메뉴 건너뛰기




Volumn 17, Issue 5, 2014, Pages 697-703

In vivo activity of modafinil on dopamine transporter measured with positron emission tomography and [18F]FE-PE2I

Author keywords

Abuse liability; dopamine transporter; modafinil; positron emission tomography

Indexed keywords

DOPAMINE TRANSPORTER; METHYLPHENIDATE; MODAFINIL; N (3 IODOPROP 2E ENYL) 2 BETA CARBOMETHOXY 3 BETA (4 METHYLPHENYL)NORTROPANE F 18; RADIOLIGAND; UNCLASSIFIED DRUG; (E)-N-(3-IODOPROP-2-ENYL)-2BETA-CARBOFLUOROETHOXY-3BETA-(4'-METHYL-PHENYL) NORTROPANE; BENZHYDRYL DERIVATIVE; NORTROPANE DERIVATIVE; RADIOPHARMACEUTICAL AGENT; WAKEFULNESS PROMOTING AGENT;

EID: 84897453966     PISSN: 14611457     EISSN: 14695111     Source Type: Journal    
DOI: 10.1017/S1461145713001612     Document Type: Article
Times cited : (36)

References (51)
  • 2
    • 77957837936 scopus 로고    scopus 로고
    • Positron emission tomography measurement of dopamine D2 receptor occupancy in the pituitary and cerebral cortex: Relation to antipsychotic- induced hyperprolactinemia
    • Arakawa R, Okumura M, Ito H, Takano A, Takahashi H, Takano H, Maeda J, Okubo Y, Suhara T (2010) Positron emission tomography measurement of dopamine D2 receptor occupancy in the pituitary and cerebral cortex: Relation to antipsychotic-induced hyperprolactinemia. J Clin Psychiatry 71:1131-1137
    • (2010) J Clin Psychiatry , vol.71 , pp. 1131-1137
    • Arakawa, R.1    Okumura, M.2    Ito, H.3    Takano, A.4    Takahashi, H.5    Takano, H.6    Maeda, J.7    Okubo, Y.8    Suhara, T.9
  • 4
    • 84876703918 scopus 로고    scopus 로고
    • Psychological and physiological effects of bupropion compared to methylphenidate after prolonged administration in healthy volunteers (NCT00285155
    • Chevassus H, Farret A, Gagnol JP, Ponçon CA, Costa F, Roux C, Galtier F, Petit P (2012) Psychological and physiological effects of bupropion compared to methylphenidate after prolonged administration in healthy volunteers (NCT00285155). Eur J Clin Pharmacol 69:779-787
    • (2012) Eur J Clin Pharmacol , vol.69 , pp. 779-787
    • Chevassus, H.1    Farret, A.2    Gagnol, J.P.3    Ponçon, C.A.4    Costa, F.5    Roux, C.6    Galtier, F.7    Petit, P.8
  • 5
    • 14444270841 scopus 로고    scopus 로고
    • Synthesis and ligand binding of nortropane derivatives: N-substituted 2beta-carbomethoxy-3beta-(4'-iodophenyl)nortropane and N-(3-iodoprop-(2E)-enyl)- 2beta-carbomethoxy-3beta-(3', 4'-disubstituted phenyl)nortropane. New high-Affinity and selective compounds for the dopamine transporter
    • Emond P, Garreau L, Chalon S, Boazi M, Caillet M, Bricard J, Frangin Y, Mauclaire L, Besnard JC, Guilloteau D (1997) Synthesis and ligand binding of nortropane derivatives: N-substituted 2beta-carbomethoxy-3beta-(4'-iodophenyl) nortropane and N-(3-iodoprop-(2E)-enyl)-2beta-carbomethoxy-3beta-(3', 4'-disubstituted phenyl)nortropane. New high-Affinity and selective compounds for the dopamine transporter. J Med Chem 40:1366-1372
    • (1997) J Med Chem , vol.40 , pp. 1366-1372
    • Emond, P.1    Garreau, L.2    Chalon, S.3    Boazi, M.4    Caillet, M.5    Bricard, J.6    Frangin, Y.7    Mauclaire, L.8    Besnard, J.C.9    Guilloteau, D.10
  • 6
    • 47149108159 scopus 로고    scopus 로고
    • PE2I: A radiopharmaceutical for in vivo exploration of the dopamine transporter
    • Emond P, Guilloteau D, Chalon S (2008) PE2I: A radiopharmaceutical for in vivo exploration of the dopamine transporter. CNS Neurosci Ther 14:47-64
    • (2008) CNS Neurosci Ther , vol.14 , pp. 47-64
    • Emond, P.1    Guilloteau, D.2    Chalon, S.3
  • 7
    • 0028178856 scopus 로고
    • PET study of [11C]beta-CIT binding to monoamine transporters in the monkey and human brain
    • Farde L, Halldin C, Muller L, Suhara T, Karlsson P, Hall H (1994) PET study of [11C]beta-CIT binding to monoamine transporters in the monkey and human brain. Synapse 16:93-103
    • (1994) Synapse , vol.16 , pp. 93-103
    • Farde, L.1    Halldin, C.2    Muller, L.3    Suhara, T.4    Karlsson, P.5    Hall, H.6
  • 9
    • 33747615950 scopus 로고    scopus 로고
    • The science of stimulant abuse
    • Greenhill LL (2006) The science of stimulant abuse. Pediatr Ann 35:552-556
    • (2006) Pediatr Ann , vol.35 , pp. 552-556
    • Greenhill, L.L.1
  • 10
    • 0029666198 scopus 로고    scopus 로고
    • Comparison of [3H]paroxetine and [3H]cyanoimipramine for quantitative measurement of serotonin transporter sites in human brain
    • Gurevich EV, Joyce JN (1996) Comparison of [3H]paroxetine and [3H]cyanoimipramine for quantitative measurement of serotonin transporter sites in human brain. Neuropsychopharmacology 14:309-323
    • (1996) Neuropsychopharmacology , vol.14 , pp. 309-323
    • Gurevich, E.V.1    Joyce, J.N.2
  • 13
    • 34547846251 scopus 로고    scopus 로고
    • Consensus nomenclature for in vivo imaging of reversibly binding radioligands
    • Innis RB et al. (2007) Consensus nomenclature for in vivo imaging of reversibly binding radioligands. J Cereb Blood Flow Metab 27:1533-1539
    • (2007) J Cereb Blood Flow Metab , vol.27 , pp. 1533-1539
    • Innis, R.B.1
  • 14
    • 0035721734 scopus 로고    scopus 로고
    • Error analysis for quantification of [11 C]FLB 457 binding to extrastriatal D(2) dopamine receptors in the human brain
    • Ito H, Sudo Y, Suhara T, Okubo Y, Halldin C, Farde L (2001) Error analysis for quantification of [(11)C]FLB 457 binding to extrastriatal D(2) dopamine receptors in the human brain. Neuroimage 13:531-539
    • (2001) Neuroimage , vol.13 , pp. 531-539
    • Ito, H.1    Sudo, Y.2    Suhara, T.3    Okubo, Y.4    Halldin, C.5    Farde, L.6
  • 15
    • 0343963779 scopus 로고    scopus 로고
    • Evaluation of the abuse liability of modafinil and other drugs for excessive daytime sleepiness associated with narcolepsy
    • Jasinski DR, Kovacević-Ristanović R (2000) Evaluation of the abuse liability of modafinil and other drugs for excessive daytime sleepiness associated with narcolepsy. Clin Neuropharmacol 23:149-156
    • (2000) Clin Neuropharmacol , vol.23 , pp. 149-156
    • Jasinski, D.R.1    Kovacević-Ristanović, R.2
  • 16
    • 33744912786 scopus 로고    scopus 로고
    • Quantitative analyses of regional [11C]PE2I binding to the dopamine transporter in the human brain: A PET study
    • Jucaite A, Odano I, Olsson H, Pauli S, Halldin C, Farde L (2006) Quantitative analyses of regional [11C]PE2I binding to the dopamine transporter in the human brain: A PET study. Eur J Nucl Med Mol Imaging 33:657-668
    • (2006) Eur J Nucl Med Mol Imaging , vol.33 , pp. 657-668
    • Jucaite, A.1    Odano, I.2    Olsson, H.3    Pauli, S.4    Halldin, C.5    Farde, L.6
  • 17
    • 0035007998 scopus 로고    scopus 로고
    • Assessing the abuse potential of methylphenidate in nonhuman and human subjects: A review
    • Kollins SH, MacDonald EK, Rush CR (2001) Assessing the abuse potential of methylphenidate in nonhuman and human subjects: A review. Pharmacol Biochem Behav 68:611-627
    • (2001) Pharmacol Biochem Behav , vol.68 , pp. 611-627
    • Kollins, S.H.1    MacDonald, E.K.2    Rush, C.R.3
  • 18
    • 34347330048 scopus 로고    scopus 로고
    • Modafinil: Mischaracterization
    • author reply 971-972
    • Kruszewski SP, Klotz SG (2007) Modafinil: Mischaracterization. J Clin Psychiatry 68:970-971; author reply 971-972
    • (2007) J Clin Psychiatry , vol.68 , pp. 970-971
    • Kruszewski, S.P.1    Klotz, S.G.2
  • 19
    • 0031594290 scopus 로고    scopus 로고
    • 18F] CFT [(18F)WIN 35428] a radioligand to study the dopamine transporter with PET: Characterization in human subjects
    • Laakso A, Bergman J, Haaparanta M, Vilkman H, Solin O, Hietala J (1998) [18F]CFT [(18F)WIN 35428], a radioligand to study the dopamine transporter with PET: Characterization in human subjects. Synapse 28:244-250
    • (1998) Synapse , vol.28 , pp. 244-250
    • Laakso, A.1    Bergman, J.2    Haaparanta, M.3    Vilkman, H.4    Solin, O.5    Hietala, J.6
  • 20
    • 0030468875 scopus 로고    scopus 로고
    • Simplified reference tissue model for PET receptor studies
    • Lammertsma AA, Hume SP (1996) Simplified reference tissue model for PET receptor studies. Neuroimage 4:153-158
    • (1996) Neuroimage , vol.4 , pp. 153-158
    • Lammertsma, A.A.1    Hume, S.P.2
  • 23
    • 0031945368 scopus 로고    scopus 로고
    • Altropane, a SPECT or PET imaging probe for dopamine neurons: I. Dopamine transporter binding in primate brain
    • Madras BK, Meltzer PC, Liang AY, Elmaleh DR, Babich J, Fischman AJ (1998) Altropane, a SPECT or PET imaging probe for dopamine neurons: I. Dopamine transporter binding in primate brain. Synapse 29:93-104
    • (1998) Synapse , vol.29 , pp. 93-104
    • Madras, B.K.1    Meltzer, P.C.2    Liang, A.Y.3    Elmaleh, D.R.4    Babich, J.5    Fischman, A.J.6
  • 25
    • 42049116942 scopus 로고    scopus 로고
    • Poll results: Look who's doping
    • Maher B (2008) Poll results: Look who's doping. Nature 452:674-675
    • (2008) Nature , vol.452 , pp. 674-675
    • Maher, B.1
  • 27
    • 43649090464 scopus 로고    scopus 로고
    • Modafinil: A review of neurochemical actions and effects on cognition
    • Minzenberg MJ, Carter CS (2008) Modafinil: A review of neurochemical actions and effects on cognition. Neuropsychopharmacology 33:1477-1502
    • (2008) Neuropsychopharmacology , vol.33 , pp. 1477-1502
    • Minzenberg, M.J.1    Carter, C.S.2
  • 28
    • 4143088220 scopus 로고    scopus 로고
    • Modafinil: Preclinical, clinical, and post-marketing surveillance-A review of abuse liability issues
    • Myrick H, Malcolm R, Taylor B, LaRowe S (2004) Modafinil: Preclinical, clinical, and post-marketing surveillance-A review of abuse liability issues. Ann Clin Psychiatry 16:101-109
    • (2004) Ann Clin Psychiatry , vol.16 , pp. 101-109
    • Myrick, H.1    Malcolm, R.2    Taylor, B.3    LaRowe, S.4
  • 29
    • 84855169033 scopus 로고    scopus 로고
    • Quantitative PET analyses of regional [11C] PE2I binding to the dopamine transporter-Application to juvenile myoclonic epilepsy
    • Odano I, Varrone A, Savic I, Ciumas C, Karlsson P, Jucaite A, Halldin C, Farde L (2012) Quantitative PET analyses of regional [11C]PE2I binding to the dopamine transporter-Application to juvenile myoclonic epilepsy. Neuroimage 59:3582-3593
    • (2012) Neuroimage , vol.59 , pp. 3582-3593
    • Odano, I.1    Varrone, A.2    Savic, I.3    Ciumas, C.4    Karlsson, P.5    Jucaite, A.6    Halldin, C.7    Farde, L.8
  • 30
    • 84859718047 scopus 로고    scopus 로고
    • Provigil (modafinil
    • PDR Network Chesanow N, Fleming H (eds, 60th edn. New Jersey: Thompson PDR
    • PDR Network (2006) Provigil (modafinil). In: Chesanow N, Fleming H (eds) Physicians' desk reference, 60th edn, pp1002-1007. New Jersey: Thompson PDR
    • (2006) Physicians' desk reference , pp. 1002-1007
  • 31
    • 0023265754 scopus 로고
    • Cocaine receptors on dopamine transporters are related to selfadministration of cocaine
    • Ritz MC, Lamb RJ, Goldberg SR, Kuhar MJ (1987) Cocaine receptors on dopamine transporters are related to selfadministration of cocaine. Science 237:1219-1223
    • (1987) Science , vol.237 , pp. 1219-1223
    • Ritz, M.C.1    Lamb, R.J.2    Goldberg, S.R.3    Kuhar, M.J.4
  • 34
    • 85047697315 scopus 로고    scopus 로고
    • Dose effects of modafinil in sustaining wakefulness in narcolepsy patients with residual evening sleepiness
    • Schwartz JR, Feldman NT, Bogan RK (2005) Dose effects of modafinil in sustaining wakefulness in narcolepsy patients with residual evening sleepiness. J Neuropsychiatry Clin Neurosci 17:405-412
    • (2005) J Neuropsychiatry Clin Neurosci , vol.17 , pp. 405-412
    • Schwartz, J.R.1    Feldman, N.T.2    Bogan, R.K.3
  • 36
    • 84875316350 scopus 로고    scopus 로고
    • Surveillance of diversion and nonmedical use of extended-release prescription amphetamine and oral methylphenidate in the United States
    • Sembower MA, Ertischek MD, Buchholtz C, Dasgupta N, Schnoll SH (2013) Surveillance of diversion and nonmedical use of extended-release prescription amphetamine and oral methylphenidate in the United States. J Addict Dis 32:26-38
    • (2013) J Addict Dis , vol.32 , pp. 26-38
    • Sembower, M.A.1    Ertischek, M.D.2    Buchholtz, C.3    Dasgupta, N.4    Schnoll, S.H.5
  • 38
    • 78049427180 scopus 로고    scopus 로고
    • A positron emission tomography study examining the dopaminergic activity of armodafinil in adults using [11C]altropane and [11C]raclopride
    • Spencer TJ, Madras BK, Bonab AA, Dougherty DD, Clarke A, Mirto T, Martin J, Fischman AJ (2010) A positron emission tomography study examining the dopaminergic activity of armodafinil in adults using [11C]altropane and [11C]raclopride. Biol Psychiatry 68:964-970
    • (2010) Biol Psychiatry , vol.68 , pp. 964-970
    • Spencer, T.J.1    Madras, B.K.2    Bonab, A.A.3    Dougherty, D.D.4    Clarke, A.5    Mirto, T.6    Martin, J.7    Fischman, A.J.8
  • 39
    • 84859128111 scopus 로고    scopus 로고
    • Understanding the central pharmacokinetics of spheroidal oral drug absorption system (SODAS) dexmethylphenidate: A positron emission tomography study of dopamine transporter receptor occupancy measured with C-11 altropane
    • Spencer TJ, Bonab AA, Dougherty DD, Mirto T, Martin J, Clarke A, Fischman AJ (2012) Understanding the central pharmacokinetics of spheroidal oral drug absorption system (SODAS) dexmethylphenidate: A positron emission tomography study of dopamine transporter receptor occupancy measured with C-11 altropane. J Clin Psychiatry 73:346-352
    • (2012) J Clin Psychiatry , vol.73 , pp. 346-352
    • Spencer, T.J.1    Bonab, A.A.2    Dougherty, D.D.3    Mirto, T.4    Martin, J.5    Clarke, A.6    Fischman, A.J.7
  • 41
    • 84874935839 scopus 로고    scopus 로고
    • Striatal and extrastriatal dopamine D2 receptor occupancy by a novel antipsychotic, Blonanserin: A PET study with [11C]Raclopride and [11C]FLB 457 in schizophrenia
    • Tateno A, Arakawa R, Okumura M, Fukuta H, Honjo K, Ishihara K, Nakamura H, Kumita S, Okubo Y (2013) Striatal and extrastriatal dopamine D2 receptor occupancy by a novel antipsychotic, Blonanserin: A PET study with [11C]Raclopride and [11C]FLB 457 in schizophrenia. J Clin Psychopharmacol 33:162-169
    • (2013) J Clin Psychopharmacol , vol.33 , pp. 162-169
    • Tateno, A.1    Arakawa, R.2    Okumura, M.3    Fukuta, H.4    Honjo, K.5    Ishihara, K.6    Nakamura, H.7    Kumita, S.8    Okubo, Y.9
  • 42
    • 3042776615 scopus 로고    scopus 로고
    • Autoradiographic distribution of serotonin transporters and receptor subtypes in human brain
    • Varnas K, Halldin C, Hall H (2004) Autoradiographic distribution of serotonin transporters and receptor subtypes in human brain. Hum Brain Mapp 22:246-260
    • (2004) Hum Brain Mapp , vol.22 , pp. 246-260
    • Varnas, K.1    Halldin, C.2    Hall, H.3
  • 43
    • 70349123080 scopus 로고    scopus 로고
    • In vitro autoradiography and in vivo evaluation in cynomolgus monkey of [18F] FE-PE2I, a new dopamine transporter PET radioligand
    • Varrone A, Steiger C, Schou M, Takano A, Finnema SJ, Guilloteau D, Gulyas B, Halldin C (2009) In vitro autoradiography and in vivo evaluation in cynomolgus monkey of [18F] FE-PE2I, a new dopamine transporter PET radioligand. Synapse 63:871-880
    • (2009) Synapse , vol.63 , pp. 871-880
    • Varrone, A.1    Steiger, C.2    Schou, M.3    Takano, A.4    Finnema, S.J.5    Guilloteau, D.6    Gulyas, B.7    Halldin, C.8
  • 44
    • 79851498843 scopus 로고    scopus 로고
    • Kinetic analysis and quantification of the dopamine transporter in the nonhuman primate brain with 11C-PE2I and 18F-FE-PE2I
    • Varrone A, Tóth M, Steiger C, Takano A, Guilloteau D, Ichise M, Gulyás B, Halldin C (2011) Kinetic analysis and quantification of the dopamine transporter in the nonhuman primate brain with 11C-PE2I and 18F-FE-PE2I. J Nucl Med 52:132-139
    • (2011) J Nucl Med , vol.52 , pp. 132-139
    • Varrone, A.1    Tóth, M.2    Steiger, C.3    Takano, A.4    Guilloteau, D.5    Ichise, M.6    Gulyás, B.7    Halldin, C.8
  • 45
    • 84856315375 scopus 로고    scopus 로고
    • Simplified quantification and whole-body distribution of [18F] FE-PE2I in nonhuman primates: Prediction for human studies
    • Varrone A, Gulyás B, Takano A, Stabin MG, Jonsson C, Halldin C (2012) Simplified quantification and whole-body distribution of [18F]FE-PE2I in nonhuman primates: Prediction for human studies. Nucl Med Biol 39:295-303
    • (2012) Nucl Med Biol , vol.39 , pp. 295-303
    • Varrone, A.1    Gulyás, B.2    Takano, A.3    Stabin, M.G.4    Jonsson, C.5    Halldin, C.6
  • 51
    • 0032979760 scopus 로고    scopus 로고
    • Open-label, single-dose pharmacokinetic study of modafinil tablets: Influence of age and gender in normal subjects
    • Wong YN, King SP, Simcoe D, Gorman S, Laughton W, McCormick GC, Grebow P (1999) Open-label, single-dose pharmacokinetic study of modafinil tablets: Influence of age and gender in normal subjects. J Clin Pharmacol 39:281-288
    • (1999) J Clin Pharmacol , vol.39 , pp. 281-288
    • Wong, Y.N.1    King, S.P.2    Simcoe, D.3    Gorman, S.4    Laughton, W.5    McCormick, G.C.6    Grebow, P.7


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.