메뉴 건너뛰기




Volumn 43, Issue 5, 2013, Pages 1517-1522

Hematein, a casein kinase II inhibitor, inhibits lung cancer tumor growth in a murine xenograft model

Author keywords

Casein kinase II; Hematein; Lung cancer; Wnt; Xenograft

Indexed keywords

ANTINEOPLASTIC AGENT; CASEIN KINASE II; CASEIN KINASE II ALPHA; HEMATEIN; PROTEIN KINASE B; T CELL FACTOR PROTEIN; UNCLASSIFIED DRUG; WNT PROTEIN;

EID: 84885037892     PISSN: 10196439     EISSN: 17912423     Source Type: Journal    
DOI: 10.3892/ijo.2013.2087     Document Type: Article
Times cited : (20)

References (27)
  • 1
    • 0037334895 scopus 로고    scopus 로고
    • One-thousand-and-one substrates of protein kinase ck2?
    • Meggio F and Pinna LA: One-thousand-and-one substrates of protein kinase CK2? FASEB J 17: 349-368, 2003.
    • (2003) FASEB J , vol.17 , pp. 349-368
    • Meggio, F.1    Pinna, L.A.2
  • 2
    • 0038340907 scopus 로고    scopus 로고
    • The raison d'etre of constitutively active protein kinases: The lesson of ck2
    • Pinna LA: The raison d'etre of constitutively active protein kinases: the lesson of CK2. Acc Chem Res 36: 378-384, 2003.
    • (2003) Acc Chem Res , vol.36 , pp. 378-384
    • Pinna, L.A.1
  • 4
    • 0028985936 scopus 로고
    • Casein kinase ii alpha transgene-induced murine lymphoma: Relation to theileriosis in cattle
    • Seldin DC and Leder P: Casein kinase II alpha transgene-induced murine lymphoma: relation to theileriosis in cattle. Science 267: 894-897, 1995.
    • (1995) Science , vol.267 , pp. 894-897
    • Seldin, D.C.1    Leder, P.2
  • 5
    • 0035669740 scopus 로고    scopus 로고
    • Protein kinase ck2: Signaling and tumorigenesis in the mammary gland
    • Landesman-Bollag E, Song DH, Romieu-Mourez R, et al: Protein kinase CK2: signaling and tumorigenesis in the mammary gland. Mol Cell Biochem 227: 153-165, 2001.
    • (2001) Mol Cell Biochem , vol.227 , pp. 153-165
    • Landesman-Bollag, E.1    Song, D.H.2    Romieu-Mourez, R.3
  • 6
    • 33847361829 scopus 로고    scopus 로고
    • Protein kinase ck2alpha as an unfavorable prognostic marker and novel therapeutic target in acute myeloid leukemia
    • Kim JS, Eom JI, Cheong JW, et al: Protein kinase CK2alpha as an unfavorable prognostic marker and novel therapeutic target in acute myeloid leukemia. Clin Cancer Res 13: 1019-1028, 2007.
    • (2007) Clin Cancer Res , vol.13 , pp. 1019-1028
    • Kim, J.S.1    Eom, J.I.2    Cheong, J.W.3
  • 7
    • 33847655629 scopus 로고    scopus 로고
    • Nuclear localization of protein kinase ck2 catalytic subunit (ck2alpha) is associated with poor prognostic factors in human prostate cancer
    • Laramas M, Pasquier D, Filhol O, Ringeisen F, Descotes JL and Cochet C: Nuclear localization of protein kinase CK2 catalytic subunit (CK2alpha) is associated with poor prognostic factors in human prostate cancer. Eur J Cancer 43: 928-934, 2007.
    • (2007) Eur J Cancer , vol.43 , pp. 928-934
    • Laramas, M.1    Pasquier, D.2    Filhol, O.3    Ringeisen, F.4    Descotes, J.L.5    Cochet, C.6
  • 8
    • 4444298254 scopus 로고    scopus 로고
    • Casein kinase ii alpha subunit and c1-inhibitor are independent predictors of outcome in patients with squamous cell carcinoma of the lung
    • O-charoenrat P, Rusch V, Talbot SG, et al: Casein kinase II alpha subunit and C1-inhibitor are independent predictors of outcome in patients with squamous cell carcinoma of the lung. Clin Cancer Res 10: 5792-5803, 2004.
    • (2004) Clin Cancer Res , vol.10 , pp. 5792-5803
    • O-Charoenrat, P.1    Rusch, V.2    Talbot, S.G.3
  • 9
    • 0029360679 scopus 로고
    • Association of elevated protein kinase ck2 activity with aggressive behavior of squamous cell carcinoma of the head and neck
    • Gapany M, Faust RA, Tawfic S, Davis A, Adams GL and Ahmed K: Association of elevated protein kinase CK2 activity with aggressive behavior of squamous cell carcinoma of the head and neck. Mol Med 1: 659-666, 1995.
    • (1995) Mol Med , vol.1 , pp. 659-666
    • Gapany, M.1    Faust, R.A.2    Tawfic, S.3    Davis, A.4    Adams, G.L.5    Ahmed, K.6
  • 11
    • 0037093352 scopus 로고    scopus 로고
    • Protein kinase ck2 inhibitor 4,5,6,7-tetrabromobenzotriazole (tbb) induces apoptosis and caspase-dependent degradation of haematopoietic lineage cell-specific protein 1 (hs1) in jurkat cells
    • Ruzzene M, Penzo D and Pinna LA: Protein kinase CK2 inhibitor 4,5,6,7-tetrabromobenzotriazole (TBB) induces apoptosis and caspase-dependent degradation of haematopoietic lineage cell-specific protein 1 (HS1) in Jurkat cells. Biochem J 364: 41-47, 2002.
    • (2002) Biochem J , vol.364 , pp. 41-47
    • Ruzzene, M.1    Penzo, D.2    Pinna, L.A.3
  • 12
    • 3843114402 scopus 로고    scopus 로고
    • 2-dimethylamino-4,5,6,7-tetrabromo-1h-benzimidazole: A novel powerful and selective inhibitor of protein kinase ck2
    • Pagano MA, Meggio F, Ruzzene M, Andrzejewska M, Kazimierczuk Z and Pinna LA: 2-Dimethylamino-4,5,6,7-tetrabromo-1H-benzimidazole: a novel powerful and selective inhibitor of protein kinase CK2. Biochem Biophys Res Commun 321: 1040-1044, 2004.
    • (2004) Biochem Biophys Res Commun , vol.321 , pp. 1040-1044
    • Pagano, M.A.1    Meggio, F.2    Ruzzene, M.3    Andrzejewska, M.4    Kazimierczuk, Z.5    Pinna, L.A.6
  • 13
    • 0141791013 scopus 로고    scopus 로고
    • Biochemical and three-dimensional-structural study of the specific inhibition of protein kinase ck2 by [5-oxo-5,6-dihydroindolo-(1,2-a)quinazolin- 7-yl]acetic acid (iqa)
    • Sarno S, De Moliner E, Ruzzene M, et al: Biochemical and three-dimensional-structural study of the specific inhibition of protein kinase CK2 by [5-oxo-5,6-dihydroindolo-(1,2-a)quinazolin-7-yl]acetic acid (IQA). Biochem J 374: 639-646, 2003.
    • (2003) Biochem J , vol.374 , pp. 639-646
    • Sarno, S.1    De Moliner, E.2    Ruzzene, M.3
  • 14
    • 78650321320 scopus 로고    scopus 로고
    • CX-4945, an orally bioavailable selective inhibitor of protein kinase ck2, inhibits prosurvival and angiogenic signaling and exhibits antitumor efficacy
    • Siddiqui-Jain A, Drygin D, Streiner N, et al: CX-4945, an orally bioavailable selective inhibitor of protein kinase CK2, inhibits prosurvival and angiogenic signaling and exhibits antitumor efficacy. Cancer Res 70: 10288-10298, 2010.
    • (2010) Cancer Res , vol.70 , pp. 10288-10298
    • Siddiqui-Jain, A.1    Drygin, D.2    Streiner, N.3
  • 15
    • 67649289884 scopus 로고    scopus 로고
    • Identification of hematein as a novel inhibitor of protein kinase ck2 from a natural product library
    • Hung MS, Xu Z, Lin YC, et al: Identification of hematein as a novel inhibitor of protein kinase CK2 from a natural product library. BMC Cancer 9: 135, 2009.
    • (2009) BMC Cancer , vol.9 , pp. 135
    • Hung, M.S.1    Xu, Z.2    Lin, Y.C.3
  • 16
    • 0004830588 scopus 로고    scopus 로고
    • Anticomplementary activity of constituents from the heartwood of caesalpinia sappan
    • Oh SR, Kim DS, Lee IS, Jung KY, Lee JJ and Lee HK: Anticomplementary activity of constituents from the heartwood of Caesalpinia sappan. Planta Med 64: 456-458, 1998.
    • (1998) Planta Med , vol.64 , pp. 456-458
    • Oh, S.R.1    Kim, D.S.2    Lee, I.S.3    Jung, K.Y.4    Lee, J.J.5    Lee, H.K.6
  • 17
    • 0025923682 scopus 로고
    • New investigations on hematoxylin, hematein, and hematein-aluminium complexes. II. Hematein-aluminium complexes and hemalum staining
    • Bettinger C and Zimmermann HW: New investigations on hematoxylin, hematein, and hematein-aluminium complexes. II. Hematein-aluminium complexes and hemalum staining. Histochemistry 96: 215-228, 1991.
    • (1991) Histochemistry , vol.96 , pp. 215-228
    • Bettinger, C.1    Zimmermann, H.W.2
  • 18
    • 23844444239 scopus 로고    scopus 로고
    • Hierarchical docking of databases of multiple ligand conformations
    • Lorber DM and Shoichet BK: Hierarchical docking of databases of multiple ligand conformations. Curr Top Med Chem 5: 739-749, 2005.
    • (2005) Curr Top Med Chem , vol.5 , pp. 739-749
    • Lorber, D.M.1    Shoichet, B.K.2
  • 19
    • 39149130330 scopus 로고    scopus 로고
    • The ck2 alpha/ck2 beta interface of human protein kinase ck2 harbors a binding pocket for small molecules
    • Raaf J, Brunstein E, Issinger OG and Niefind K: The CK2 alpha/CK2 beta interface of human protein kinase CK2 harbors a binding pocket for small molecules. Chem Biol 15: 111-117, 2008.
    • (2008) Chem Biol , vol.15 , pp. 111-117
    • Raaf, J.1    Brunstein, E.2    Issinger, O.G.3    Niefind, K.4
  • 20
    • 84986432941 scopus 로고
    • Automated docking with grid-based energy evaluation
    • Meng EC, Shoichet BK and Kuntz ID: Automated docking with grid-based energy evaluation. J Computat Chem 13: 505-524, 1992.
    • (1992) J Computat Chem , vol.13 , pp. 505-524
    • Meng, E.C.1    Shoichet, B.K.2    Kuntz, I.D.3
  • 21
    • 50649104594 scopus 로고    scopus 로고
    • Insights from soft x-rays: The chlorine and sulfur sub-structures of a ck2alpha/drb complex
    • Raaf J, Issinger OG and Niefind K: Insights from soft X-rays: the chlorine and sulfur sub-structures of a CK2alpha/DRB complex. Mol Cell Biochem 316: 15-23, 2008.
    • (2008) Mol Cell Biochem , vol.316 , pp. 15-23
    • Raaf, J.1    Issinger, O.G.2    Niefind, K.3
  • 22
    • 20044377997 scopus 로고    scopus 로고
    • Protein kinase ck2 phosphorylates and upregulates akt/pkb
    • Di Maira G, Salvi M, Arrigoni G, et al: Protein kinase CK2 phosphorylates and upregulates Akt/PKB. Cell Death Differ 12: 668-677, 2005.
    • (2005) Cell Death Differ , vol.12 , pp. 668-677
    • Di Maira, G.1    Salvi, M.2    Arrigoni, G.3
  • 23
    • 38349116517 scopus 로고    scopus 로고
    • Too much of a good thing: The role of protein kinase ck2 in tumorigenesis and prospects for therapeutic inhibition of ck2
    • Duncan JS and Litchfield DW: Too much of a good thing: the role of protein kinase CK2 in tumorigenesis and prospects for therapeutic inhibition of CK2. Biochim Biophys Acta 1784: 33-47, 2008.
    • (2008) Biochim Biophys Acta , vol.1784 , pp. 33-47
    • Duncan, J.S.1    Litchfield, D.W.2
  • 24
    • 34548668897 scopus 로고    scopus 로고
    • Induction of cell death in antiestrogen resistant human breast cancer cells by the protein kinase ck2 inhibitor dmat
    • Yde CW, Frogne T, Lykkesfeldt AE, Fichtner I, Issinger OG and Stenvang J: Induction of cell death in antiestrogen resistant human breast cancer cells by the protein kinase CK2 inhibitor DMAT. Cancer Lett 256: 229-237, 2007.
    • (2007) Cancer Lett , vol.256 , pp. 229-237
    • Yde, C.W.1    Frogne, T.2    Lykkesfeldt, A.E.3    Fichtner, I.4    Issinger, O.G.5    Stenvang, J.6
  • 25
    • 33750053855 scopus 로고    scopus 로고
    • Casein kinase 2 (ck2) increases survivin expression via enhanced beta-catenin-t cell factor/lymphoid enhancer binding factor-dependent transcription
    • Tapia JC, Torres VA, Rodriguez DA, Leyton L and Quest AF: Casein kinase 2 (CK2) increases survivin expression via enhanced beta-catenin-T cell factor/lymphoid enhancer binding factor-dependent transcription. Proc Natl Acad Sci USA 103: 15079-15084, 2006.
    • (2006) Proc Natl Acad Sci USA , vol.103 , pp. 15079-15084
    • Tapia, J.C.1    Torres, V.A.2    Rodriguez, D.A.3    Leyton, L.4    Quest, A.F.5
  • 26
    • 84855229785 scopus 로고    scopus 로고
    • CK2 functionally interacts with akt/pkb to promote the beta-catenin-dependent expression of survivin and enhance cell survival
    • Ponce DP, Yefi R, Cabello P, et al: CK2 functionally interacts with AKT/PKB to promote the beta-catenin-dependent expression of survivin and enhance cell survival. Mol Cell Biochem 356: 127-132, 2011.
    • (2011) Mol Cell Biochem , vol.356 , pp. 127-132
    • Ponce, D.P.1    Yefi, R.2    Cabello, P.3
  • 27
    • 84862997082 scopus 로고    scopus 로고
    • Antitumoral activity of allosteric inhibitors of protein kinase ck2
    • Moucadel V, Prudent R, Sautel CF, et al: Antitumoral activity of allosteric inhibitors of protein kinase CK2. Oncotarget 2: 997-1010, 2011.
    • (2011) Oncotarget , vol.2 , pp. 997-1010
    • Moucadel, V.1    Prudent, R.2    Sautel, C.F.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.