메뉴 건너뛰기




Volumn 33, Issue 10, 2013, Pages 4285-4292

Development and pharmacokinetic evaluation of a curcumin co-solvent formulation

Author keywords

Curcumin formulation; Intramuscular; Pharmacokinetics

Indexed keywords

COSOLVENT; CURCUMIN; SOLVENT; UNCLASSIFIED DRUG;

EID: 84891369406     PISSN: 02507005     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article
Times cited : (33)

References (40)
  • 2
    • 1242307990 scopus 로고    scopus 로고
    • Protective effect of curcumin against lead neurotoxicity in rat
    • Shukla PK, Khanna VK, Khan MY et al: Protective effect of curcumin against lead neurotoxicity in rat. Hum Exp Toxicol 22: 653-658, 2003.
    • (2003) Hum Exp Toxicol , vol.22 , pp. 653-658
    • Shukla, P.K.1    Khanna, V.K.2    Khan, M.Y.3
  • 3
    • 0032991568 scopus 로고    scopus 로고
    • Curcumin inhibition of inflammatory cytokine production by human peripheralblood monocytes and alveolar macrophages
    • Abe Y, Hashimoto S and Horie T: Curcumin inhibition of inflammatory cytokine production by human peripheralblood monocytes and alveolar macrophages. Pharmacol Res 39: 41-47, 1999.
    • (1999) Pharmacol Res , vol.39 , pp. 41-47
    • Abe, Y.1    Hashimoto, S.2    Horie, T.3
  • 4
    • 36248994780 scopus 로고    scopus 로고
    • Antihyperlipidemic effect of curcumin and tetrahydrocurcumin in experimental type 2 diabetic rats
    • Pari L and Murugan P: Antihyperlipidemic effect of curcumin and tetrahydrocurcumin in experimental type 2 diabetic rats. Ren Fail 29: 881-889, 2007.
    • (2007) Ren Fail , vol.29 , pp. 881-889
    • Pari, L.1    Murugan, P.2
  • 5
    • 0037236792 scopus 로고    scopus 로고
    • Anticancer potential of curcumin: Preclinical and clinical studies
    • Aggarwal BB, Kumar A and Bharthi AC: Anticancer potential of curcumin: preclinical and clinical studies. Anticancer Res 23: 363-398, 2003.
    • (2003) Anticancer Res , vol.23 , pp. 363-398
    • Aggarwal, B.B.1    Kumar, A.2    Bharthi, A.C.3
  • 6
    • 57649179663 scopus 로고    scopus 로고
    • Anti-angiogenic effect of curcumin in pure versus in extract forms
    • Liu D, Schwimer J, Liu Z et al: Anti-angiogenic effect of curcumin in pure versus in extract forms. Pharm Biol 46: 677-682, 2008.
    • (2008) Pharm Biol , vol.46 , pp. 677-682
    • Liu, D.1    Schwimer, J.2    Liu, Z.3
  • 7
    • 0018891247 scopus 로고
    • Toxicity studies on turmeric (Curcuma longa): Acute toxicity studies in rats, guinea pigs and monkeys
    • Shankar TN, Shantha NV, Ramesh HP et al: Toxicity studies on turmeric (Curcuma longa): acute toxicity studies in rats, guinea pigs and monkeys. Indian J Exp Biol 18: 73-75, 1980.
    • (1980) Indian J Exp Biol , vol.18 , pp. 73-75
    • Shankar, T.N.1    Shantha, N.V.2    Ramesh, H.P.3
  • 8
    • 0026548715 scopus 로고
    • Toxicity studies on Alpiniagalanga and Curcuma longa
    • Qureshi S, Shah AH and Ageel AM: Toxicity studies on Alpiniagalanga and Curcuma longa. Planta Med 58: 124-127, 1992.
    • (1992) Planta Med , vol.58 , pp. 124-127
    • Qureshi, S.1    Shah, A.H.2    Ageel, A.M.3
  • 9
    • 33845365001 scopus 로고    scopus 로고
    • Targeting events in melanoma carcinogenesis for the prevention of melanoma
    • Lao CD, Demierre MF and Sondak VK: Targeting events in melanoma carcinogenesis for the prevention of melanoma. Expert Rev Anti-cancer Ther 6: 1559-1568, 2006.
    • (2006) Expert Rev Anti-cancer Ther , vol.6 , pp. 1559-1568
    • Lao, C.D.1    Demierre, M.F.2    Sondak, V.K.3
  • 11
    • 0035174504 scopus 로고    scopus 로고
    • Phase I clinical trial of curcumin, a chemo preventive agent in patients with high-risk or pre-malignant lesions
    • Cheng AL, Hsu CH, Lin JK et al: Phase I clinical trial of curcumin, a chemo preventive agent in patients with high-risk or pre-malignant lesions. Anticancer Res 21: 2895-2900, 2001.
    • (2001) Anticancer Res , vol.21 , pp. 2895-2900
    • Cheng, A.L.1    Hsu, C.H.2    Lin, J.K.3
  • 12
    • 79551514621 scopus 로고    scopus 로고
    • Identification of permeability-related hurdles in oral delivery of curcumin using the Caco-2 cell model
    • Wahlang B, Pawar YB and Bansal AK: Identification of permeability-related hurdles in oral delivery of curcumin using the Caco-2 cell model. Euro J Pharm Biopharm 77: 275-282, 2011.
    • (2011) Euro J Pharm Biopharm , vol.77 , pp. 275-282
    • Wahlang, B.1    Pawar, Y.B.2    Bansal, A.K.3
  • 13
    • 0036917173 scopus 로고    scopus 로고
    • Solubility, chemical and photochemical stability of curcumin in surfactant solutions. Studies of curcumin and curcuminoids XXVII
    • Tonnesen HH: Solubility, chemical and photochemical stability of curcumin in surfactant solutions. Studies of curcumin and curcuminoids XXVII. Pharmazie 57: 820-824, 2002.
    • (2002) Pharmazie , vol.57 , pp. 820-824
    • Tonnesen, H.H.1
  • 14
    • 0037026270 scopus 로고    scopus 로고
    • Studies of curcumin and curcuminoids XXVII. Cyclodextrin complexation: Solubility, chemical and photochemical stability
    • Tonnesen HH, Masson M and Loftsson T: Studies of curcumin and curcuminoids XXVII. Cyclodextrin complexation: Solubility, chemical and photochemical stability. Int J Pharm 244: 127-135, 2002.
    • (2002) Int J Pharm , vol.244 , pp. 127-135
    • Tonnesen, H.H.1    Masson, M.2    Loftsson, T.3
  • 15
    • 34249977666 scopus 로고    scopus 로고
    • Oral bioavailability of curcumin in rat and the herbal analysis from Curcuma longa by LC-MS/MS
    • Yang KY, Lin LC, Tseng TU et al: Oral bioavailability of curcumin in rat and the herbal analysis from Curcuma longa by LC-MS/MS. J Chromatogr B Analyt Technol Biomed Life Sci 853: 183-189, 2007.
    • (2007) J Chromatogr B Analyt Technol Biomed Life Sci , vol.853 , pp. 183-189
    • Yang, K.Y.1    Lin, L.C.2    Tseng, T.U.3
  • 16
    • 0031860081 scopus 로고    scopus 로고
    • Influence of piperine on the pharmacokinetics of curcumin in animals and human volunteers
    • Shoba G, Joy D, Joseph T et al: Influence of piperine on the pharmacokinetics of curcumin in animals and human volunteers. Planta Med 64: 353-356, 1998.
    • (1998) Planta Med , vol.64 , pp. 353-356
    • Shoba, G.1    Joy, D.2    Joseph, T.3
  • 17
    • 77949844000 scopus 로고    scopus 로고
    • Formulation design and photochemical studies on nanocrystal solid dispersion of curcumin with improved oral bioavailability
    • Onoue S, Takahashi H, Kawabata Y et al: Formulation design and photochemical studies on nanocrystal solid dispersion of curcumin with improved oral bioavailability. J Pharm Sci 99: 1871-1881, 2010.
    • (2010) J Pharm Sci , vol.99 , pp. 1871-1881
    • Onoue, S.1    Takahashi, H.2    Kawabata, Y.3
  • 18
    • 84856974148 scopus 로고    scopus 로고
    • Preparation and pharmacokinetic evaluation of curcumin solid dispersion using Solutol® HS15 as a carrier
    • Seo SW, Han HK, Chun MK et al: Preparation and pharmacokinetic evaluation of curcumin solid dispersion using Solutol® HS15 as a carrier. Int J Pharm 424: 18-25, 2012.
    • (2012) Int J Pharm , vol.424 , pp. 18-25
    • Seo, S.W.1    Han, H.K.2    Chun, M.K.3
  • 19
    • 36549042006 scopus 로고    scopus 로고
    • Solid dispersions as strategy to improve oral bioavailability of poor water soluble drugs
    • Vasconcelos T, Sarmento B and Costa P: Solid dispersions as strategy to improve oral bioavailability of poor water soluble drugs. Drug Discov Today 12: 1068-1075, 2007.
    • (2007) Drug Discov Today , vol.12 , pp. 1068-1075
    • Vasconcelos, T.1    Sarmento, B.2    Costa, P.3
  • 20
    • 70349902499 scopus 로고    scopus 로고
    • Evaluation of an oral carrier system in rats: Bioavailability and antioxidant properties of liposome-encapsulated curcumin
    • Takahashi M, Uechi S, Takara K et al: Evaluation of an oral carrier system in rats: bioavailability and antioxidant properties of liposome-encapsulated curcumin. J Agric Food Chem 57: 9141-9146, 2009.
    • (2009) J Agric Food Chem , vol.57 , pp. 9141-9146
    • Takahashi, M.1    Uechi, S.2    Takara, K.3
  • 21
    • 77953958625 scopus 로고    scopus 로고
    • The in vitro stability and in-vivo pharmacokinetics of curcumin prepared as an aqueous nanoparticulate formulation
    • Mohanty C and Sahoo SK: The in vitro stability and in-vivo pharmacokinetics of curcumin prepared as an aqueous nanoparticulate formulation. Bio-materials 25: 6597-6611, 2010.
    • (2010) Bio-materials , vol.25 , pp. 6597-6611
    • Mohanty, C.1    Sahoo, S.K.2
  • 22
    • 37549051274 scopus 로고    scopus 로고
    • Bioavailability of curcumin: Problems and promises
    • Anand P, Kunnumakkara AB, Newman RA et al: Bioavailability of curcumin: problems and promises. Mol Pharm 4: 807-818, 2007.
    • (2007) Mol Pharm , vol.4 , pp. 807-818
    • Anand, P.1    Kunnumakkara, A.B.2    Newman, R.A.3
  • 23
    • 80051487233 scopus 로고    scopus 로고
    • Advanced drug delivery systems of curcumin for cancer chemoprevention
    • Bansal SS, Goel M, Aqil F et al: Advanced drug delivery systems of curcumin for cancer chemoprevention. Cancer Prev Res (phila) 4: 1158-1171, 2011.
    • (2011) Cancer Prev Res (Phila) , vol.4 , pp. 1158-1171
    • Bansal, S.S.1    Goel, M.2    Aqil, F.3
  • 25
    • 4544383493 scopus 로고    scopus 로고
    • Nanosuspensions in drug delivery
    • RabinowBE: Nanosuspensions in drug delivery. Nat Rev Drug Discov 3: 785-796, 2004.
    • (2004) Nat Rev Drug Discov , vol.3 , pp. 785-796
    • Rabinow, B.E.1
  • 26
    • 79954481950 scopus 로고    scopus 로고
    • Sustained-release progesterone nanosuspension following intramuscular injection in ovariectomized rats
    • Salem HF: Sustained-release progesterone nanosuspension following intramuscular injection in ovariectomized rats. Int J Nanomedicine 5: 943-954, 2010.
    • (2010) Int J Nanomedicine , vol.5 , pp. 943-954
    • Salem, H.F.1
  • 27
    • 83555162530 scopus 로고    scopus 로고
    • Sustained-release delivery of octreotide from biodegradable polymeric microspheres
    • Rhee YS, Sohn M, Woo BH et al: Sustained-release delivery of octreotide from biodegradable polymeric microspheres. AAPSPharmSciTech 4: 1293-1301, 2011.
    • (2011) AAPSPharmSciTech , vol.4 , pp. 1293-1301
    • Rhee, Y.S.1    Sohn, M.2    Woo, B.H.3
  • 28
    • 84865378492 scopus 로고    scopus 로고
    • Development of biodegradable in situ implant and microparticle injectable formulations for sustained delivery of haloperidol
    • Ahmed TA, Ibrahim HM, Ibrahim F et al: Development of biodegradable in situ implant and microparticle injectable formulations for sustained delivery of haloperidol. J Pharm Sci 101: 3753-3762, 2012.
    • (2012) J Pharm Sci , vol.101 , pp. 3753-3762
    • Ahmed, T.A.1    Ibrahim, H.M.2    Ibrahim, F.3
  • 29
    • 44649099522 scopus 로고    scopus 로고
    • Formulation of a geldanamycinprodrug in mPEG-b-PCL micelles greatly enhances tolerability and pharmacokinetics in rats
    • Xiong MP, Yariez JA, Remsberg CM et al: Formulation of a geldanamycinprodrug in mPEG-b-PCL micelles greatly enhances tolerability and pharmacokinetics in rats. J Control Release 129: 33-40, 2008.
    • (2008) J Control Release , vol.129 , pp. 33-40
    • Xiong, M.P.1    Yariez, J.A.2    Remsberg, C.M.3
  • 30
    • 32444435388 scopus 로고    scopus 로고
    • Validated LC/MS/MS assay for curcumin and tetrahydrocurcumin in rat plasma and application to pharmacokinetic study of phospholipid complex of curcumin
    • Liu A, Lou H, Zhao L et al: Validated LC/MS/MS assay for curcumin and tetrahydrocurcumin in rat plasma and application to pharmacokinetic study of phospholipid complex of curcumin. J Pharm Biomed Anal 40: 720-727, 2006.
    • (2006) J Pharm Biomed Anal , vol.40 , pp. 720-727
    • Liu, A.1    Lou, H.2    Zhao, L.3
  • 31
    • 67349107075 scopus 로고    scopus 로고
    • Nanoparticle encapsulation improves oral bioavailability of curcumin by at least 9-fold when compared to curcumin administered with piperine as absorption enhancer
    • Shaikh J, Ankola DD, Beniwal V et al: Nanoparticle encapsulation improves oral bioavailability of curcumin by at least 9-fold when compared to curcumin administered with piperine as absorption enhancer. Eur J Pharm Sci 37: 223-230, 2009.
    • (2009) Eur J Pharm Sci , vol.37 , pp. 223-230
    • Shaikh, J.1    Ankola, D.D.2    Beniwal, V.3
  • 32
    • 70449637229 scopus 로고    scopus 로고
    • Design of curcumin-loaded PLGA nanoparticles formulation with enhanced cellular uptake, and increased bioactivity in vitro and superior bioavailability in-vivo
    • Anand P, Nair HB, Sung B et al: Design of curcumin-loaded PLGA nanoparticles formulation with enhanced cellular uptake, and increased bioactivity in vitro and superior bioavailability in-vivo Biochem Pharmacol 79: 330-338, 2010.
    • (2010) Biochem Pharmacol , vol.79 , pp. 330-338
    • Anand, P.1    Nair, H.B.2    Sung, B.3
  • 33
    • 77953958625 scopus 로고    scopus 로고
    • The in vitro stability and in vivo pharmacokinetics of curcumin prepared as an aqueous nanoparticulate formulation
    • Mohanty C and Sahoo SK: The in vitro stability and in vivo pharmacokinetics of curcumin prepared as an aqueous nanoparticulate formulation. Bio-materials 25: 6597-6611, 2010.
    • (2010) Bio-materials , vol.25 , pp. 6597-6611
    • Mohanty, C.1    Sahoo, S.K.2
  • 34
    • 84866758727 scopus 로고    scopus 로고
    • Paediatric Intramuscular Injections for Developing World Settings: A Review of the Literature for Best Practices
    • Walters MC and Furyk J: Paediatric Intramuscular Injections for Developing World Settings: A Review of the Literature for Best Practices. J Transcult Nurs 23: 406-409, 2012.
    • (2012) J Transcult Nurs , vol.23 , pp. 406-409
    • Walters, M.C.1    Furyk, J.2
  • 35
    • 84877281314 scopus 로고    scopus 로고
    • Oily nanosuspension for long-acting intramuscular delivery of curcumin didecanoate prodrug: Preparation characterization and in vivo evaluation
    • Wei XL, Han YR, Quan LH et al: Oily nanosuspension for long-acting intramuscular delivery of curcumin didecanoate prodrug: Preparation characterization and in vivo evaluation. Eur J Pharm Sci 49: 286-293, 2013.
    • (2013) Eur J Pharm Sci , vol.49 , pp. 286-293
    • Wei, X.L.1    Han, Y.R.2    Quan, L.H.3
  • 36
    • 1242337285 scopus 로고    scopus 로고
    • Solubilizing excipients in oral and injectable formulations
    • Strickley RG: Solubilizing excipients in oral and injectable formulations. Pharm Res 21: 201-300, 2004.
    • (2004) Pharm Res , vol.21 , pp. 201-300
    • Strickley, R.G.1
  • 37
    • 34548039925 scopus 로고    scopus 로고
    • Solubility of sparingly-soluble ionizable drugs
    • Avdeef A: Solubility of sparingly-soluble ionizable drugs. Adv Drug Deliv Rev 59: 568-590, 2007.
    • (2007) Adv Drug Deliv Rev , vol.59 , pp. 568-590
    • Avdeef, A.1
  • 38
    • 0020647736 scopus 로고
    • The biodegradation of N-methyl-2-pyrrolidone in water by sewage bacteria
    • Chow ST and Ng TL: The biodegradation of N-methyl-2-pyrrolidone in water by sewage bacteria. Water Res 17: 117-118, 1983.
    • (1983) Water Res , vol.17 , pp. 117-118
    • Chow, S.T.1    Ng, T.L.2
  • 39
    • 78650325260 scopus 로고    scopus 로고
    • Review of pharmaceutical applications of N-methyl-2-pyrrolidone
    • Jouyban A, Fakhree MA and Shayanfar A: Review of pharmaceutical applications of N-methyl-2-pyrrolidone. J Pharm Pharm Sci 13: 524-535, 2010.
    • (2010) J Pharm Pharm Sci , vol.13 , pp. 524-535
    • Jouyban, A.1    Fakhree, M.A.2    Shayanfar, A.3
  • 40
    • 67349179610 scopus 로고    scopus 로고
    • Nanoparticle-based targeted drug delivery
    • Singh R and Lillard JW Jr.: Nanoparticle-based targeted drug delivery. Exp Mol Pathol 86: 215-223, 2009.
    • (2009) Exp Mol Pathol , vol.86 , pp. 215-223
    • Singh, R.1    Lillard Jr., J.W.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.