New 4-thiazolidinones from 5-ethyl pyridine-2-ethanol: Their antibacterial, antifungal, and antitubercular activity

Medicinal Chemistry Research

Volumn 23, Issue 3, 2014, Pages 1360-1370

  Patel, Navin B ^a   Patel, Hemant R ^a   Shaikh, Faiyazalam M ^a   Rajani, Dhanji ^a  

^a VEER NARMAD SOUTH GUJARAT UNIVERSITY   (India)

Author keywords

Antibacterial; Antifungal; Antitubercular; Schiff base; Thiazolidinone

Indexed keywords

EID: 84893715814     PISSN: 10542523     EISSN: 15548120     Source Type: Journal    
DOI: 10.1007/s00044-013-0736-8     Document Type: Article

References (37)

1. Ansari KF, Lal C (2009) Synthesis and evaluation of some new benzimidazole derivatives as potential antimicrobial agents. Eur J Med Chem 44:2294-2299
2. Barbosa TP, Sousa SCO, Amorim FM, Rodrigues YKS, de Assis PAC, Caldas JPA, Oliveira MR, Vasconcellos MLAA (2011) Design, synthesis and antileishmanial in vitro activity of new series of chalcones-like compounds: a molecular hybridization approach. Bioorg Med Chem 19:4250-4256
3. Bhandari SV, Bothara KG, Raut MK, Patil AA, Sarkate AP, Mokale VJ (2008) Design, synthesis and evaluation of antiinflammatory, analgesic and ulcerogenicity studies of novel S-substituted phenacyl-1,3,4-oxadiazole-2-thiol and Schiff bases of diclofenac acid as nonulcerogenic derivatives. Bioorg Med Chem 16:1822-1831
4. Bharti SK, Nath G, Tilak R, Singh SK (2010) Synthesis, anti-bacterial and anti-fungal activities of some novel Schiff bases containing 2,4-disubstituted thiazole ring. Eur J Med Chem 45:651-660
5. Chandrappa S, Prasad SBB, Vinaya K, Kumar CSA, Thimmegowda NR, Rangappa KS (2008) Synthesis and in vitro antiproliferative activity against human cancer cell lines of novel 5-(4-methyl-benzylidene)-thiazolidine-2,4-diones. Invest New Drugs 26:437-444
6. Fuloria N, Singh V, Yar MS, Ali M (2009) Syntheis, characterization and antimicrobial evalution of novel imines and thiazolidinones. Acta Polo Pharma Drug Res 66:141-146
7. Gaonkar SL, Rai KML, Prabhuswamy B (2006) Synthesis and antimicrobial studies of a new series of 2-{4-[2-(5-ethylpyridin-2-yl)ethoxy]phenyl}-5- substituted-1,3,4-oxadiazoles. Eur J Med Chem 41:841-846
8. Gurupadayya BM, Gopal M, Padmashali B, Manohara YN (2008) Synthesis and pharmacological evalution of azetidin-2-ones and thiazolidin-4-ones encompassing benzothiazole. Ind J Pharm Sci 70(577):572
9. Kamel MM, Ali HI, Anwar MM, Mohamed NA, Soliman AM (2010) Synthesis, antitumor activity and molecular docking study of novel sulfonamide-Schiff's bases, thiazolidinones, benzothiazinones and their C-nucleoside derivatives. Eur J Med Chem 45:572-580
10. Kavitha CV, Basappa Swamy SN, Mantelingu K, Doreswamy S, Sridhar MA, Prasad JS, Kanchugarakoppal Rangappa S (2006) Synthesis of new bioactive venlafaxine analogs: novel thiazolidin-4-ones as antimicrobials. Bioorg Med Chem 14:2290-2299
11. Kucukguzel G, Kocatepe A, Clercq ED, Sahin F, Gulluce M (2006) Synthesis and biological activity of 4-thiazolidinones, thiosemicarbazides derived from diflunisal hydrazide. Eur J Med Chem 41:353-359
12. Kumar A, Rajput C, Bhati S (2007) Synthesis of 3-[4′-(p- chlorophenyl)-thiazol-2′-yl]-2-[(substituted azetidinone/thiazolidinone)- aminomethyl]-6-bromoquinazolin-4-ones as anti-inflammatory agent. Bioorg Med Chem 15:3089-3096
13. Mulwad VV, Mir AA, Parmar HT (2009) Syntheis and anntimicrobial screening of 5-benzylidine-2-imino-3-(2-oxo-2H-benzopyran-6-yl)-thiazolidin-4-one and its derivatives. Ind J Chem 48B:137-141
14. Ottana R, Maccari R, Barreca ML, Bruno G, Rotondo A, Rossi A, Chiricosta G, Paola RD, Sautebin L, Cuzzocrea S, Vigorita MG (2005) 5-Arylidene-2-imino-4- thiazolidinones: design and synthesis of novel anti-inflammatory agents. Bioorg Med Chem 13:4243-4252
15. Panneerselvam P, Rather BA, Reddy DRS, Kumar NR (2009) Synthesis and anti-microbial screening of some Schiff bases of 3-amino-6,8-dibromo-2- phenylquinazolin-4(3H)-ones. Eur J Med Chem 44:2328-2333
16. Patel NB, Patel VN (2007) Synthesis and antimicrobial evaluation of new (4-oxo-thiazolidinyl)quinazolin-4(3H)ones of 2-[(2,6-dichlorophenyl)amino] phenylacetic acid. Iran J Pham Res 6:251-258
17. Patel NB, Patel SD (2009a) Synthesis and antimicrobial studies of some 4-thiazolidinone containing fluoroquinolones analogous. Der Pharma Chemica 1(2):199-209
18. Patel NB, Patel HR (2009b) Synthesis and pharmacological studies of 5-ethyl pyridin-2-ethanol analogs derivatives. Arkivoc 12:302-321
19. Patel NB, Patel HR (2010a) Design and synthesis of 2-(5-ethyl-pyridine-2- yl) ethanol analogs as potential microbial agents. Int J Drug Design Discov 1:93-106
20. Patel NB, Patel SD (2010b) Synthesis and antimicrobial study of fluoroquinolonebased 4-thiazolidinones. Med Chem Res. doi: 10.1007/s00044-009- 9228-2
21. Patel NB, Rathod RD (2007) Syntheis and antimicrobial studies of analouges of intermediate of sildenafil. J Saudi Chem Soc 11:93-100
22. Patel NB, Shaikh FM (2010) Synthesis and anti microbial studies of new pyridine analogs 4-thiazolidinones containing 2-amino-6-methoxybenzothiazole. Saudi Pharma J 18(3):129-136. doi: 10.1016/j.jsps.2010.05.002
23. Patel NB, Khan IH, Rajani S (2010a) Pharmacological evaluation and characterizations of newly synthesized 1,2,4-triazoles. Eur J Med Chem 45:4293-4299. doi: 10.1016/j.ejmech.2010.06.031
24. Patel NB, Patel VN, Patel HR, Shaikh FM, Patel JC (2010b) Sytnhesis and microbial studies of (4-oxo-thiazolidinyl sulfonamides bearing quinazolin-4(3H)-ones. Acta Polo Pharma Drug Res 67:267-275
25. Petrikaite V, Tarasevicius E, Pavilonis A (2007) New thiazolidones-4 with sulfamethizole-2 substituent as potential antifungal and antimicrobial preparations. Biologija 53:45-50
26. Raparti V, Chitre T, Bothara K, Kumar V, Dangre S, Khachane C, Gore S, Deshmane B (2009) Novel 4-(morpholin-4-yl)-N0-(arylidene)benzohydrazides: synthesis, antimycobacterial activity and QSAR investigations. Eur J Med Chem 44:3954-3960
27. Rattan A (2000) Antimicrobials in laboratory medicine. Churchill B I Livingstone, New Delhi, pp 85-108
28. Rawal RK, Tripathi R, Katti SB, Pannecouque C, Clercq ED (2007) Design, synthesis, and evaluation of 2-aryl-3-heteroaryl-1,3-thiazolidin-4-ones as anti-HIV agents. Bioorg Med Chem 15:1725-1731
29. Ronad PM, Noolvi MN, Sapkal S, Dharbhamulla S, Maddi VS (2010) Synthesis and antimicrobial activity of 7-(2-substituted phenylthiazolidinyl)-benzopyran- 2-one derivatives. Eur J Med Chem 45:85-89. doi: 10.1016/j.ejmech.2009.09.028
30. Saeed A, Abbas N, Florke U (2007) Synthesis and antibacterial activity of some novel 2-aroylimino-3-aryl-thiazolidin-4-ones. J Braz Chem Soc 18:559-565
31. Sattigeri VJ, Soni A, Singhal S, Khan S, Pandya M, Bhateja P, Mathur T, Rattan A, Khanna JM, Mehta A (2005) Synthesis and antimicrobial activity of novel thiazolidinones. Arkivoc 2:46-59
32. Sayyed M, Mokle S, Bokhare M, Mankar A, Surwase S, Bhusare S, Vibhutea Y (2006) Synthesis of some new 2,3-diaryl-1,3-thiazolidin-4-ones as antibacterial agents. Arkivoc 2:187-192
33. Shah TJ, Desai VA (2007) Synthesis of some novel fluorinated 4-thiazolidinones containing amide linkages and their antimicrobial screening. Arkivoc 16:218-228
34. Shreenivas MT, Chetan BP, Bhat AR (2009) Synthesis and pharmacological evaluation of certain schiff bases and thiazoldine derivatives as AT1 angiotension-II(AII) receptor antagonists. J Pharma Sci Tech 1:88-94
35. Tarnalli AD, Bhat AR, Srinivas S, Sarvanan E (2008) Antiinflammatory, analgesic and antipyretic activity of certain thiazolidinones. Ind J Pharm Sci 70:159-164
36. Tatar E, Kucukguzel I, Clercq ED, Sahin F, Gulluce M (2008) Synthesis, characterization and screening of antimicrobial, antituberculosis, antiviral and anticancer activity of novel 1,3-thiazolidine-4-ones derived from 1-[2-(benzoylamino)-4- (methylthio)butyryl]-4-alkyl/arylalkyl thiosemicarbazides. Arkivoc 16:191-210
37. Vicini P, Geronikaki A, Anastasia K, Incerti M, Zani F (2006) Synthesis and antimicrobial activity of novel 2-thiazolylimino-5-arylidene-4- thiazolidinones. Bioorg Med Chem 14:3859-3864