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Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 19, 2013, Pages 5279-5282

Design, synthesis and biological evaluation of peptide derivatives of l-dopa as anti-parkinsonian agents

(9) Zhou, Tao a Hider, Robert C b Jenner, Peter b Campbell, Bruce b Hobbs, Christopher J b Rose, Sarah b Jairaj, Mark b Tayarani Binazir, Kayhan A b Syme, Alexander b

a ZHEJIANG GONGSHANG UNIVERSITY (China)

b KING'S COLLEGE LONDON (United Kingdom)

Author keywords

l Dopa; Parkinson's disease 6 Hydroxydopamine (6 OHDA) lesioned rat; Prodrug

Indexed keywords

DIPEPTIDE DERIVATIVE; LEVODOPA; OXIDOPAMINE;

AREA UNDER THE CURVE; ARTICLE; BIOLOGICAL ACTIVITY; DRUG DESIGN; DRUG SCREENING; DRUG SYNTHESIS; NONHUMAN; PARKINSON DISEASE;

PARKINSONIA; RATTUS;

6-HYDROXYDOPAMINE (6-OHDA) LESIONED RAT; L-DOPA; PARKINSON'S DISEASE; PRODRUG;

ANIMALS; ANTIPARKINSON AGENTS; DIPEPTIDES; DISEASE MODELS, ANIMAL; DRUG DESIGN; LEVODOPA; MALE; MOLECULAR STRUCTURE; MOTOR ACTIVITY; PEPTIDES; RATS; RATS, WISTAR;

EID: 84883489496 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2013.08.007 Document Type: Article

Times cited : (12)

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