SCOPUS 정보 검색 플랫폼

Bioorganic and Medicinal Chemistry Letters

Volumn 25, Issue 3, 2015, Pages 459-461

Hydroxamic acid based histone deacetylase inhibitors with confirmed activity against the malaria parasite

(3) Giannini, Giuseppe a Battistuzzi, Gianfranco a Vignola, Davide a

a Sigma Tau SpA (Italy)

Author keywords

Antimalarial activity; Antiprotozoan drug; HDAC inhibitors; Hydroxamic acid; Plasmodium falciparum

Indexed keywords

ANTIPROTOZOAL AGENT; BENZNIDAZOLE; CHLOROQUINE; HISTONE DEACETYLASE INHIBITOR; HYDROXAMIC ACID DERIVATIVE; MELARSOPROL; METRONIDAZOLE; MILTEFOSINE; PODOPHYLLOTOXIN; ST 7464 AA1; ST 7612 AA1; ST 8039 AA1; ST 8074 AA1; ST 8078 AA1; ST 8081 AA1; ST 8086 AA1; ST 8087 AA1; THIOL DERIVATIVE; UNCLASSIFIED DRUG; VORINOSTAT; ANTIMALARIAL AGENT; DIPEPTIDE; HISTONE DEACETYLASE; HYDROXAMIC ACID; ISOPROTEIN; ST8086AA1;

ANIMAL EXPERIMENT; ANIMAL MODEL; ANTIMALARIAL ACTIVITY; ARTICLE; DRUG CYTOTOXICITY; DRUG STRUCTURE; GIARDIA INTESTINALIS; IC50; IN VITRO STUDY; IN VIVO STUDY; LEISHMANIA DONOVANI; MALARIA; MALARIA FALCIPARUM; MOUSE; NONHUMAN; PLASMODIUM; PLASMODIUM FALCIPARUM; TRYPANOSOMA BRUCEI; TRYPANOSOMA CRUZI; TRYPANOSOMA RHODESIENSE; ANIMAL; ANTAGONISTS AND INHIBITORS; CHEMISTRY; DISEASE MODEL; DRUG EFFECTS; HUMAN; METABOLISM; PARASITE; TUMOR CELL LINE; VETERINARY;

EUKARYOTA; PLASMODIUM (APICOMPLEXA); PLASMODIUM FALCIPARUM; PROKARYOTA;

ANIMALS; ANTIMALARIALS; CELL LINE, TUMOR; DIPEPTIDES; DISEASE MODELS, ANIMAL; HISTONE DEACETYLASE INHIBITORS; HISTONE DEACETYLASES; HUMANS; HYDROXAMIC ACIDS; MALARIA; MICE; PARASITES; PLASMODIUM FALCIPARUM; PROTEIN ISOFORMS;

EID: 84920735768 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2014.12.051 Document Type: Article

Times cited : (37)

References (16)

1
- 84897973164
- K.T. Andrews, G. Fisher, and T.S. Skinner-Adams Int. J. Parasitol.: Drugs Drug Resist. 4 2014 95
- (2014) Int. J. Parasitol.: Drugs Drug Resist. , vol.4 , pp. 95
- Andrews, K.T.¹ Fisher, G.² Skinner-Adams, T.S.³

2
- 78149283647
- N.C. Wheatley, K.T. Andrews, T.L. Tran, A.J. Lucke, R.C. Reid, and D.P. Fairlie Bioorg. Med. Chem. Lett. 20 2010 7080
- (2010) Bioorg. Med. Chem. Lett. , vol.20 , pp. 7080
- Wheatley, N.C.¹ Andrews, K.T.² Tran, T.L.³ Lucke, A.J.⁴ Reid, R.C.⁵ Fairlie, D.P.⁶

3
- 84908676164
- Q. Sodji, V. Patil, S. Jain, J.R. Kornacki, M. Mrksich, B.L. Tekwani, and A.K. Oyelere Bioorg. Med. Chem. Lett. 24 2014 4826
- (2014) Bioorg. Med. Chem. Lett. , vol.24 , pp. 4826
- Sodji, Q.¹ Patil, V.² Jain, S.³ Kornacki, J.R.⁴ Mrksich, M.⁵ Tekwani, B.L.⁶ Oyelere, A.K.⁷

4
- 65449122745
- K.T. Andrews, T.N. Tran, N.C. Wheatley, and D.P. Fairlie Curr. Top. Med. Chem. 9 2009 292
- (2009) Curr. Top. Med. Chem. , vol.9 , pp. 292
- Andrews, K.T.¹ Tran, T.N.² Wheatley, N.C.³ Fairlie, D.P.⁴

5
- 84902147732
- F.K. Hansen, S.D. Sumanadasa, K. Stenzel, S. Duffy, S. Meister, L. Marek, R. Schmetter, K. Kuna, A. Hamacher, B. Mordmüller, M.U. Kassack, E.A. Winzeler, V.M. Avery, K.T. Andrews, and T. Kurz Eur. J. Med. Chem. 82 2014 204
- (2014) Eur. J. Med. Chem. , vol.82 , pp. 204
- Hansen, F.K.¹ Sumanadasa, S.D.² Stenzel, K.³ Duffy, S.⁴ Meister, S.⁵ Marek, L.⁶ Schmetter, R.⁷ Kuna, K.⁸ Hamacher, A.⁹ Mordmüller, B.¹⁰ Kassack, M.U.¹¹ Winzeler, E.A.¹² Avery, V.M.¹³ Andrews, K.T.¹⁴ Kurz, T.¹⁵

6
- 84864722456
- G. Giannini, W. Cabri, C. Fattorusso, and M. Rodriquez Future Med. Chem. - Targeted Oncol. 4 2012 1439
- (2012) Future Med. Chem. - Targeted Oncol. , vol.4 , pp. 1439
- Giannini, G.¹ Cabri, W.² Fattorusso, C.³ Rodriquez, M.⁴

7
- 84908388243
- G. Giannini, L. Vesci, G. Battistuzzi, D. Vignola, F.M. Milazzo, M.B. Guglielmi, M. Barbarino, M. Santaniello, N. Fantò, M. Mor, S. Rivara, D. Pala, M. Taddei, C. Pisano, and W. Cabri J. Med. Chem. 57 2014 8358
- (2014) J. Med. Chem. , vol.57 , pp. 8358
- Giannini, G.¹ Vesci, L.² Battistuzzi, G.³ Vignola, D.⁴ Milazzo, F.M.⁵ Guglielmi, M.B.⁶ Barbarino, M.⁷ Santaniello, M.⁸ Fantò, N.⁹ Mor, M.¹⁰ Rivara, S.¹¹ Pala, D.¹² Taddei, M.¹³ Pisano, C.¹⁴ Cabri, W.¹⁵

8
- 84920731361
- accepted for publication
- L. Vesci, E. Bernasconi, F. Milazzo, R. De Santis, E. Gaudio, I. Kwee, A. Rinaldi, S. Pace, V. Carollo, G. Giannini, and F. Bertoni Oncotarget J. 2015 accepted for publication
- (2015) Oncotarget J.
- Vesci, L.¹ Bernasconi, E.² Milazzo, F.³ De Santis, R.⁴ Gaudio, E.⁵ Kwee, I.⁶ Rinaldi, A.⁷ Pace, S.⁸ Carollo, V.⁹ Giannini, G.¹⁰ Bertoni, F.¹¹

9
- 84891496536
- M. Taddei, E. Cini, L. Giannotti, G. Giannini, G. Battistuzzi, D. Vignola, L. Vesci, and W. Cabri Bioorg. Med. Chem. Lett. 24 2014 61
- (2014) Bioorg. Med. Chem. Lett. , vol.24 , pp. 61
- Taddei, M.¹ Cini, E.² Giannotti, L.³ Giannini, G.⁴ Battistuzzi, G.⁵ Vignola, D.⁶ Vesci, L.⁷ Cabri, W.⁸

10
- 42049106596
- K.T. Andrews, T.N. Tran, A.J. Lucke, P. Kahnberg, G.T. Le, G.M. Boyle, D.L. Gardiner, T.S. Skinner-Adams, and D.P. Fairlie Antimicrob. Agents Chemother. 52 2008 1454
- (2008) Antimicrob. Agents Chemother. , vol.52 , pp. 1454
- Andrews, K.T.¹ Tran, T.N.² Lucke, A.J.³ Kahnberg, P.⁴ Le, G.T.⁵ Boyle, G.M.⁶ Gardiner, D.L.⁷ Skinner-Adams, T.S.⁸ Fairlie, D.P.⁹

11
- 84862571804
- S.D.M. Sumanadasa, C.D. Goodman, A.J. Lucke, T. Skinner-Adams, I. Sahama, A. Haque, T.A. Do, G.I. McFadden, D.P. Fairlie, and K.T. Andrews Antimicrob. Agents Chemother. 56 2012 3849
- (2012) Antimicrob. Agents Chemother. , vol.56 , pp. 3849
- Sumanadasa, S.D.M.¹ Goodman, C.D.² Lucke, A.J.³ Skinner-Adams, T.⁴ Sahama, I.⁵ Haque, A.⁶ Do, T.A.⁷ McFadden, G.I.⁸ Fairlie, D.P.⁹ Andrews, K.T.¹⁰

12
- 72049116798
- V. Patil, W. Guerrant, P.C. Chen, B. Gryder, D.B. Benicewicz, S.I. Khan, B.L. Tekwani, and A.K. Oyelere Bioorg. Med. Chem. 18 2010 415
- (2010) Bioorg. Med. Chem. , vol.18 , pp. 415
- Patil, V.¹ Guerrant, W.² Chen, P.C.³ Gryder, B.⁴ Benicewicz, D.B.⁵ Khan, S.I.⁶ Tekwani, B.L.⁷ Oyelere, A.K.⁸

13
- 84920731360
- J.M. Kelly, M.C. Taylor, D. Horn, E. Loza, I. Kalvinsh, and F. Björkling Bioorg. Med. Chem. Lett. 2012 1886 22
- (1886) Bioorg. Med. Chem. Lett. , vol.2012 , pp. 22
- Kelly, J.M.¹ Taylor, M.C.² Horn, D.³ Loza, E.⁴ Kalvinsh, I.⁵ Björkling, F.⁶

14
- 84920731359
- Preliminary Tests was performed by Marcel Kaiser - Swiss Tropical and Public Health Institute, Parasite Chemotherapy. Socinstrasse 57, CH-4002 Basel, Switzerland
- Preliminary Tests was performed by Marcel Kaiser - Swiss Tropical and Public Health Institute, Parasite Chemotherapy. Socinstrasse 57, CH-4002 Basel, Switzerland.

15
- 84920729076
- World Health Organization World Health Organization: Geneva, Switzerland
- World Health Organization. World Malaria Report; Fact Sheet No. 94; World Health Organization: Geneva, Switzerland, 2013.
- (2013) World Malaria Report; Fact Sheet No. 94

16
- 84920731358
- F. Oger, A. Lecorgne, E. Sala, V. Nardese, F. Demay, S. Chevance, D.C. Desravines, N. Aleksandrova, R. Le Guével, S. Lorenzi, A.R. Beccari, P. Barath, D.J. Hart, A. Bondon, D. Carettoni, G. Simonneaux, and G. Salbert J. Med. Chem. 2010 1937 53
- (1937) J. Med. Chem. , vol.2010 , pp. 53
- Oger, F.¹ Lecorgne, A.² Sala, E.³ Nardese, V.⁴ Demay, F.⁵ Chevance, S.⁶ Desravines, D.C.⁷ Aleksandrova, N.⁸ Le Guével, R.⁹ Lorenzi, S.¹⁰ Beccari, A.R.¹¹ Barath, P.¹² Hart, D.J.¹³ Bondon, A.¹⁴ Carettoni, D.¹⁵ Simonneaux, G.¹⁶ Salbert, G.¹⁷

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.