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Bioorganic and Medicinal Chemistry Letters

Volumn 24, Issue 19, 2014, Pages 4729-4734

Design, synthesis and biological evaluation of β-boswellic acid based HDAC inhibitors as inducers of cancer cell death

(8) Sharma, Simmi a Ahmad, Mudassier a Bhat, Javeed Ahmad a Kumar, Arvind a,b Kumar, Manjeet a Zargar, Mohmmad Afzal c Hamid, Abid a Shah, Bhahwal Ali a,b

a CSIR INDIAN INSTITUTE OF INTEGRATIVE MEDICINE (India)

b ACADEMY OF SCIENTIFIC AND INNOVATIVE RESEARCH ACSIR (India)

c UNIVERSITY OF KASHMIR (India)

Author keywords

Anti cancer; HDAC; Hydroxamic acid; Boswellic acid

Indexed keywords

11 OXO BETA BOSWELLIC ACID; 3 ALPHA ACETOXY 4 BETA AMINO 11 OXO 24 NORURS 12 ENE; 3 ALPHA ACETOXY 4 BETA AMINO 24 NORURS 12 ENE; ANTINEOPLASTIC AGENT; BETA BOSWELLIC ACID DERIVATIVE; BOSWELLIC ACID; HISTONE DEACETYLASE INHIBITOR; UNCLASSIFIED DRUG; HISTONE DEACETYLASE; TRITERPENE;

A549 CELL LINE; ARTICLE; CANCER CELL DESTRUCTION; CONCENTRATION RESPONSE; CONTROLLED STUDY; CYTOTOXICITY; DRUG DESIGN; DRUG SCREENING; DRUG SYNTHESIS; ENZYME ACTIVE SITE; G1 PHASE CELL CYCLE CHECKPOINT; HCT116 CELL LINE; HL 60 CELL LINE; HUMAN; HUMAN CELL; IC50; MCF 7 CELL LINE; MITOCHONDRIAL MEMBRANE POTENTIAL; MOLECULAR MODEL; CELL CYCLE; CELL DEATH; CELL PROLIFERATION; CHEMICAL STRUCTURE; CHEMISTRY; DOSE RESPONSE; DRUG EFFECTS; METABOLISM; STRUCTURE ACTIVITY RELATION; SYNTHESIS; TUMOR CELL LINE;

ANTINEOPLASTIC AGENTS; CELL CYCLE; CELL DEATH; CELL LINE, TUMOR; CELL PROLIFERATION; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG DESIGN; DRUG SCREENING ASSAYS, ANTITUMOR; HCT116 CELLS; HISTONE DEACETYLASE INHIBITORS; HISTONE DEACETYLASES; HL-60 CELLS; HUMANS; MCF-7 CELLS; MODELS, MOLECULAR; MOLECULAR STRUCTURE; STRUCTURE-ACTIVITY RELATIONSHIP; TRITERPENES;

EID: 84907227111 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2014.08.007 Document Type: Article

Times cited : (22)

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