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Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 18, 2013, Pages 5170-5173

Synthesis and evaluation of a 125I-labeled iminodihydroquinoline-derived tracer for imaging of voltage-gated sodium channels

(5) Pérez Medina, Carlos a Patel, Niral a,b Robson, Mathew c Lythgoe, Mark F b Årstad, Erik a

a UNIVERSITY COLLEGE LONDON (United Kingdom)

b UNIVERSITY COLLEGE LONDON (United Kingdom)

c UNIVERSITY COLLEGE LONDON (United Kingdom)

Author keywords

Imaging; Iodine 125; SPECT Voltage gated sodium channel; WIN17317 3

Indexed keywords

DIHYDROQUINOLINE DERIVATIVE; NEURONAL TRACT TRACER; VOLTAGE GATED SODIUM CHANNEL; IMINODIHYDROQUINOLINE; QUINOLINE DERIVATIVE; RADIOACTIVE IODINE; VOLTAGE GATED SODIUM CHANNEL BLOCKING AGENT; WIN 17317-3;

ALKYLATION; AMINO ACID SEQUENCE; ANIMAL CELL; ANIMAL TISSUE; ARTICLE; BLOOD BRAIN BARRIER; CHO CELL; DECARBOXYLATION; DRUG HALF LIFE; DRUG PROTEIN BINDING; DRUG SYNTHESIS; DRUG UPTAKE; HYDROLYSIS; ISOTOPE LABELING; NONHUMAN; PH; RADIOACTIVITY; RAT; ANIMAL; BAGG ALBINO MOUSE; CHEMICAL STRUCTURE; CHEMISTRY; CRICETULUS; DOSE RESPONSE; DRUG EFFECT; FEMALE; HUMAN; IMAGING; IODINE-125; METABOLISM; MOUSE; SINGLE PHOTON EMISSION COMPUTER TOMOGRAPHY; STRUCTURE ACTIVITY RELATION; TISSUE DISTRIBUTION; VOLTAGE-GATED SODIUM CHANNEL; WIN17317-3; CHO CELL LINE; DRUG EFFECTS;

RATTUS;

IMAGING; IODINE-125; SPECT; VOLTAGE-GATED SODIUM CHANNEL; WIN17317-3;

ANIMALS; CHO CELLS; CRICETULUS; DOSE-RESPONSE RELATIONSHIP, DRUG; FEMALE; HUMANS; IODINE RADIOISOTOPES; MICE; MICE, INBRED BALB C; MOLECULAR STRUCTURE; QUINOLINES; STRUCTURE-ACTIVITY RELATIONSHIP; TISSUE DISTRIBUTION; VOLTAGE-GATED SODIUM CHANNEL BLOCKERS; VOLTAGE-GATED SODIUM CHANNELS;

EID: 84882581961 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2013.07.014 Document Type: Article

Times cited : (7)

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