Preparation and evaluation of solid lipid nanoparticles based nanogel for dermal delivery of meloxicam

Chemistry and Physics of Lipids

Volumn 175-176, Issue , 2013, Pages 65-72

  Khurana, S ^a   Bedi, P M S ^a   Jain, N K ^a,b  

^a GURU NANAK DEV UNIVERSITY   (India)

^b DR H S GOUR UNIVERSITY   (India)

Author keywords

Carrageenan induced paw edema model; Controlled release; Meloxicam; Skin penetration; Solid lipid nanoparticles; Sustained release

Indexed keywords

CARRAGEENAN; MELOXICAM; SOLID LIPID NANOPARTICLE;

ANIMAL EXPERIMENT; ANIMAL TISSUE; ANTIINFLAMMATORY ACTIVITY; ARTICLE; CONTROLLED DRUG RELEASE; CONTROLLED STUDY; DIFFERENTIAL SCANNING CALORIMETRY; DRUG PENETRATION; DRUG TOLERABILITY; FLOW MEASUREMENT; FLUIDIZATION; GEL; HISTOPATHOLOGY; IN VITRO STUDY; IN VIVO STUDY; INFRARED SPECTROSCOPY; LIPID BILAYER; MOUSE; NANOEMULSION; NONHUMAN; PARTICLE SIZE; PAW EDEMA; PHOTON CORRELATION SPECTROSCOPY; PHYSICAL CHEMISTRY; PRIORITY JOURNAL; RAT; SKIN PERMEABILITY; STRATUM CORNEUM; VISCOELASTICITY;

MUS; RATTUS;

CARRAGEENAN INDUCED PAW EDEMA MODEL; CONTROLLED RELEASE; MELOXICAM; SKIN PENETRATION; SOLID LIPID NANOPARTICLES; SUSTAINED RELEASE;

ADMINISTRATION, CUTANEOUS; ANIMALS; ANTI-INFLAMMATORY AGENTS, NON-STEROIDAL; DRUG CARRIERS; EDEMA; LIPIDS; MICE; NANOPARTICLES; POLYETHYLENE GLYCOLS; POLYETHYLENEIMINE; RATS; SKIN; SKIN ABSORPTION; THIAZINES; THIAZOLES;

EID: 84883637791     PISSN: 00093084     EISSN: 18732941     Source Type: Journal    
DOI: 10.1016/j.chemphyslip.2013.07.010     Document Type: Article

References (36)

1. S.B. Abramson, and Y. Yazici Biologics in development for rheumatoid arthritis: Relevance to osteoarthritis Adv. Drug Deliv. Rev. 58 2006 212 225
2. M.A. Bolzinger, S. Briancon, J. Pelletier, and Y. Chevalier Penetration of drugs through skin, a complex rate controlling membrane Curr. Opin. Colloid Interface Sci. 17 2012 156 165
3. S. Bose, and B. Michniak-Kohn Preparation and characterization of lipid based nanosystems for topical delivery of quercetin Eur. J. Pharm. Sci. 48 2013 442 542
4. M. Bousmina Rheology of polymer blends: linear model for viscoelastic emulsions Rheol. Acta 38 1999 73 83
5. V. Chawla, and S.A. Saraf Rheological studies on solid lipid nanoparticle based carbopol gels of aceclofenac Colloids Surf. B Biointerfaces 92 2012 293 298
6. M. Cohen-Avrahami, D. Libster, A. Aserin, and N. Garti Penetratin-induced transdermal delivery from HII mesophases of sodium diclofenac J. Control. Release 159 2012 419 428
7. W. Dai, D. Zhang, C. Duan, L. Jia, Y. Wang, F. Feng, and Q. Zhang Preparation and characteristics of oridonin-loaded nanostructured lipid carriers as a controlled-release J. Microencapsul. 27 2010 234 241
8. G. Deli, S. Hatziantoniou, Y. Nikas, and C. Demetzos Solid lipid nanoparticles and nanoemulsions containing ceramides: preparation and physicochemical characterization J. Liposome. Res. 19 2009 180 188
9. T. De Vringer, and H.A.G. De Ronde Preparation and structure of a water-in-oil cream containing lipid nanoparticles J. Pharm. Sci. 84 1995 466 472
10. M. Distel, C. Mueller, E. Bluhmkij, and J. Fries Safety of meloxicam: a global analysis of clinical trials Br. J. Rheumatol. 35 1996 68 77
11. E. Esposito, L. Ravani, C. Contado, A. Costenaro, M. Drechsler, D. Rossi, E. Menegatti, A. Grandini, and R. Cortesi Clotrimazole nanoparticle gel for mucosal administration Mater. Sci. Eng. C 33 2013 411 418
12. D.E. Furst Meloxicam: selective COX-2 inhibition in clinical practice Semin. Arthritis Rheum. 126 1997 21 27 (Pubitemid 27274439)
13. N. Gerwin, C. Hops, and A. Lucke Intraarticular drug delivery in osteoarthritis B Adv. Drug Deliv. Rev. 58 2006 226 242
14. S.K. Gupta, P. Bansal, R.K. Bhardwaj, J. Jaiswal, and T. Velpandian Comparison of analgesic and anti-inflammatory activity of meloxicam gel with diclofenac and piroxicam gels in animal models: pharmacokinetic parameters after topical application Skin Pharmacol. Appl. Skin Physiol. 15 2002 105 111 (Pubitemid 34195795)
15. A. Hasanovic, R. Winkler, G.P. Resch, and C. Valenta Modification of the conformational skin structure by treatment with liposomal formulations and its correlation to the penetration depth of aciclovir Eur. J. Pharm. Biopharm. 79 2011 76 81
16. V. Jenning, A. Gysler, M. Schafer-Korting, and S.H. Gohla Vitamin A loaded solid lipid nanoparticles for topical use: occlusive properties and drug targeting to the upper skin Eur. J. Pharm. Biopharm. 49 2000 211 218 (Pubitemid 30229868)
17. K. Jores, W. Mehnert, M. Drechsler, H. Bunjes, C. Johann, and K. Mader Investigations on the structure of solid lipid nanoparticles (SLN) and oil-loaded solid lipid nanoparticles by photon correlation spectroscopy, field-flow fractionation and transmission electron microscopy J. Control. Release 95 2004 217 227 (Pubitemid 38230037)
18. S. Khurana, P.M.S. Bedi, and N.K. Jain Development of nanostructured lipid carriers (NLC) for controlled delivery of mefenamic acid Int. J. Biomed. Nanosci. Nanotechnol. 2 2012 232 250
19. S. Khurana, P.M.S. Bedi, and N.K. Jain Development of nanostructured lipid carriers (NLC) for controlled delivery of meloxicam Int. J. Biomed. Nanosci. Nanotechnol. 1 2010 247 266
20. S. Khurana, N.K. Jain, and P.M.S. Bedi Nanoemulsion based gel for transdermal delivery of meloxicam: physico-chemical, mechanistic investigation Life Sci. 92 2013 383 392
21. S.F. Lanes, L.A. Rodriguez, and G.E. Hwang Baseline risk of gastrointestinal disorders among new users of meloxicam, ibuprofen, diclofenac, naproxen and indomethacin Pharmacoepidemiol. Drug Saf. 9 2000 113 117 (Pubitemid 30307352)
22. C.H. Lee, V. Moturi, and Y. Lee Thixotropic property in pharmaceutical formulations J Control. Release 136 2009 88 98
23. S.J. Lim, and C.K. Kim Formulation parameters determining the physicochemical characteristics of solid lipid nanoparticles loaded with all-trans retinoic acid Int. J. Pharm. 243 2002 135 146
24. R.M. Martin, P. Biswas, and R.D. Mann The incidence of adverse events and risk factors for upper gastrointestinal disorders associated with meloxicam use amongst 19087 patients in general practice in England: cohort study Br. J. Clin. Pharmacol. 50 2000 35 42 (Pubitemid 30416969)
25. J.S. Negi, P. Chattopadhyay, A.K. Sharma, and V. Ram Development of solid lipid nanoparticles (SLNs) of lopinavir using hot self nano-emulsification (SNE) technique Eur. J. Pharm. Sci. 48 2013 231 239
26. K. Padois, C. Cantienic, V. Bertholle, C. Bardel, F. Pirot, and F. Falson Solid lipid nanoparticles suspension versus commercial solutions for dermal delivery of minoxidil Int. J. Pharm. 416 2011 300 304
27. L.D. Quan, G.M. Thiele, J. Tian, and D. Wang The development of novel therapies for rheumatoid arthritis Expert Opin. Ther. Pat. 18 2008 723 738
28. E.B. Souto, S.A. Wissing, C.M. Barbosa, and R.H. Muller Comparatives study between the viscoelastic behaviors of different lipid nanoparticle formulations J. Cosmet. Sci. 55 2004 463 471 (Pubitemid 39643346)
29. D.C. Swartzendruber, P.W. Wertz, K.C. Madison, and D.T. Downing Evidence that the corneocyte has a chemically bound lipid envelope J. Invest. Dermatol. 88 1987 709 713 (Pubitemid 17077741)
30. V. Teeranachaideekul, E.B. Souto, V.B. Junyaprasert, H. Rainer, and R.H. Muller Cetyl palmitate-based NLC for topical delivery of coenzyme Q10-development, physicochemical characterization and in vitro release studies Eur. J. Pharm. Biopharm. 67 2007 141 148 (Pubitemid 46991336)
31. S. Utreja, and N.K. Jain Solid lipid nanoparticles N.K. Jain, Advances in Controlled and Novel Drug Delivery 2001 CBS Publishers and Distributors New Delhi 408 425
32. S. Utreja, A.J. Khopade, and N.K. Jain Lipoprotein-mimicking biovectorized systems for methotrexate delivery Pharm. Acta Helv. 73 1999 275 279 (Pubitemid 29324992)
33. S. Wartewig, R. Neubert, W. Rettig, and K. Hesse Structure of stratum corneum lipids characterized by FT-Raman spectroscopy and DSC. IV. Mixtures of ceramides and oleic acid Chem. Phys. Lipids 91 1998 145 152 (Pubitemid 28142962)
34. L. Xu, J. Pan, Q. Chen, Q. Yu, H. Chen, H. Xu, Y. Qiu, and X. Yang In vivo evaluation of the safety of triptolide-loaded hydrogel-thickened microemulsion Food Chem. Toxicol. 46 2008 3792 3799
35. E. Zimmermann, E.B. Souto, and R.H. Muller Physicochemical investigations on the structure of drug-free and drug-loaded solid lipid nanoparticles (SLN) by means of DSC and 1H NMR Pharmazie 60 2005 508 513 (Pubitemid 41025565)
36. A. zur Muhlen, C. Schwarz, and W. Mehnert Solid lipid nanoparticles (SLN) for controlled drug delivery-drug release and release mechanism Eur. J. Pharm. Biopharm. 45 1998 149 155 (Pubitemid 28167741)