Rational design, synthesis and anti-proliferative evaluation of novel benzosuberone tethered with hydrazide-hydrazones

Bioorganic and Medicinal Chemistry Letters

Volumn 24, Issue 21, 2014, Pages 5041-5044

  Yadagiri, Bandi ^a   Holagunda, Uma Devi ^a   Bantu, Rajashaker ^a   Nagarapu, Lingaiah ^a   Guguloth, Vijayacharan ^a   Polepally, Sowjanya ^a   Jain, Nishanth ^a  

^a INDIAN INSTITUTE OF CHEMICAL TECHNOLOGY   (India)

Author keywords

Anti proliferative; Benzosuberone; Cell lines; Hydrazide hydrazones

Indexed keywords

ALDEHYDE; ANTINEOPLASTIC AGENT; BENZOSUBERONE; FUNCTIONAL GROUP; GROWTH INHIBITOR; HYDRAZIDE DERIVATIVE; HYDRAZONE DERIVATIVE; UNCLASSIFIED DRUG; COUMARIN DERIVATIVE; HYDRAZINE; HYDRAZINE DERIVATIVE;

ANTIPROLIFERATIVE ACTIVITY; ARTICLE; CANCER CELL LINE; DRUG DESIGN; DRUG SYNTHESIS; ELECTRON SPIN RESONANCE; GROWTH INHIBITION; HELA CELL LINE; HIGH RESOLUTION MELTING ANALYSIS; HUMAN; HUMAN CELL; PROTON NUCLEAR MAGNETIC RESONANCE; SUBSTITUTION REACTION; CELL PROLIFERATION; CHEMISTRY; DRUG EFFECTS; STRUCTURE ACTIVITY RELATION; SYNTHESIS; TUMOR CELL LINE;

ANTINEOPLASTIC AGENTS; CELL LINE, TUMOR; CELL PROLIFERATION; COUMARINS; DRUG DESIGN; HELA CELLS; HUMANS; HYDRAZINES; HYDRAZONES; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84908008288     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2014.09.018     Document Type: Article

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