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Volumn 70, Issue 42, 2014, Pages 7740-7745

Synthesis of cell-permeable stapled BH3 peptide-based Mcl-1 inhibitors containing simple aryl and vinylaryl cross-linkers

(5) Muppidi, Avinash a Doi, Kenichiro b Ramil, Carlo P a Wang, Hong Gang b Lin, Qing a

a UNIVERSITY AT BUFFALO (United States)

b PENN STATE COLLEGE OF MEDICINE (United States)

Author keywords

Cross linkers; Inhibitors; Peptides; Protein protein interaction; Stapled peptides

Indexed keywords

BH3 PROTEIN; PROTEIN INHIBITOR; PROTEIN MCL 1; PROTEIN MCL 1 INHIBITOR; UNCLASSIFIED DRUG; VINYL DERIVATIVE;

ARTICLE; CELL MEMBRANE PERMEABILITY; CIRCULAR DICHROISM; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; ELECTROSPRAY MASS SPECTROMETRY; HYDROPHOBICITY; PHYSICAL CHEMISTRY; PROTEIN CROSS LINKING; PROTEIN PROTEIN INTERACTION; PROTEIN SECONDARY STRUCTURE; SIMULATION;

EID: 84907927054 PISSN: 00404020 EISSN: 14645416 Source Type: Journal
DOI: 10.1016/j.tet.2014.05.104 Document Type: Article

Times cited : (29)

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