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Organic and Biomolecular Chemistry

Volumn 13, Issue 14, 2015, Pages 4149-4154

Design, synthesis, and kinetic analysis of potent protein N-terminal methyltransferase 1 inhibitors

(4) Zhang, Gang a Richardson, Stacie Lynn a Mao, Yunfei a Huang, Rong a

a VIRGINIA COMMONWEALTH UNIVERSITY (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ALKYLATION; AMINO ACIDS; MASS SPECTROMETRY; PROTEINS; SUBSTRATES;

ANTI-CANCER THERAPEUTICS; BIOLOGICAL FUNCTIONS; COMPETITIVE INHIBITION; KINETIC ANALYSIS; METHYLTRANSFERASES; PEPTIDE SUBSTRATES; S ADENOSYL L METHIONINES; SELECTIVE INHIBITORS;

BIOSYNTHESIS;

ENZYME INHIBITOR; PROTEIN METHYLTRANSFERASE;

ANTAGONISTS AND INHIBITORS; CHEMICAL STRUCTURE; CHEMISTRY; DRUG DESIGN; KINETICS; PROTEIN CONFORMATION; SYNTHESIS;

DRUG DESIGN; ENZYME INHIBITORS; KINETICS; MODELS, MOLECULAR; PROTEIN CONFORMATION; PROTEIN METHYLTRANSFERASES;

EID: 84925739378 PISSN: 14770520 EISSN: None Source Type: Journal
DOI: 10.1039/c5ob00120j Document Type: Article

Times cited : (45)

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