ARTICLE;
CANCER CELL CULTURE;
CHEMICAL REACTION;
CLICK REACTION;
CYCLOADDITION;
CYTOTOXICITY;
DRUG STRUCTURE;
DRUG SYNTHESIS;
HUMAN;
HUMAN CELL;
IC 50;
PROTON NUCLEAR MAGNETIC RESONANCE;
Synthesis and biological activity studies of new hybrid molecules containing tryptamine moiety
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Design and synthesis of new N-(5-trifluoromethyl)-1 H-1,2,4-triazol-3-yl benzenesulfonamides as possible antimalarial prototypes
Boechat N, Pinheiro LCS, Santos-Filho OA, Silva IC (2011) Design and synthesis of new N-(5-trifluoromethyl)-1 H-1,2,4-triazol-3-yl benzenesulfonamides as possible antimalarial prototypes. Molecules 16:8083-8097
Evaluation of a tetrazolium-based semiautomated colorimetric assay: Assessment of radiosensitivity
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Sulfonamide-1,2,4-triazole derivatives as antifungal and antibacterial agents: Synthesis, biological evaluation, lipophilicity, and conformational studies
DOI 10.1016/j.bmc.2007.10.082, PII S0968089607009509
Ezabadi IR, Camoutsis C, Zoumpoulakis P, Geronikaki A, Soković M, Glamočlija J, Cirić A (2008) Sulfonamide-1,2,4-triazole derivatives as antifungal and antibacterial agents: synthesis, biological evaluation, lipophilicity, and conformational studies. Bioorg Med Chem 16:1150-1161 (Pubitemid 351193036)
Synthesis and biological evaluation of new 3,5-di(trifluoromethyl)-1,2,4- triazolesulfonylurea and thiourea derivatives as antidiabetic and antimicrobial agents
Faidallah HM, Khan KA, Asiri AM (2011) Synthesis and biological evaluation of new 3,5-di(trifluoromethyl)-1,2,4-triazolesulfonylurea and thiourea derivatives as antidiabetic and antimicrobial agents. J Fluorine Chem 132:870-877
New triazole and triazolothiadiazine derivatives as possible antimicrobial agents
Kaplancikli ZA, Turan-Zitouni G, Ozdemir AA, Revial G (2008) New triazole and triazolothiadiazine derivatives as possible antimicrobial agents. Eur J Med Chem 43:155-159
Rapid colorimetric assay for cellular growth and survival: Application to proliferation and cytotoxicity assays
Mosmann T (1983) Rapid colorimetric assay for cellular growth and survival: application to proliferation and cytotoxicity assays. J Immunol Methods 65:55-63
Parallel synthesis of novel antitumor agents: 1,2,3-triazoles bearing biologically active sulfonamide moiety and their 3D-QSAR
Ou L, Han S, Ding W, Jia P, Yang B, Medina-Franco JL, Giulianotti MA, Chen JZ, Yu Y (2011) Parallel synthesis of novel antitumor agents: 1,2,3-triazoles bearing biologically active sulfonamide moiety and their 3D-QSAR. Mol Divers 15:927-946
Synthesis and cytotoxicity of novel N-sulfonyl-1,2,3,4- tetrahydroisoquinoline thiosemicarbazone derivatives
Pingaew R, Prachayasittikul S, Ruchirawat S, Prachayasittikul V (2013) Synthesis and cytotoxicity of novel N-sulfonyl-1,2,3,4-tetrahydroisoquinoline thiosemicarbazone derivatives. Med Chem Res 22:267-277
Design and synthesis of antibreast cancer agents from 4-piperazinylquinoline: A hybrid pharmacophore approach
Solomon VR, Hua C, Lee H (2010) Design and synthesis of antibreast cancer agents from 4-piperazinylquinoline: a hybrid pharmacophore approach. Bioorg Med Chem 18:1563-1572
COX-2 selective inhibitors, carbonic anhydrase inhibition and anticancer properties of sulfonamides belonging to this class of pharmacological agents
Supuran CT, Casini A, Mastrolorenzo A, Scozzafava A (2004) COX-2 selective inhibitors, carbonic anhydrase inhibition and cytotoxic properties of sulfonamides belonging to this class of pharmacological agents. Mini Rev Med Chem 4:625-632 (Pubitemid 38961227)
New quinolin-4-yl-1,2,3-triazoles carrying amides and amidopiperazines as potential antitubercular agents
Thomas KD, Adhikari AV, Chowdhury IH, Sumesh E, Pal NK (2011) New quinolin-4-yl-1,2,3-triazoles carrying amides and amidopiperazines as potential antitubercular agents. Eur J Med Chem 46:2503-2512
Synthesis of novel sulfanilamide-derived 1,2,3-triazoles and their evaluation for antibacterial and antifungal activities
Wang XL, Wan K, Zhou CH (2010) Synthesis of novel sulfanilamide-derived 1,2,3-triazoles and their evaluation for antibacterial and antifungal activities. Eur J Med Chem 45:4631-4639
DOI 10.1016/j.bmcl.2006.11.079, PII S0960894X06013862
Wilkinson BL, Bornaghi LF, Wright AD, Houston TA, Poulsen SA (2007) Anti-mycobacterial activity of a bis-sulfonamide. Bioorg Med Chem Lett 17:1355-1357 (Pubitemid 46240841)
Carbonic anhydrase IX: A new druggable target for the design of antitumor agents
DOI 10.1002/med.20112
Winum JY, Rami M, Scozzafava A, Montero JL, Supuran C (2008) Carbonic anhydrase IX: a new druggable target for the design of antitumor agents. Med Res Rev 28:445-463 (Pubitemid 351590542)
