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Volumn 424, Issue 1-2, 2012, Pages 18-25

Preparation and pharmacokinetic evaluation of curcumin solid dispersion using Solutol ® HS15 as a carrier

Author keywords

Bioavailability; Chemical stability; Dissolution; Solubility; Solvent method

Indexed keywords

CREMOPHOR; CURCUMIN; POVIDONE; SOLUTOL HS 15;

EID: 84856974148     PISSN: 03785173     EISSN: 18733476     Source Type: Journal    
DOI: 10.1016/j.ijpharm.2011.12.051     Document Type: Article
Times cited : (102)

References (28)
  • 2
    • 8044223405 scopus 로고    scopus 로고
    • Hypolipidemic action of curcumin, the active principle of turmeric (Curcuma longa) in streptozotocin induced diabetic rats
    • DOI 10.1023/A:1006819605211
    • P.S. Babu, and K. Srinivasan Hypolipidemic action of curcumin, the active principle of tumeric (Curcuma longa) in streptozotocin induced diabetic rats Mol. Cell. Biochem. 166 1997 169 175 (Pubitemid 27085099)
    • (1997) Molecular and Cellular Biochemistry , vol.166 , Issue.1-2 , pp. 169-175
    • Suresh Babu, P.1    Srinivasan, K.2
  • 3
    • 0018887037 scopus 로고
    • Preliminary study on antirheumatic activity of curcumin (diferuloyl methane)
    • S.D. Deodhar, R. Sethi, and R.C. Srimal Preliminary study on antirhematic activity of curcumin (diferuloyl methane) Indian J. Med. Res. 71 1980 632 634 (Pubitemid 10058826)
    • (1980) Indian Journal of Medical Research , vol.71 , Issue.4 , pp. 632-634
    • Deodhar, S.D.1    Sethi, R.2    Srimal, R.C.3
  • 4
    • 0037074108 scopus 로고    scopus 로고
    • The mechanism of drug release from solid dispersion in water-soluble polymers
    • D.Q.M. Graig The mechanism of drug release from solid dispersion in water-soluble polymers Int. J. Pharm. 231 2002 131 144
    • (2002) Int. J. Pharm. , vol.231 , pp. 131-144
    • Graig, D.Q.M.1
  • 5
    • 24944508639 scopus 로고    scopus 로고
    • Improved solubility and dissolution rate of piroxicam using gelucire 44/14 and labrasol
    • DOI 10.1016/j.farmac.2005.04.014, PII S0014827X05001382
    • A. Karata, N. Yüksel, and T. Baykara Improved solubility and dissolution rate of piroxicam using gelucire 44/14 and labrasol Farmaco 60 2005 777 782 (Pubitemid 41317704)
    • (2005) Farmaco , vol.60 , Issue.9 , pp. 777-782
    • Karatas, A.1    Yuksel, N.2    Baykara, T.3
  • 6
    • 0021033789 scopus 로고
    • Antihepatotoxic principles of Curcuma longa rhizomes
    • Y. Kiso, Y. Suzuki, N. Watanabe, Y. Oshima, and H. Hikino Antihepatotoxic principles of Curcuma longa rhizomes Planta Med. 49 1983 185 187 (Pubitemid 14220766)
    • (1983) Planta Medica , vol.49 , Issue.3 , pp. 185-187
    • Kiso, Y.1    Suzuki, Y.2    Watanabe, N.3
  • 7
    • 0035895309 scopus 로고    scopus 로고
    • 10: Formulation development and bioavailability assessment
    • DOI 10.1016/S0378-5173(00)00614-1, PII S0378517300006141
    • T.R. Kommuru, B. Gurley, M.A. Khan, and I.K. Reddy Self-emulsifying drug delivery systems (SEDDS) of Coenzyme Q10: formulation development and bioavailability assessment Int. J. Pharm. 212 2001 233 246 (Pubitemid 32119449)
    • (2001) International Journal of Pharmaceutics , vol.212 , Issue.2 , pp. 233-246
    • Kommuru, T.R.1    Gurley, B.2    Khan, M.A.3    Reddy, I.K.4
  • 8
    • 0022357855 scopus 로고
    • Potential anticancer activity of turmeric (Curcuma longa)
    • DOI 10.1016/0304-3835(85)90159-4
    • R. Kuttan, P. Bhanumathy, K. Nirmala, and M.C. George Potential anticancer activity of tumeric (Curcuma longa) Cancer Lett. 29 1985 197 202 (Pubitemid 16175818)
    • (1985) Cancer Letters , vol.29 , Issue.2 , pp. 197-202
    • Kuttan, R.1    Bhanumathy, P.2    Nirmala, K.3    George, M.C.4
  • 10
    • 0034601240 scopus 로고    scopus 로고
    • Improving drug solubility for oral delivery using solid dispersions
    • DOI 10.1016/S0939-6411(00)00076-X, PII S093964110000076X
    • C. Leuner, and J. Dressman Improving drug solubility for oral delivery using solid dispersion Eur. J. Pharm. Biopharm. 50 2000 47 60 (Pubitemid 30326688)
    • (2000) European Journal of Pharmaceutics and Biopharmaceutics , vol.50 , Issue.1 , pp. 47-60
    • Leuner, C.1    Dressman, J.2
  • 11
    • 33845484838 scopus 로고    scopus 로고
    • Bioavailability enhancement of an active substance by supercritical antisolvent precipitation
    • DOI 10.1016/j.supflu.2006.03.027, PII S0896844606001100
    • V. Majerik, G. Charbit, E. Badens, G. Horváth, L. Szokonya, N. Bosc, and E. Teillaud Bioavailability enhancement of an active substance by supercritical antisolvent precipitation J. Supercrit. Fluids 40 2007 101 110 (Pubitemid 44914177)
    • (2007) Journal of Supercritical Fluids , vol.40 , Issue.1 , pp. 101-110
    • Majerik, V.1    Charbit, G.2    Badens, E.3    Horvath, G.4    Szokonya, L.5    Bosc, N.6    Teillaud, E.7
  • 12
    • 45749102576 scopus 로고    scopus 로고
    • Encapsulation of curcumin in cationic micelles suppresses alkaline hydrolysis
    • H.M.L. Mandy, H. Colangelo, and T.W. Kee Encapsulation of curcumin in cationic micelles suppresses alkaline hydrolysis Langmuir 24 2008 5672 5675
    • (2008) Langmuir , vol.24 , pp. 5672-5675
    • Mandy, H.M.L.1    Colangelo, H.2    Kee, T.W.3
  • 13
    • 0030002254 scopus 로고    scopus 로고
    • Protective role of curcumin against isoproterenol induced myocardial infarction in rats
    • DOI 10.1007/BF00420910
    • C. Nirmala, and R. Puvanakrishnan Protective role of curcumin against isoproterenol induced myocardial infraction in rats Mol. Cell. Biochem. 159 1996 85 93 (Pubitemid 26252465)
    • (1996) Molecular and Cellular Biochemistry , vol.159 , Issue.2 , pp. 85-93
    • Nirmala, C.1    Puvanakrishnan, R.2
  • 14
    • 1142297630 scopus 로고    scopus 로고
    • Characterization of curcumin-PVP solid dispersion obtained by spray drying
    • DOI 10.1016/j.ijpharm.2003.11.014
    • A. Paradkar, A.A. Ambike, B.K. Jadhav, and K.R. Mahadik Characterization of curcumin-PVP solid dispersion obtained by spray drying Int. J. Pharm. 271 2004 281 286 (Pubitemid 38210105)
    • (2004) International Journal of Pharmaceutics , vol.271 , Issue.1-2 , pp. 281-286
    • Paradkar, A.1    Ambike, A.A.2    Jadhav, B.K.3    Mahadik, K.R.4
  • 16
    • 0018891247 scopus 로고
    • Toxicity studies on turmeric (Curcuma longa): Acute toxicity studies in rats, guinea pigs & monkeys
    • T.N. Shankar, N.V. Shantha, H.P. Ramesh, I.A. Murthy, and V.S. Murthy Toxicity studies on tumeric (Curcuma longa): acute toxicity studies in rats, guinea pigs & monkey Indian J. Exp. Biol. 18 1980 73 75 (Pubitemid 10143537)
    • (1980) Indian Journal of Experimental Biology , vol.18 , Issue.1 , pp. 73-75
    • Bhavani Shankar, T.N.1    Shantha, N.V.2    Ramesh, H.P.3
  • 17
    • 0031860081 scopus 로고    scopus 로고
    • Influence of piperine on the pharmacokinetics of curcumin in animals and human volunteers
    • DOI 10.1055/s-2006-957450
    • G. Shoba, D. Joy, T. Joseph, M. Majeed, R. Rajendran, and P.S. Srinivas Influence of piperine on the pharmacokinetics of curcumin in animals and human volunteer Planta Med. 64 1998 353 356 (Pubitemid 28234275)
    • (1998) Planta Medica , vol.64 , Issue.4 , pp. 353-356
    • Shoba, G.1    Joy, D.2    Joseph, T.3    Majeed, M.4    Rajendran, R.5    Srinivas, P.S.S.R.6
  • 18
    • 0015785965 scopus 로고
    • Pharmacology of diferuloyl methane (curcumin), a non-steroidal anti-inflammatory agent
    • R.C. Srimal, and B.N. Dhawan Pharmacology of diferuloyl methane (curcumin), a non-steroidal anti-inflammatory agent J. Pharm. Pharmacol. 25 1973 447 452
    • (1973) J. Pharm. Pharmacol. , vol.25 , pp. 447-452
    • Srimal, R.C.1    Dhawan, B.N.2
  • 20
    • 0031423468 scopus 로고    scopus 로고
    • Spectroscopic characterization of interactions between PVP and indomethacin in amorphous molecular dispersions
    • DOI 10.1023/A:1012167410376
    • L.S. Taylor, and G. Zografi Spectroscopic characterization interactions between PVP and indomethacin in amorphous molecular dispersions Pharm. Res. 14 1997 1691 1698 (Pubitemid 28062912)
    • (1997) Pharmaceutical Research , vol.14 , Issue.12 , pp. 1691-1698
    • Taylor, L.S.1    Zografi, G.2
  • 22
    • 0022066944 scopus 로고
    • Studies on curcumin and curcuminoids VI. Kinetics of curcumin degradation in aqueous solution
    • H.H. Tønnesen, and J. Karlsen Studies on curcumin and curcuminoids VI. Kinetics of curcumin degradation in aqueous solution Z. Lebensm. Unters. Forsch. 180 1985 402 404
    • (1985) Z. Lebensm. Unters. Forsch. , vol.180 , pp. 402-404
    • Tønnesen, H.H.1    Karlsen, J.2
  • 23
    • 0036917173 scopus 로고    scopus 로고
    • Solubility, chemical and photochemical stability of curcumin in surfactant solutions
    • H.H. Tønnesen Solubility, chemical and photochemical stability of curcumin in surfactant solutions. Studies of curcumin and curcuminoids VIII Pharmazie 57 2002 820 824 (Pubitemid 36014615)
    • (2002) Pharmazie , vol.57 , Issue.12 , pp. 820-824
    • Tonnesen, H.H.1
  • 24
    • 34248684129 scopus 로고    scopus 로고
    • Studies on curcumin and curcuminoids. XXXI. Symmetric and asymmetric curcuminoids: Stability, activity and complexation with cyclodextrin
    • DOI 10.1016/j.ijpharm.2007.01.013, PII S0378517307000488
    • H.H. Tønnesen, T. Loftsson, M. Masson, and M.A. Tomren Studies on curcumin and curcuminoids XXXI. Symmetric and asymmetric curcuminmoids: stability, activity and complexation with cyclodextrin Int. J. Pharm. 338 2007 27 34 (Pubitemid 46777212)
    • (2007) International Journal of Pharmaceutics , vol.338 , Issue.1-2 , pp. 27-34
    • Tomren, M.A.1    Masson, M.2    Loftsson, T.3    Tonnesen, H.H.4
  • 25
    • 84856963813 scopus 로고    scopus 로고
    • Evaluation of Inutec SP1 as a new carrier in the formulation of solid dispersions for poorly soluble drugs
    • G. Van den Mooter, I. Weuts, D.T. Ridder, and N. Blaton Evaluation of Inutec SP1 as a new carrier in the formulation of solid dispersions for poorly soluble drugs Int. J. Pharm. Sci. 26 2006 219 230
    • (2006) Int. J. Pharm. Sci. , vol.26 , pp. 219-230
    • Van Den Mooter, G.1    Weuts, I.2    Ridder, D.T.3    Blaton, N.4
  • 27
    • 0030839940 scopus 로고    scopus 로고
    • Stability of curcumin in buffer solutions and characterization of its degradation products
    • Y.J. Wang, M.H. Pan, A.L. Cheng, L.I. Lin, Y.S. Ho, C.Y. Hsieh, and J.K. Lin Stability of curcumin in buffer solutions and characterization of its degradation products Pharm. Biomed. Anal. 15 1997 1867 1876
    • (1997) Pharm. Biomed. Anal. , vol.15 , pp. 1867-1876
    • Wang, Y.J.1    Pan, M.H.2    Cheng, A.L.3    Lin, L.I.4    Ho, Y.S.5    Hsieh, C.Y.6    Lin, J.K.7


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.