Histone deacetylase inhibitors down-regulate G-protein-coupled estrogen receptor and the GPER-antagonist G-15 inhibits proliferation in endometriotic cells

Fertility and Sterility

Volumn 100, Issue 3, 2013, Pages 770-776

  Imesch, Patrick ^a   Samartzis, Eleftherios P ^a   Dedes, Konstantin J ^a   Fink, Daniel ^a   Fedier, André ^a,b  

^a UNIVERSITÄTSSPITAL ZÜRICH   (Switzerland)

^b UNIVERSITY OF BASEL   (Switzerland)

Author keywords

endometriosis; estrogen receptors; G 15; GPER; histone deacetylase inhibitors

Indexed keywords

ESTROGEN RECEPTOR ALPHA; ESTROGEN RECEPTOR BETA; G PROTEIN COUPLED ESTROGEN RECEPTOR; G PROTEIN COUPLED ESTROGEN RECEPTOR ANTAGONIST G 15; G PROTEIN COUPLED RECEPTOR; PROTEIN KINASE B; RECEPTOR BLOCKING AGENT; ROMIDEPSIN; UNCLASSIFIED DRUG; VORINOSTAT;

ARTICLE; CELL ASSAY; CELL IMMORTALIZATION; CELL PROLIFERATION; CELL STIMULATION; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG EFFECT; ENDOMETRIUM CELL; ENZYME PHOSPHORYLATION; FEMALE; HISTONE ACETYLATION; HUMAN; HUMAN CELL; IN VITRO STUDY; PRIORITY JOURNAL; PROTEIN DEPHOSPHORYLATION; QUANTITATIVE ANALYSIS; REAL TIME POLYMERASE CHAIN REACTION; RECEPTOR DOWN REGULATION; UNIVERSITY HOSPITAL; WESTERN BLOTTING;

ENDOMETRIOSIS; ESTROGEN RECEPTORS; G-15; GPER; HISTONE DEACETYLASE INHIBITORS;

BENZODIOXOLES; CELL LINE, TRANSFORMED; CELL PROLIFERATION; DEPSIPEPTIDES; DOWN-REGULATION; DRUG EVALUATION, PRECLINICAL; ENDOMETRIOSIS; ENDOMETRIUM; ESTROGEN RECEPTOR ALPHA; ESTROGEN RECEPTOR BETA; FEMALE; GENE EXPRESSION REGULATION; HISTONE DEACETYLASE INHIBITORS; HUMANS; HYDROXAMIC ACIDS; QUINOLINES; RECEPTORS, ESTROGEN; RECEPTORS, G-PROTEIN-COUPLED;

EID: 84883450694     PISSN: 00150282     EISSN: 15565653     Source Type: Journal    
DOI: 10.1016/j.fertnstert.2013.05.008     Document Type: Article

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