메뉴 건너뛰기




Volumn 29, Issue 1, 2015, Pages 113-123

Suitability of skin integrity tests for dermal absorption studies in vitro

Author keywords

Dermal absorption; Integrity tests; Internal reference standard; Skin barrier function; TEER; TEWL

Indexed keywords

ALCOHOL; CAFFEINE; MANNITOL; METHYLENE BLUE; TESTOSTERONE; TRITIUM; WATER;

EID: 84908374204     PISSN: 08872333     EISSN: 18793177     Source Type: Journal    
DOI: 10.1016/j.tiv.2014.09.007     Document Type: Article
Times cited : (94)

References (44)
  • 2
    • 33746256892 scopus 로고    scopus 로고
    • A liquid chromatography-fluorimetric method for the in vitro estimation of the skin penetration of disodium phenyldibenzimidazole tetrasulfonate from sunscreen formulations through human skin
    • Balaguer A., Salvador A., Chisvert A., Melia M., Herraez M., Diez O. A liquid chromatography-fluorimetric method for the in vitro estimation of the skin penetration of disodium phenyldibenzimidazole tetrasulfonate from sunscreen formulations through human skin. Anal. Bioanal. Chem. 2006, 385:1225-1232.
    • (2006) Anal. Bioanal. Chem. , vol.385 , pp. 1225-1232
    • Balaguer, A.1    Salvador, A.2    Chisvert, A.3    Melia, M.4    Herraez, M.5    Diez, O.6
  • 3
    • 0000969569 scopus 로고
    • Penetration enhancers - mode of action in humans
    • In: Shroot, B., Schäfer, H. (Eds.)
    • Barry, B.W., 1987. Penetration enhancers - mode of action in humans. In: Shroot, B., Schäfer, H. (Eds.), Skin Pharmacokinetics, pp. 121-137.
    • (1987) Skin Pharmacokinetics , pp. 121-137
    • Barry, B.W.1
  • 4
    • 0011519983 scopus 로고
    • Validation of the integrity of epidermal membranes during assessment of percutaneous penetration
    • Brain, K.R., James, V.J., Walters, K.A., 1995. Validation of the integrity of epidermal membranes during assessment of percutaneous penetration. Predict. Percut. Penet.
    • (1995) Predict. Percut. Penet
    • Brain, K.R.1    James, V.J.2    Walters, K.A.3
  • 5
    • 84908363500 scopus 로고    scopus 로고
    • British Crop Production Council, Hampshire, UK
    • Britisch Crop Protection Council, 2011. The e-pesticide manual V5.2. British Crop Production Council, Hampshire, UK.
    • (2011) The e-pesticide manual V5.2
  • 6
    • 0022976340 scopus 로고
    • Methods for in vitro percutaneous-absorption studies. 7. Use of excised human-skin
    • Bronaugh R.L., Stewart R.F., Simon M. Methods for in vitro percutaneous-absorption studies. 7. Use of excised human-skin. J. Pharm. Sci. 1986, 75:1094-1097.
    • (1986) J. Pharm. Sci. , vol.75 , pp. 1094-1097
    • Bronaugh, R.L.1    Stewart, R.F.2    Simon, M.3
  • 7
    • 24644475769 scopus 로고    scopus 로고
    • Effects of single and repeated exposure to biocidal active substances on the barrier function of the skin in vitro
    • Buist H.E., van de Sandt J.J.M., van Burgsteden J.A., de Heer C. Effects of single and repeated exposure to biocidal active substances on the barrier function of the skin in vitro. Regul. Toxicol. Pharmacol. 2005, 43:76-84.
    • (2005) Regul. Toxicol. Pharmacol. , vol.43 , pp. 76-84
    • Buist, H.E.1    van de Sandt, J.J.M.2    van Burgsteden, J.A.3    de Heer, C.4
  • 9
    • 1642378629 scopus 로고    scopus 로고
    • Multi-species assessment of electrical resistance as a skin integrity marker for in vitro percutaneous absorption studies
    • Davies D.J., Ward R.J., Heylings J.R. Multi-species assessment of electrical resistance as a skin integrity marker for in vitro percutaneous absorption studies. Toxicol. In Vitro 2004, 18:351-358.
    • (2004) Toxicol. In Vitro , vol.18 , pp. 351-358
    • Davies, D.J.1    Ward, R.J.2    Heylings, J.R.3
  • 11
    • 0022645793 scopus 로고
    • A method of predicting percutaneous-absorption rates from vehicle to vehicle - an experimental assessment
    • Dugard P.H., Scott R.C. A method of predicting percutaneous-absorption rates from vehicle to vehicle - an experimental assessment. Int. J. Pharm. 1986, 28:219-227.
    • (1986) Int. J. Pharm. , vol.28 , pp. 219-227
    • Dugard, P.H.1    Scott, R.C.2
  • 12
    • 84908500656 scopus 로고    scopus 로고
    • Guidance on Dermal Absorption
    • EFSA Panel on Plant Protection Products and their Residues, 2012. Guidance on Dermal Absorption. EFSA J., 10.
    • (2012) EFSA J. , pp. 10
  • 13
    • 73549090800 scopus 로고    scopus 로고
    • Correlation of transepidermal water loss with skin barrier properties in vitro: comparison of three evaporimeters
    • Elkeeb R., Hui X.Y., Chan H.D., Tian L.L., Maibach H.I. Correlation of transepidermal water loss with skin barrier properties in vitro: comparison of three evaporimeters. Skin Res. Technol. 2010, 16:9-15.
    • (2010) Skin Res. Technol. , vol.16 , pp. 9-15
    • Elkeeb, R.1    Hui, X.Y.2    Chan, H.D.3    Tian, L.L.4    Maibach, H.I.5
  • 14
    • 0036889871 scopus 로고    scopus 로고
    • Rapid integrity assessment of rat and human epidermal membranes for in vitro dermal regulatory testing: correlation of electrical resistance with tritiated water permeability
    • Fasano W.J., Manning L.A., Green J.W. Rapid integrity assessment of rat and human epidermal membranes for in vitro dermal regulatory testing: correlation of electrical resistance with tritiated water permeability. Toxicol. In Vitro 2002, 16:731-740.
    • (2002) Toxicol. In Vitro , vol.16 , pp. 731-740
    • Fasano, W.J.1    Manning, L.A.2    Green, J.W.3
  • 15
    • 0016053262 scopus 로고
    • Mass-transport phenomena and models - theoretical concepts
    • Flynn G.L., Yalkowsk S.H., Roseman T.J. Mass-transport phenomena and models - theoretical concepts. J. Pharm. Sci. 1974, 63:479-510.
    • (1974) J. Pharm. Sci. , vol.63 , pp. 479-510
    • Flynn, G.L.1    Yalkowsk, S.H.2    Roseman, T.J.3
  • 17
    • 61349127266 scopus 로고    scopus 로고
    • Closed-chamber transepidermal water loss measurement: microclimate, calibration and performance
    • Imhof R., De Jesus M., Xiao P., Ciortea L.I., Berg E. Closed-chamber transepidermal water loss measurement: microclimate, calibration and performance. Int. J. Cosmetic Sci. 2009, 31:97-118.
    • (2009) Int. J. Cosmetic Sci. , vol.31 , pp. 97-118
    • Imhof, R.1    De Jesus, M.2    Xiao, P.3    Ciortea, L.I.4    Berg, E.5
  • 20
    • 0030748491 scopus 로고    scopus 로고
    • Electrical resistance and tritiated water permeability as indicators of barrier integrity of in vitro human skin
    • Lawrence J.N. Electrical resistance and tritiated water permeability as indicators of barrier integrity of in vitro human skin. Toxicol. In Vitro 1997, 11:241-249.
    • (1997) Toxicol. In Vitro , vol.11 , pp. 241-249
    • Lawrence, J.N.1
  • 21
    • 8644243613 scopus 로고
    • Partition coefficients and their uses
    • Leo A., Hansch C., Elkins D. Partition coefficients and their uses. Chem. Rev. 1971, 71. 525+.
    • (1971) Chem. Rev. , vol.71 , pp. 525+
    • Leo, A.1    Hansch, C.2    Elkins, D.3
  • 22
    • 14844331069 scopus 로고    scopus 로고
    • The correlation between transepidermal water loss and percutaneous absorption: an overview
    • Levin J., Maibach H. The correlation between transepidermal water loss and percutaneous absorption: an overview. J. Control. Rel. 2005, 103:291-299.
    • (2005) J. Control. Rel. , vol.103 , pp. 291-299
    • Levin, J.1    Maibach, H.2
  • 24
    • 41949140167 scopus 로고    scopus 로고
    • Inter- and intra-individual variability in human skin barrier function: a large scale retrospective study
    • Meidan V.M., Roper C.S. Inter- and intra-individual variability in human skin barrier function: a large scale retrospective study. Toxicol. In Vitro 2008, 22:1062-1069.
    • (2008) Toxicol. In Vitro , vol.22 , pp. 1062-1069
    • Meidan, V.M.1    Roper, C.S.2
  • 25
    • 84908363497 scopus 로고    scopus 로고
    • Merck, Safety Data Sheet Caffeine
    • Merck, 2006. Safety Data Sheet Caffeine.
    • (2006)
  • 26
    • 33645890848 scopus 로고    scopus 로고
    • TEWL measurements as a routine method for evaluating the integrity of epidermis sheets in static Franz type diffusion cells in vitro. Limitations shown by transport data testing
    • Netzlaff F., Kostka K.H., Lehr C.M., Schäfer U.F. TEWL measurements as a routine method for evaluating the integrity of epidermis sheets in static Franz type diffusion cells in vitro. Limitations shown by transport data testing. Eur. J. Pharm. Biopharm. 2006, 63:44-50.
    • (2006) Eur. J. Pharm. Biopharm. , vol.63 , pp. 44-50
    • Netzlaff, F.1    Kostka, K.H.2    Lehr, C.M.3    Schäfer, U.F.4
  • 27
    • 13244297586 scopus 로고    scopus 로고
    • Guidance document for the conduct of skin absorption studies - OECD Series in Testing and assessment - Number 28.
    • Organisation for Economic Co-operation and Development
    • OECD, 2004a. Guidance document for the conduct of skin absorption studies - OECD Series in Testing and assessment - Number 28. Organisation for Economic Co-operation and Development.
    • (2004)
  • 28
    • 25644432500 scopus 로고    scopus 로고
    • OECD Guideline for the testing of chemicals. Skin absorption: in vitro method 428
    • Organisation for Economic Co-operation and Development
    • OECD, 2004b. OECD Guideline for the testing of chemicals. Skin absorption: in vitro method 428. Organisation for Economic Co-operation and Development.
    • (2004)
  • 30
    • 0029027865 scopus 로고
    • The effect of temperature upon the permeation of polar and ionic solutes through human epidermal membrane
    • Peck K.D., Ghanem A.H., Higuchi W.I. The effect of temperature upon the permeation of polar and ionic solutes through human epidermal membrane. J. Pharm. Sci. 1995, 84:975-982.
    • (1995) J. Pharm. Sci. , vol.84 , pp. 975-982
    • Peck, K.D.1    Ghanem, A.H.2    Higuchi, W.I.3
  • 32
    • 84908376669 scopus 로고    scopus 로고
    • Absorption
    • Wiley-Blackwell, J.E. Riviere (Ed.)
    • Riviere J.E. Absorption. Comparative Pharmacokinetics 2011, 39-71. Wiley-Blackwell. J.E. Riviere (Ed.).
    • (2011) Comparative Pharmacokinetics , pp. 39-71
    • Riviere, J.E.1
  • 34
    • 34347368059 scopus 로고
    • Invivo relationship between trans-epidermal water-loss and percutaneous-absorption in man
    • Rougier A., Lotte C., Maibach H.I. Invivo relationship between trans-epidermal water-loss and percutaneous-absorption in man. Clin. Res. 1988, 36:A690.
    • (1988) Clin. Res. , vol.36 , pp. A690
    • Rougier, A.1    Lotte, C.2    Maibach, H.I.3
  • 35
    • 0003921350 scopus 로고    scopus 로고
    • Factors effecting percutaneous absorption
    • In: Schäfer, H., Redelmeier, T.E., Skin Barrier
    • Schäfer, H., Redelmeier, T.E., 1996a. Factors effecting percutaneous absorption. In: Schäfer, H., Redelmeier, T.E., Skin Barrier, Principles of Percutaneous Absorption, 153-212.
    • (1996) Principles of Percutaneous Absorption , pp. 153-212
    • Schäfer, H.1    Redelmeier, T.E.2
  • 36
    • 0000152584 scopus 로고    scopus 로고
    • Prediction and Measurement of Percutaneous Absorption
    • Schäfer, H., Redelmeier, T.E., Skin Barrier
    • Schäfer, H., Redelmeier, T.E., 1996b Prediction and Measurement of Percutaneous Absorption. In: Schäfer, H., Redelmeier, T.E., Skin Barrier, Principles of Percutaneous Absorption, 118-152.
    • (1996) Principles of Percutaneous Absorption , pp. 118-152
    • Schäfer, H.1    Redelmeier, T.E.2
  • 39
    • 57349107203 scopus 로고    scopus 로고
    • Alteration of skin hydration and its barrier function by vehicle and permeation enhancers: a study using TGA, FTIR, TEWL and drug permeation as markers
    • Shah D.K., Khandavilli S., Panchagnula R. Alteration of skin hydration and its barrier function by vehicle and permeation enhancers: a study using TGA, FTIR, TEWL and drug permeation as markers. Meth. Find. Exp. Clin. Pharmacol. 2008, 30:499-512.
    • (2008) Meth. Find. Exp. Clin. Pharmacol. , vol.30 , pp. 499-512
    • Shah, D.K.1    Khandavilli, S.2    Panchagnula, R.3
  • 40
    • 84908363495 scopus 로고    scopus 로고
    • Sigma-Aldrich, Sicherheitsdatenblatt D-Mannitol.
    • Sigma-Aldrich, 2007. Sicherheitsdatenblatt D-Mannitol.
    • (2007)
  • 41
    • 0021365145 scopus 로고
    • Variations in permeability of human-skin within and between specimens
    • Southwell D., Barry B.W., Woodford R. Variations in permeability of human-skin within and between specimens. Int. J. Pharm. 1984, 18:299-309.
    • (1984) Int. J. Pharm. , vol.18 , pp. 299-309
    • Southwell, D.1    Barry, B.W.2    Woodford, R.3
  • 44
    • 0020599769 scopus 로고
    • Solubility and partitioning. 6. Octanol solubility and octanol-water partition-coefficients
    • Yalkowsky S.H., Valvani S.C., Roseman T.J. Solubility and partitioning. 6. Octanol solubility and octanol-water partition-coefficients. J. Pharm. Sci. 1983, 72:866-870.
    • (1983) J. Pharm. Sci. , vol.72 , pp. 866-870
    • Yalkowsky, S.H.1    Valvani, S.C.2    Roseman, T.J.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.