-175
- Liu, Y.¹ Bajjuri, K.M.² Liu, C.³ Sinha, S.C.⁴

35
- 72049083697
- A. Dal Pozzo, M.-H. Ni, E. Esposito, S. Dallavalle, L. Musso, A. Bargiotti, C. Pisano, L. Vesci, F. Bucci, M. Castorina, R. Foderà, G. Giannini, C. Aulicino, S. Penco, Bioorg. Med. Chem. 2010, 18, 64-72.
- (2010) Bioorg. Med. Chem. , vol.18 , pp. 64-72
- Dal Pozzo, A.¹ Ni, M.-H.² Esposito, E.³ Dallavalle, S.⁴ Musso, L.⁵ Bargiotti, A.⁶ Pisano, C.⁷ Vesci, L.⁸ Bucci, F.⁹ Castorina, M.¹⁰ Foderà, R.¹¹ Giannini, G.¹² Aulicino, C.¹³ Penco, S.¹⁴

36
- 84919921845
- 3- cells with the intrinsic selectivity factor of the free cationic, membrane-disrupting peptide KLA (S>1.5).
- (2014) J. Am. Chem. Soc. , vol.136 , pp. 17734-17737
- Ma, X.¹ Jia, J.² Cao, R.³ Wang, X.⁴ Fei, H.⁵

37
- 80052740269
- X. Wang, D. Ma, W. C. Olson, W. D. W. Heston, Mol. Cancer Ther. 2011, 10, 1728-1739.
- (2011) Mol. Cancer Ther. , vol.10 , pp. 1728-1739
- Wang, X.¹ Ma, D.² Olson, W.C.³ Heston, W.D.W.⁴

38
- 77950321217
- Y. Meyer, J. A. Richard, B. Delest, P. Noack, P. Y. Renard, A. Romieu, Org. Biomol. Chem. 2010, 8, 1777-1780.
- (2010) Org. Biomol. Chem. , vol.8 , pp. 1777-1780
- Meyer, Y.¹ Richard, J.A.² Delest, B.³ Noack, P.⁴ Renard, P.Y.⁵ Romieu, A.⁶

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.