Development of an efficient Pd-catalyzed coupling process for axitinib

Organic Process Research and Development

Volumn 18, Issue 1, 2014, Pages 266-274

  Chekal, Brian P ^a   Guinness, Steven M ^a   Lillie, Brett M ^a   McLaughlin, Robert W ^a   Palmer, Charles W ^a   Post, Ronald J ^a   Sieser, Janice E ^a   Singer, Robert A ^a   Sluggett, Gregory W ^a   Vaidyanathan, Rajappa ^a   Withbroe, Gregory J ^a  

^a PFIZER INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

COUPLING AGENTS; OPTIMIZATION;

CONTROL STRATEGIES; COUPLING PROCESS; HECK REACTIONS; IMPURITIES IN; MANUFACTURING PROCESS; PD-CATALYZED COUPLING REACTIONS;

CATALYSIS;

EID: 84899845032     PISSN: 10836160     EISSN: 1520586X     Source Type: Journal    
DOI: 10.1021/op400088k     Document Type: Article

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