3D printing of modified-release aminosalicylate (4-ASA and 5-ASA) tablets

European Journal of Pharmaceutics and Biopharmaceutics

Volumn 89, Issue , 2015, Pages 157-162

  Goyanes, Alvaro ^a   Buanz, Asma B M ^a   Hatton, Grace B ^a   Gaisford, Simon ^a,b   Basit, Abdul W ^a,b  

^a UNIVERSITY OF LONDON   (United Kingdom)

^b FABRX LTD   (United Kingdom)

Author keywords

3D printing; Aminosalicylates; Bicarbonate buffer; Colonic drug delivery; Controlled release; Fused deposition modeling; Mesalamine; Personalized dosing; Printing medicines

Indexed keywords

AMINOSALICYLIC ACID; MESALAZINE; POLYVINYL ALCOHOL; SOLUTION AND SOLUBILITY; TABLET;

ARTICLE; COMPUTER PROGRAM; DIFFERENTIAL SCANNING CALORIMETRY; DRUG DEGRADATION; DRUG RELEASE; DRUG SOLUBILITY; DRUG SOLUTION; HUMAN; INTESTINE FLUID; MELTING POINT; TABLET; TABLET HARDNESS; TABLET SURFACE; TABLET THICKNESS; THERMAL ANALYSIS; THERMOGRAVIMETRY; THERMOSTABILITY; THREE DIMENSIONAL PRINTING; CHEMISTRY; HEAT; MEDICINAL CHEMISTRY; PHARMACEUTICS; PROCEDURES; SOLUTION AND SOLUBILITY;

AMINOSALICYLIC ACID; CALORIMETRY, DIFFERENTIAL SCANNING; CHEMISTRY, PHARMACEUTICAL; HOT TEMPERATURE; MESALAMINE; PHARMACEUTICAL SOLUTIONS; POLYVINYL ALCOHOL; PRINTING, THREE-DIMENSIONAL; TABLETS; TECHNOLOGY, PHARMACEUTICAL;

EID: 84920472123     PISSN: 09396411     EISSN: 18733441     Source Type: Journal    
DOI: 10.1016/j.ejpb.2014.12.003     Document Type: Article

References (27)

1. D.G. Yu, L.M. Zhu, C.J. Branford-White, and X.L. Yang Three-dimensional printing in pharmaceutics: promises and problems J. Pharm. Sci. 97 2008 3666 3690
2. L.-N. Wang Printing medicines: a new era of dispensing and drug formulation? Pharm. J. 291 2013 25 26
3. S.E. Moulton, and G.G. Wallace 3-Dimensional (3D) fabricated polymer based drug delivery systems J. Control. Release 194 2014 27 34
4. M. Alomari, F.H. Mohamed, A.W. Basit, and S. Gaisford Personalised dosing: printing a dose of one's own medicine Int. J. Pharm. 2014 10.1016/j.ijpharm.2014.12.006
5. N. Scoutaris, A.L. Hook, P.R. Gellert, C.J. Roberts, M.R. Alexander, and D.J. Scurr ToF-SIMS analysis of chemical heterogenities in inkjet micro-array printed drug/polymer formulations J. Mater. Sci. Mater. Med. 23 2012 385 391
6. A.B. Buanz, M.H. Saunders, A.W. Basit, and S. Gaisford Preparation of personalized-dose salbutamol sulphate oral films with thermal ink-jet printing Pharm. Res. 28 2011 2386 2392
7. G. Sharma, W. Mueannoom, A.B. Buanz, K.M. Taylor, and S. Gaisford In vitro characterisation of terbutaline sulphate particles prepared by thermal ink-jet spray freeze drying Int. J. Pharm. 447 2013 165 170
8. W. Mueannoom, A. Srisongphan, K.M. Taylor, S. Hauschild, and S. Gaisford Thermal ink-jet spray freeze-drying for preparation of excipient-free salbutamol sulphate for inhalation Eur. J. Pharm. Biopharm. 80 2012 149 155
9. C.C. Wang, M.R. Tejwani Motwani, W.J. Roach, J.L. Kay, J. Yoo, H.L. Surprenant, D.C. Monkhouse, and T.J. Pryor Development of near zero-order release dosage forms using three-dimensional printing (3-DP) technology Drug Dev. Ind. Pharm. 32 2006 367 376
10. W. Huang, Q. Zheng, W. Sun, H. Xu, and X. Yang Levofloxacin implants with predefined microstructure fabricated by three-dimensional printing technique Int. J. Pharm. 339 2007 33 38
11. U. Gbureck, E. Vorndran, F.A. Muller, and J.E. Barralet Low temperature direct 3D printed bioceramics and biocomposites as drug release matrices J. Control. Release 122 2007 173 180
12. W.E. Katstra, R.D. Palazzolo, C.W. Rowe, B. Giritlioglu, P. Teung, and M.J. Cima Oral dosage forms fabricated by three dimensional printing J. Control. Release 66 2000 1 9
13. C.W. Rowe, W.E. Katstra, R.D. Palazzolo, B. Giritlioglu, P. Teung, and M.J. Cima Multimechanism oral dosage forms fabricated by three dimensional printing J. Control. Release 66 2000 11 17
14. D.G. Yu, X.L. Yang, W.D. Huang, J. Liu, Y.G. Wang, and H. Xu Tablets with material gradients fabricated by three-dimensional printing J. Pharm. Sci. 96 2007 2446 2456
15. S.A. Khaled, J.C. Burley, M.R. Alexander, and C.J. Roberts Desktop 3D printing of controlled release pharmaceutical bilayer tablets Int. J. Pharm. 461 2014 105 111
16. D.G. Yu, C. Branford-White, Y.C. Yang, L.M. Zhu, E.W. Welbeck, and X.L. Yang A novel fast disintegrating tablet fabricated by three-dimensional printing Drug Dev. Ind. Pharm. 35 2009 1530 1536
17. D.G. Yu, X.X. Shen, C. Branford-White, L.M. Zhu, K. White, and X.L. Yang Novel oral fast-disintegrating drug delivery devices with predefined inner structure fabricated by three-dimensional printing J. Pharm. Pharmacol. 61 2009 323 329
18. A. Goyanes, A.B. Buanz, A.W. Basit, and S. Gaisford Fused-filament 3D printing (3DP) for fabrication of tablets Int. J. Pharm. 476 2014 88 92
19. E.L. McConnell, F. Liu, and A.W. Basit Colonic treatments and targets: issues and opportunities J. Drug Target. 17 2009 335 363
20. C. Tuleu, A.W. Basit, W.A. Waddington, P.J. Ell, and J.M. Newton Colonic delivery of 4-aminosalicylic acid using amylose-ethylcellulose-coated hydroxypropylmethylcellulose capsules Aliment. Pharmacol. Ther. 16 2002 1771 1779
21. DrugBank. < http://www.drugbank.ca/drugs/DB00244 > (last accessed 08.14).
22. S.H. Yalkowsky, and Y. He Handbook of Aqueous Solubility Data 2003 CRC Press Boca Raton
23. H.A. Merchant, J. Frost, A.W. Basit, Apparatus and Method for Testing Medicaments, PCT/GB2013/051145, 2012.
24. H.A. Merchant, A. Goyanes, N. Parashar, and A.W. Basit Predicting the gastrointestinal behaviour of modified-release products: utility of a novel dynamic dissolution test apparatus involving the use of bicarbonate buffers Int. J. Pharm. 475 2014 585 591
25. F. Liu, H.A. Merchant, R.P. Kulkarni, M. Alkademi, and A.W. Basit Evolution of a physiological pH 6.8 bicarbonate buffer system: application to the dissolution testing of enteric coated products Eur. J. Pharm. Biopharm. 78 2011 151 157
26. H.M. Fadda, H.A. Merchant, B.T. Arafat, and A.W. Basit Physiological bicarbonate buffers: stabilisation and use as dissolution media for modified release systems Int. J. Pharm. 382 2009 56 60
27. S. Gupta, T.J. Webster, and A. Sinha Evolution of PVA gels prepared without crosslinking agents as a cell adhesive surface J. Mater. Sci. Mater. Med. 22 2011 1763 1772