SCOPUS 정보 검색 플랫폼

Journal of Labelled Compounds and Radiopharmaceuticals

Volumn 57, Issue 1, 2014, Pages 18-24

Synthesis and preliminary evaluation of 2-arylhydroxyquinoline derivatives for tau imaging

(9) Tago, Tetsuro a Furumoto, Shozo a,b Okamura, Nobuyuki b Harada, Ryuichi b Ishikawa, Yoichi a Arai, Hiroyuki a Yanai, Kazuhiko b Iwata, Ren a Kudo, Yukitsuka a

a TOHOKU UNIVERSITY (Japan)

b TOHOKU UNIVERSITY SCHOOL OF MEDICINE (Japan)

Author keywords

Alzheimer's disease; imaging; positron emission tomography; tau

Indexed keywords

BINDING ENERGY; DIAGNOSIS; NEURODEGENERATIVE DISEASES; PATHOLOGY; POSITRONS; PROBES; RADIOGRAPHY;

ALZHEIMERS DISEASE; BINDING AFFINITIES; CLINICAL SYMPTOMS; NEUROFIBRILLARY TANGLES; NON-INVASIVE DETECTION; POST INJECTION; SENILE PLAQUES; TAU; TAU PATHOLOGY; TAU PROTEINS;

POSITRON EMISSION TOMOGRAPHY;

AMYLOID BETA PROTEIN; CARBON 11; FLUORINE 18; QUINOLINOL DERIVATIVE; RADIOPHARMACEUTICAL AGENT; TAU PROTEIN; THK 951 C 11; UNCLASSIFIED DRUG;

ALZHEIMER DISEASE; ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; AUTORADIOGRAPHY; BINDING AFFINITY; BINDING ASSAY; BLOOD BRAIN BARRIER; CONTROLLED STUDY; DRUG SYNTHESIS; EX VIVO STUDY; FLUORESCENCE; GAMMA COUNTER; HIPPOCAMPUS; ISOTOPE LABELING; LIPOPHILICITY; MALE; MOUSE; NEUROFIBRILLARY TANGLE; NONHUMAN; POSITRON EMISSION TOMOGRAPHY; PROTEIN BINDING; RADIOACTIVITY; SUZUKI REACTION; TAUOPATHY;

ALZHEIMER'S DISEASE; IMAGING; POSITRON EMISSION TOMOGRAPHY; TAU;

AGED, 80 AND OVER; ANIMALS; CARBON RADIOISOTOPES; CHEMISTRY TECHNIQUES, SYNTHETIC; FEMALE; HIPPOCAMPUS; HUMANS; HYDROPHOBIC AND HYDROPHILIC INTERACTIONS; HYDROXYLATION; HYDROXYQUINOLINES; MICE; POSITRON-EMISSION TOMOGRAPHY; TAU PROTEINS;

EID: 84892805762 PISSN: 03624803 EISSN: 10991344 Source Type: Journal
DOI: 10.1002/jlcr.3133 Document Type: Article

Times cited : (34)

References (33)

1
- 0024601426
- K. Ogomori, T. Kitamoto, J. Tateishi, Y. Sato, M. Suetsugu, M. Abe, Am. J. Pathol. 1989, 134, 243-51.
- (1989) Am. J. Pathol. , vol.134 , pp. 243-251
- Ogomori, K.¹ Kitamoto, T.² Tateishi, J.³ Sato, Y.⁴ Suetsugu, M.⁵ Abe, M.⁶

2
- 0025863618
- H. Braak, E. Braak, Acta Neuropathol. 1991, 82, 239-59.
- (1991) Acta Neuropathol. , vol.82 , pp. 239-259
- Braak, H.¹ Braak, E.²

3
- 0037319171
- P. M. Thompson, K. M. Hayashi, G. de Zubicaray, A. L. Janke, S. E. Rose, J. Semple, D. Herman, M. S. Hong, S. S. Dittmer, D. M. Doddrell, A. W. Toga, J. Neurosci. 2003, 23, 994-1005.
- (2003) J. Neurosci. , vol.23 , pp. 994-1005
- Thompson, P.M.¹ Hayashi, K.M.² De Zubicaray, G.³ Janke, A.L.⁴ Rose, S.E.⁵ Semple, J.⁶ Herman, D.⁷ Hong, M.S.⁸ Dittmer, S.S.⁹ Doddrell, D.M.¹⁰ Toga, A.W.¹¹

4
- 84872379077
- C. R. Jack, D. S. Knopman, W. J. Jagust, R. C. Petersen, M. W. Weiner, P. S. Aisen, L. M. Shaw, P. Vemuri, H. J. Wiste, S. D. Weigand, T. G. Lesnick, V. S. Pankratz, M. C. Donohue, J. Q. Trojanowski, Lancet Neurol. 2013, 12, 207-16.
- (2013) Lancet Neurol. , vol.12 , pp. 207-216
- Jack, C.R.¹ Knopman, D.S.² Jagust, W.J.³ Petersen, R.C.⁴ Weiner, M.W.⁵ Aisen, P.S.⁶ Shaw, L.M.⁷ Vemuri, P.⁸ Wiste, H.J.⁹ Weigand, S.D.¹⁰ Lesnick, T.G.¹¹ Pankratz, V.S.¹² Donohue, M.C.¹³ Trojanowski, J.Q.¹⁴

5
- 30344455572
- E. D. Agdeppa, V. Kepe, J. Liu, S. Flores-torres, N. Satyamurthy, A. Petric, G. M. Cole, G. W. Small, S. Huang, J. R. Barrio, J. Neurosci. 2001, 21, 1-5.
- (2001) J. Neurosci. , vol.21 , pp. 1-5
- Agdeppa, E.D.¹ Kepe, V.² Liu, J.³ Flores-Torres, S.⁴ Satyamurthy, N.⁵ Petric, A.⁶ Cole, G.M.⁷ Small, G.W.⁸ Huang, S.⁹ Barrio, J.R.¹⁰

6
- 0038792263
- C. A. Mathis, Y. Wang, D. P. Holt, G. Huang, M. L. Debnath, W. E. Klunk, J. Med. Chem. 2003, 46, 2740-2754.
- (2003) J. Med. Chem. , vol.46 , pp. 2740-2754
- Mathis, C.A.¹ Wang, Y.² Holt, D.P.³ Huang, G.⁴ Debnath, M.L.⁵ Klunk, W.E.⁶

7
- 70350716476
- S. R. Choi, G. Golding, Z. Zhuang, W. Zhang, N. Lim, F. Hefti, T. E. Benedum, M. R. Kilbourn, D. Skovronsky, H. F. Kung, J. Nucl. Med. 2009, 50, 1887-94.
- (2009) J. Nucl. Med. , vol.50 , pp. 1887-1894
- Choi, S.R.¹ Golding, G.² Zhuang, Z.³ Zhang, W.⁴ Lim, N.⁵ Hefti, F.⁶ Benedum, T.E.⁷ Kilbourn, M.R.⁸ Skovronsky, D.⁹ Kung, H.F.¹⁰

8
- 34248579112
- Y. Kudo, N. Okamura, S. Furumoto, M. Tashiro, K. Furukawa, M. Maruyama, M. Itoh, R. Iwata, K. Yanai, H. Arai, J. Nucl. Med. 2007, 48, 553-561.
- (2007) J. Nucl. Med. , vol.48 , pp. 553-561
- Kudo, Y.¹ Okamura, N.² Furumoto, S.³ Tashiro, M.⁴ Furukawa, K.⁵ Maruyama, M.⁶ Itoh, M.⁷ Iwata, R.⁸ Yanai, K.⁹ Arai, H.¹⁰

9
- 0037195577
- M.-P. Kung, C. Hou, Z.-P. Zhuang, B. Zhang, D. Skovronsky, J. Q. Trojanowski, V. M.-Y. Lee, H. F. Kung, Brain res. 2002, 956, 202-10.
- (2002) Brain Res. , vol.956 , pp. 202-210
- Kung, M.-P.¹ Hou, C.² Zhuang, Z.-P.³ Zhang, B.⁴ Skovronsky, D.⁵ Trojanowski, J.Q.⁶ Lee, V.M.-Y.⁷ Kung, H.F.⁸

10
- 84860326653
- M. M. Svedberg, O. Rahman, H. Hall, Nucl. Med. Biol. 2012, 39, 484-501.
- (2012) Nucl. Med. Biol. , vol.39 , pp. 484-501
- Svedberg, M.M.¹ Rahman, O.² Hall, H.³

11
- 43849084404
- V. L. Villemagne, K. E. Pike, D. Darby, P. Maruff, G. Savage, S. Ng, U. Ackermann, T. F. Cowie, J. Currie, S. G. Chan, G. Jones, H. Tochon-Danguy, G. O'Keefe, C. L. Masters, C. C. Rowe, Neuropsychologia 2008, 46, 1688-97.
- (2008) Neuropsychologia , vol.46 , pp. 1688-1697
- Villemagne, V.L.¹ Pike, K.E.² Darby, D.³ Maruff, P.⁴ Savage, G.⁵ Ng, S.⁶ Ackermann, U.⁷ Cowie, T.F.⁸ Currie, J.⁹ Chan, S.G.¹⁰ Jones, G.¹¹ Tochon-Danguy, H.¹² O'Keefe, G.¹³ Masters, C.L.¹⁴ Rowe, C.C.¹⁵

12
- 78751546481
- C. M. Clark, J. A. Schneider, B. J. Bedell, T. G. Beach, W. B. Bilker, M. A. Mintun, M. J. Pontecorvo, F. Hefti, A. P. Carpenter, M. L. Flitter, M. J. Krautkramer, H. F. Kung, R. E. Coleman, C. H. Sadowsky, E. M. Reiman, S. P. Zehntner, D. M. Skovronsky, JAMA 2011, 305, 275-284.
- (2011) JAMA , vol.305 , pp. 275-284
- Clark, C.M.¹ Schneider, J.A.² Bedell, B.J.³ Beach, T.G.⁴ Bilker, W.B.⁵ Mintun, M.A.⁶ Pontecorvo, M.J.⁷ Hefti, F.⁸ Carpenter, A.P.⁹ Flitter, M.L.¹⁰ Krautkramer, M.J.¹¹ Kung, H.F.¹² Coleman, R.E.¹³ Sadowsky, C.H.¹⁴ Reiman, E.M.¹⁵ Zehntner, S.P.¹⁶ Skovronsky, D.M.¹⁷

13
- 79958792912
- K. Herholz, K. Ebmeier, Lancet Neurol. 2011, 10, 667-70.
- (2011) Lancet Neurol. , vol.10 , pp. 667-670
- Herholz, K.¹ Ebmeier, K.²

14
- 79551495391
- V. L. Villemagne, K. E. Pike, G. Chételat, K. A. Ellis, R. S. Mulligan, P. Bourgeat, U. Ackermann, G. Jones, C. Szoeke, O. Salvado, R. Martins, G. O'Keefe, C. A. Mathis, W. E. Klunk, D. Ames, C. L. Masters, C. C. Rowe, Ann. Neurol. 2011, 69, 181-92.
- (2011) Ann. Neurol. , vol.69 , pp. 181-192
- Villemagne, V.L.¹ Pike, K.E.² Chételat, G.³ Ellis, K.A.⁴ Mulligan, R.S.⁵ Bourgeat, P.⁶ Ackermann, U.⁷ Jones, G.⁸ Szoeke, C.⁹ Salvado, O.¹⁰ Martins, R.¹¹ O'Keefe, G.¹² Mathis, C.A.¹³ Klunk, W.E.¹⁴ Ames, D.¹⁵ Masters, C.L.¹⁶ Rowe, C.C.¹⁷

15
- 0025904444
- V. M. Lee, B. J. Balin, L. Otvos, J. Q. Trojanowski, Science 1991, 251, 675-8.
- (1991) Science , vol.251 , pp. 675-678
- Lee, V.M.¹ Balin, B.J.² Otvos, L.³ Trojanowski, J.Q.⁴

16
- 80053212816
- R. Medeiros, D. Baglietto-Vargas, F. M. LaFerla, CNS Neurosci. Ther. 2011, 17, 514-24.
- (2011) CNS Neurosci. Ther. , vol.17 , pp. 514-524
- Medeiros, R.¹ Baglietto-Vargas, D.² Laferla, F.M.³

17
- 0026740795
- P. V. Arriagada, J. H. Growdon, E. T. Hedley-Whyte, B. T. Hyman, Neurology 1992, 42, 631-631.
- (1992) Neurology , vol.42 , pp. 631-631
- Arriagada, P.V.¹ Growdon, J.H.² Hedley-Whyte, E.T.³ Hyman, B.T.⁴

18
- 0030660554
- D. W. Dickson, Neurobiol. Aging 1997, 18, S21-S26.
- (1997) Neurobiol. Aging , vol.18
- Dickson, D.W.¹

19
- 37349096335
- P. T. Nelson, G. A. Jicha, F. A. Schmitt, H. Liu, D. G. Davis, M. S. Mendiondo, E. L. Abner, W. R. Markesbery, J. Neuropathol. Exp. Neurol. 2007, 66, 1136-46.
- (2007) J. Neuropathol. Exp. Neurol. , vol.66 , pp. 1136-1146
- Nelson, P.T.¹ Jicha, G.A.² Schmitt, F.A.³ Liu, H.⁴ Davis, D.G.⁵ Mendiondo, M.S.⁶ Abner, E.L.⁷ Markesbery, W.R.⁸

20
- 84860215480
- et al.
- P. T. Nelson, I. Alafuzoff, E. H. Bigio, C. Bouras, H. Braak, N. J. Cairns, R. J. Castellani, B. J. Crain, P. Davies, K. Del Tredici, C. Duyckaerts, M. P. Frosch, V. Haroutunian, P. R. Hof, C. M. Hulette, B. T. Hyman, T. Iwatsubo, K. A. Jellinger, G. A. Jicha, et al., J. Neuropathol. Exp. Neurol. 2012, 71, 362-81.
- (2012) J. Neuropathol. Exp. Neurol. , vol.71 , pp. 362-381
- Nelson, P.T.¹ Alafuzoff, I.² Bigio, E.H.³ Bouras, C.⁴ Braak, H.⁵ Cairns, N.J.⁶ Castellani, R.J.⁷ Crain, B.J.⁸ Davies, P.⁹ Del Tredici, K.¹⁰ Duyckaerts, C.¹¹ Frosch, M.P.¹² Haroutunian, V.¹³ Hof, P.R.¹⁴ Hulette, C.M.¹⁵ Hyman, B.T.¹⁶ Iwatsubo, T.¹⁷ Jellinger, K.A.¹⁸ Jicha, G.A.¹⁹

21
- 77049090834
- L. E. Rojo, J. Alzate-Morales, I. N. Saavedra, P. Davies, R. B. Maccioni, J. Alzheimers Dis. 2010, 19, 573-89.
- (2010) J. Alzheimers Dis. , vol.19 , pp. 573-589
- Rojo, L.E.¹ Alzate-Morales, J.² Saavedra, I.N.³ Davies, P.⁴ Maccioni, R.B.⁵

22
- 84863748837
- V. Villemagne, S. Furumoto, M. T. Fodero-Tavoletti, R. Harada, R. S. Mulligan, Y. Kudo, C. L. Masters, K. Yanai, C. C. Rowe, N. Okamura, Future Neurol. 2012, 7, 409-421.
- (2012) Future Neurol. , vol.7 , pp. 409-421
- Villemagne, V.¹ Furumoto, S.² Fodero-Tavoletti, M.T.³ Harada, R.⁴ Mulligan, R.S.⁵ Kudo, Y.⁶ Masters, C.L.⁷ Yanai, K.⁸ Rowe, C.C.⁹ Okamura, N.¹⁰

23
- 84874288678
- D. T. Chien, S. Bahri, A. K. Szardenings, J. C. Walsh, F. Mu, M.-Y. Su, W. R. Shankle, A. Elizarov, H. C. Kolb, J. Alzheimer's Dis. 2013, 34, 457-68.
- (2013) J. Alzheimer's Dis. , vol.34 , pp. 457-468
- Chien, D.T.¹ Bahri, S.² Szardenings, A.K.³ Walsh, J.C.⁴ Mu, F.⁵ Su, M.-Y.⁶ Shankle, W.R.⁷ Elizarov, A.⁸ Kolb, H.C.⁹

24
- 84887416188
- et al., in press, doi: 10.1016/j.jalz.2012.11.008.
- C.-F. Xia, J. Arteaga, G. Chen, U. Gangadharmath, L. F. Gomez, D. Kasi, C. Lam, Q. Liang, C. Liu, V. P. Mocharla, F. Mu, A. Sinha, H. Su, A. K. Szardenings, J. C. Walsh, E. Wang, C. Yu, W. Zhang, T. Zhao, et al., Alzheimer's Dement. 2013, in press, doi: 10.1016/j.jalz.2012.11.008.
- (2013) Alzheimer's Dement.
- Xia, C.-F.¹ Arteaga, J.² Chen, G.³ Gangadharmath, U.⁴ Gomez, L.F.⁵ Kasi, D.⁶ Lam, C.⁷ Liang, Q.⁸ Liu, C.⁹ Mocharla, V.P.¹⁰ Mu, F.¹¹ Sinha, A.¹² Su, H.¹³ Szardenings, A.K.¹⁴ Walsh, J.C.¹⁵ Wang, E.¹⁶ Yu, C.¹⁷ Zhang, W.¹⁸ Zhao, T.¹⁹

25
- 84865602256
- et al.
- W. Zhang, J. Arteaga, D. K. Cashion, G. Chen, U. Gangadharmath, L. F. Gomez, D. Kasi, C. Lam, Q. Liang, C. Liu, V. P. Mocharla, F. Mu, A. Sinha, A. K. Szardenings, E. Wang, J. C. Walsh, C. Xia, C. Yu, T. Zhao, et al., J. Alzheimer's Dis. 2012, 31, 601-12.
- (2012) J. Alzheimer's Dis. , vol.31 , pp. 601-612
- Zhang, W.¹ Arteaga, J.² Cashion, D.K.³ Chen, G.⁴ Gangadharmath, U.⁵ Gomez, L.F.⁶ Kasi, D.⁷ Lam, C.⁸ Liang, Q.⁹ Liu, C.¹⁰ Mocharla, V.P.¹¹ Mu, F.¹² Sinha, A.¹³ Szardenings, A.K.¹⁴ Wang, E.¹⁵ Walsh, J.C.¹⁶ Xia, C.¹⁷ Yu, C.¹⁸ Zhao, T.¹⁹

26
- 28044460038
- N. Okamura, T. Suemoto, S. Furumoto, M. Suzuki, H. Shimadzu, H. Akatsu, T. Yamamoto, H. Fujiwara, M. Nemoto, M. Maruyama, H. Arai, K. Yanai, T. Sawada, Y. Kudo, J. Neurosci. 2005, 25, 10857-62.
- (2005) J. Neurosci. , vol.25 , pp. 10857-10862
- Okamura, N.¹ Suemoto, T.² Furumoto, S.³ Suzuki, M.⁴ Shimadzu, H.⁵ Akatsu, H.⁶ Yamamoto, T.⁷ Fujiwara, H.⁸ Nemoto, M.⁹ Maruyama, M.¹⁰ Arai, H.¹¹ Yanai, K.¹² Sawada, T.¹³ Kudo, Y.¹⁴

27
- 79953651513
- M. T. Fodero-Tavoletti, N. Okamura, S. Furumoto, R. S. Mulligan, A. R. Connor, C. A. McLean, D. Cao, A. Rigopoulos, G. A. Cartwright, G. O'Keefe, S. Gong, P. A. Adlard, K. J. Barnham, C. C. Rowe, C. L. Masters, Y. Kudo, R. Cappai, K. Yanai, V. L. Villemagne, Brain 2011, 134, 1089-100.
- (2011) Brain , vol.134 , pp. 1089-1100
- Fodero-Tavoletti, M.T.¹ Okamura, N.² Furumoto, S.³ Mulligan, R.S.⁴ Connor, A.R.⁵ McLean, C.A.⁶ Cao, D.⁷ Rigopoulos, A.⁸ Cartwright, G.A.⁹ O'Keefe, G.¹⁰ Gong, S.¹¹ Adlard, P.A.¹² Barnham, K.J.¹³ Rowe, C.C.¹⁴ Masters, C.L.¹⁵ Kudo, Y.¹⁶ Cappai, R.¹⁷ Yanai, K.¹⁸ Villemagne, V.L.¹⁹

28
- 84881451115
- N. Okamura, S. Furumoto, R. Harada, T. Tago, T. Yoshikawa, M. Fodero-Tavoletti, R. S. Mulligan, V. L. Villemagne, H. Akatsu, T. Yamamoto, H. Arai, R. Iwata, K. Yanai, Y. Kudo, J. Nucl. Med. 2013, 54, 1420-7.
- (2013) J. Nucl. Med. , vol.54 , pp. 1420-1427
- Okamura, N.¹ Furumoto, S.² Harada, R.³ Tago, T.⁴ Yoshikawa, T.⁵ Fodero-Tavoletti, M.⁶ Mulligan, R.S.⁷ Villemagne, V.L.⁸ Akatsu, H.⁹ Yamamoto, T.¹⁰ Arai, H.¹¹ Iwata, R.¹² Yanai, K.¹³ Kudo, Y.¹⁴

29
- 80051753142
- OECD GUIDELINE FOR THE TESTING OF CHEMICALS doi: 10.1787/9789264069824-en
- OECD GUIDELINE FOR THE TESTING OF CHEMICALS, Partition coefficient (n-octanol/water), high performance liquid chromatography (HPLC) method, doi: 10.1787/9789264069824-en.
- Partition Coefficient (N-octanol/water), High Performance Liquid Chromatography (HPLC) Method

30
- 0037126688
- S. Barghorn, E. Mandelkow, Biochemistry 2002, 41, 14885-96.
- (2002) Biochemistry , vol.41 , pp. 14885-14896
- Barghorn, S.¹ Mandelkow, E.²

31
- 12144289490
- N. Okamura, T. Suemoto, H. Shimadzu, M. Suzuki, T. Shiomitsu, H. Akatsu, T. Yamamoto, M. Staufenbiel, K. Yanai, H. Arai, H. Sasaki, Y. Kudo, T. Sawada, J. Neurosci. 2004, 24, 2535-41.
- (2004) J. Neurosci. , vol.24 , pp. 2535-2541
- Okamura, N.¹ Suemoto, T.² Shimadzu, H.³ Suzuki, M.⁴ Shiomitsu, T.⁵ Akatsu, H.⁶ Yamamoto, T.⁷ Staufenbiel, M.⁸ Yanai, K.⁹ Arai, H.¹⁰ Sasaki, H.¹¹ Kudo, Y.¹² Sawada, T.¹³

32
- 78049301875
- M. Biancalana, S. Koide, Biochim. Biophys. Acta 2010, 1804, 1405-12.
- (1804) Biochim. Biophys. Acta , vol.2010 , pp. 1405-1412
- Biancalana, M.¹ Koide, S.²

33
- 84882238957
- A. Forsberg, A. Juréus, Z. Cselényi, M. Eriksdotter, Y. Freund-Levi, F. Jeppsson, B.-M. Swahn, J. Sandell, P. Julin, M. Schou, J. Andersson, P. Johnström, K. Varnäs, C. Halldin, L. Farde, S. Svensson, Eur. J. Nucl. Med. Mol. Imaging 2013, 40, 580-93.
- (2013) Eur. J. Nucl. Med. Mol. Imaging , vol.40 , pp. 580-593
- Forsberg, A.¹ Juréus, A.² Cselényi, Z.³ Eriksdotter, M.⁴ Freund-Levi, Y.⁵ Jeppsson, F.⁶ Swahn, B.-M.⁷ Sandell, J.⁸ Julin, P.⁹ Schou, M.¹⁰ Andersson, J.¹¹ Johnström, P.¹² Varnäs, K.¹³ Halldin, C.¹⁴ Farde, L.¹⁵ Svensson, S.¹⁶

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.